Optimization of the in Vitro and in Vivo Properties of a Novel Series of 2,4,5-Trisubstituted Imidazoles as Potent Cholecystokinin-2 (CCK2) Antagonists
Buck, Ildiko M, Black, James W, Cooke, Tracey, Dunstone, David J, Gaffen, John D, Griffin, Eric P, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Lilley, Elliot J, Linney, Ian D, Low, Caroline M. R, McDonald, Iain M, Pether, Michael J, Roberts, Sonia P, Shankley, Nigel P, Shaxted, Mark E, Steel, Katherine I. M, Sykes, David A, Tozer, Matthew J, Watt, Gillian F, Walker, Martin K, Wright, Laurence, Wright, Paul T
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
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2,7-Dioxo-2,3,4,5,6,7-hexahydro-1H-benzo[h][1,4]diazonine as a New Template for the Design of CCK2 Receptor Antagonists
McDonald, Iain M, Dunstone, David J, Kalindjian, S. Barret, Linney, Ian D, Low, Caroline M. R, Pether, Michael J, Steel, Katherine I. M, Tozer, Matthew J, Vinter, J. G
Published in Journal of medicinal chemistry (21.09.2000)
Published in Journal of medicinal chemistry (21.09.2000)
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ω-(Imidazol-4-yl)alkane-1-sulfonamides: a new series of potent histamine H 3 receptor antagonists
Tozer, Matthew J., Buck, Ildiko M., Cooke, Tracey, Kalindjian, S.Barret, Pether, Michael J., Steel, Katherine I.M.
Published in Bioorganic & medicinal chemistry (01.02.2002)
Published in Bioorganic & medicinal chemistry (01.02.2002)
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Development of Peptide 3D Structure Mimetics: Rational Design of Novel Peptoid Cholecystokinin Receptor Antagonists
Low, Caroline M. R, Black, James W, Broughton, Howard B, Buck, Ildiko M, Davies, Jonathan M. R, Dunstone, David J, Hull, Robert A. D, Kalindjian, S. Barret, McDonald, Iain M, Pether, Michael J, Shankley, Nigel P, Steel, Katherine I. M
Published in Journal of medicinal chemistry (21.09.2000)
Published in Journal of medicinal chemistry (21.09.2000)
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4-Chlorobenzyl sulfonamide and sulfamide derivatives of histamine homologues: The design of potent histamine H 3 receptor antagonists
Tozer, Matthew J., Buck, Ildiko M., Cooke, Tracey, Kalindjian, S.Barret, McDonald, Iain M., Pether, Michael J., Steel, Katherine I.M.
Published in Bioorganic & medicinal chemistry letters (01.11.1999)
Published in Bioorganic & medicinal chemistry letters (01.11.1999)
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Non-Peptide Cholecystokinin-B/Gastrin Receptor Antagonists Based on Bicyclic, Heteroaromatic Skeletons
Kalindjian, S. Barret, Buck, Ildiko M, Davies, Jonathan M. R, Dunstone, David J, Hudson, Martin L, Low, Caroline M. R, McDonald, Iain M, Pether, Michael J, Steel, Katherine I. M, Tozer, Matthew J, Vinter, J. G
Published in Journal of medicinal chemistry (26.04.1996)
Published in Journal of medicinal chemistry (26.04.1996)
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Improving the Affinity and Selectivity of a Nonpeptide Series of Cholecystokinin-B/Gastrin Receptor Antagonists Based on the Dibenzobicyclo[2.2.2]octane Skeleton
Kalindjian, S. Barret, Buck, Ildiko M, Cushnir, Julia R, Dunstone, David J, Hudson, Martin L, Low, Caroline M. R, McDonald, Iain M, Pether, Michael J, Steel, Katherine I. M, Tozer, Matthew J
Published in Journal of medicinal chemistry (01.10.1995)
Published in Journal of medicinal chemistry (01.10.1995)
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