Potent and highly selective kappa opioid receptor agonists incorporating chroman- and 2,3-dihydrobenzofuran-based constraints
Chu, Guo-Hua, Gu, Minghua, Cassel, Joel A., Belanger, Serge, Graczyk, Thomas M., DeHaven, Robert N., Conway-James, Nathalie, Koblish, Mike, Little, Patrick J., DeHaven-Hudkins, Diane L., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
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General and efficient synthetic approach to novel tricyclic spiroketones
Chu, Guo-Hua, Le Bourdonnec, Bertrand, Gu, Minghua, Saeui, Christopher T., Dolle, Roland E.
Published in Tetrahedron (04.07.2009)
Published in Tetrahedron (04.07.2009)
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Journal Article
5,7-Dimethoxy-3-(4-Pyridinyl)Quinoline Is a Potent and Selective Inhibitor of Human Vascular .beta.-Type Platelet-Derived Growth Factor Receptor Tyrosine Kinase
Dolle, Roland E, Dunn, Joseph A, Bobko, Mark, Singh, Baldev, Kuster, Joan E, Baizman, Eugene, Harris, Alex L, Sawutz, David G, Miller, Deborah, Wang, Su, Faltynek, Connie R, Xie, Wen, Sarup, Jay, Bode, D. Christopher, Pagani, Edward D, Silver, Paul J
Published in Journal of medicinal chemistry (19.08.1994)
Published in Journal of medicinal chemistry (19.08.1994)
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Journal Article
Enantiospecific synthesis of (-)-tabtoxinine .beta.-lactam
Dolle, Roland E, Li, Chun Sing, Novelli, Riccardo, Kruse, Lawrence I, Eggleston, Drake
Published in Journal of organic chemistry (01.01.1992)
Published in Journal of organic chemistry (01.01.1992)
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Journal Article
Studies on the acid-catalyzed homonuclear steroidal diene isomerization
Dolle, Roland E, Schmidt, Stanley J, Eggleston, Drake, Kruse, Lawrence I
Published in Journal of organic chemistry (01.04.1988)
Published in Journal of organic chemistry (01.04.1988)
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SPIROCYCLIC HETEROCYCLIC DERIVATIVES AND METHODS OF THEIR USE
LE BOURDONNEC BERTRAND, ZHOU JEAN Q, LEISTER LARA K, DOLLE ROLAND E, AJELLO CHRISTOPHER W, CHU GUO HUA, GU MINGHUA, TUTHILL PAUL ANSON
Year of Publication 06.02.2014
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Year of Publication 06.02.2014
Patent
Synthesis of Novel Thiol-Containing Citric Acid Analogs. Kinetic Evaluation of These and Other Potential Active-Site-Directed and Mechanism-Based Inhibitors of ATP Citrate Lyase
Dolle, Roland E, Gribble, Andy, Wilkes, Tracey, Kruse, Lawrence I, Eggleston, Drake, Saxty, Barbara A, Wells, Timothy N. C, Groot, Pieter H. E
Published in Journal of medicinal chemistry (01.02.1995)
Published in Journal of medicinal chemistry (01.02.1995)
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ATP-citrate-lyase as a target for hypolipidemic intervention. Sulfoximine and 3-hydroxy-.beta.-lactam containing analogs of citric acid as potential tight-binding inhibitors
Dolle, Roland E, McNair, David, Hughes, Mark J, Kruse, Lawrence I, Eggelston, Drake, Saxty, Barbara A, Wells, Timothy N. C, Groot, Pieter H. E
Published in Journal of medicinal chemistry (01.12.1992)
Published in Journal of medicinal chemistry (01.12.1992)
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