Effect of oral exposure to the acaricide pirimicarb, a new varroacide candidate, on Apis mellifera feeding rate
Riva, Clémence, Sokolowski, Michel BC, Normand, Julien, Santos, Jana Sopkova‐de Oliveira, Halm‐Lemeille, Marie‐Pierre
Published in Pest management science (01.08.2018)
Published in Pest management science (01.08.2018)
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Selecting the first chemical molecule inhibitor of HSP110 for colorectal cancer therapy
Gozzi, Gustavo J., Gonzalez, Daniel, Boudesco, Christophe, Dias, Alexandre M. M., Gotthard, Guillaume, Uyanik, Burhan, Dondaine, Lucile, Marcion, Guillaume, Hermetet, François, Denis, Camille, Hardy, Laurianne, Suzanne, Peggy, Douhard, Romain, Jego, Gaetan, Dubrez, Laurence, Demidov, Oleg N., Neiers, Fabrice, Briand, Loïc, Sopková-de Oliveira Santos, Jana, Voisin-Chiret, Anne-Sophie, Garrido, Carmen
Published in Cell death and differentiation (01.01.2020)
Published in Cell death and differentiation (01.01.2020)
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Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer's Disease
Toublet, François-Xavier, Lecoutey, Cédric, Lalut, Julien, Hatat, Bérénice, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopkova de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in Molecules (Basel, Switzerland) (31.07.2019)
Published in Molecules (Basel, Switzerland) (31.07.2019)
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Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5‑HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers
Dubost, Emmanuelle, Dumas, Noé, Fossey, Christine, Magnelli, Rosa, Butt-Gueulle, Sabrina, Ballandonne, Céline, Caignard, Daniel H, Dulin, Fabienne, Sopkova de-Oliveira Santos, Jana, Millet, Philippe, Charnay, Yves, Rault, Sylvain, Cailly, Thomas, Fabis, Frederic
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
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Structure-guided design of pyridoclax derivatives based on Noxa / Mcl-1 interaction mode
Hedir, Siham, De Giorgi, Marcella, Fogha, Jade, De Pascale, Martina, Weiswald, Louis-Bastien, Brotin, Emilie, Marekha, Bogdan, Denoyelle, Christophe, Denis, Camille, Suzanne, Peggy, Gautier, Fabien, Juin, Philippe, Ligat, Laetitia, Lopez, Frédéric, Carlier, Ludovic, Legay, Rémi, Bureau, Ronan, Rault, Sylvain, Poulain, Laurent, Oliveira Santos, Jana Sopková-de, Voisin-Chiret, Anne Sophie
Published in European journal of medicinal chemistry (05.11.2018)
Published in European journal of medicinal chemistry (05.11.2018)
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Synthesis of Pyridoclax Analogues: Insight into Their Druggability by Investigating Their Physicochemical Properties and Interactions with Membranes
De Pascale, Martina, Iacopetta, Domenico, Since, Marc, Corvaisier, Sophie, Vie, Véronique, Paboeuf, Gilles, Hennequin, Didier, Perato, Serge, De Giorgi, Marcella, Sinicropi, Maria Stefania, Sopkova‐De Oliveira Santos, Jana, Voisin‐Chiret, Anne‐Sophie, Malzert‐Freon, Aurélie
Published in ChemMedChem (07.01.2020)
Published in ChemMedChem (07.01.2020)
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Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation
Peauger, Ludovic, Azzouz, Rabah, Gembus, Vincent, Ţînţaş, Mihaela-Liliana, Sopková-de Oliveira Santos, Jana, Bohn, Pierre, Papamicaël, Cyril, Levacher, Vincent
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
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Benzylphenylpyrrolizinones with Anti‐amyloid and Radical Scavenging Effects, Potentially Useful in Alzheimer's Disease Treatment
Jourdan, Jean‐Pierre, Since, Marc, El Kihel, Laïla, Lecoutey, Cédric, Corvaisier, Sophie, Legay, Rémi, Sopková‐de Oliveira Santos, Jana, Cresteil, Thierry, Malzert‐Fréon, Aurélie, Rochais, Christophe, Dallemagne, Patrick
Published in ChemMedChem (21.06.2017)
Published in ChemMedChem (21.06.2017)
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Protein Crystallography under Xenon and Nitrous Oxide Pressure: Comparison with In Vivo Pharmacology Studies and Implications for the Mechanism of Inhaled Anesthetic Action
Colloc’h, Nathalie, Sopkova-de Oliveira Santos, Jana, Retailleau, Pascal, Vivarès, Denis, Bonneté, Françoise, Langlois d’Estainto, Béatrice, Gallois, Bernard, Brisson, Alain, Risso, Jean-Jacques, Lemaire, Marc, Prangé, Thierry, Abraini, Jacques H.
Published in Biophysical journal (01.01.2007)
Published in Biophysical journal (01.01.2007)
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Insights into Mcl-1 Conformational States and Allosteric Inhibition Mechanism from Molecular Dynamics Simulations, Enhanced Sampling, and Pocket Crosstalk Analysis
Benabderrahmane, Mohammed, Bureau, Ronan, Voisin-Chiret, Anne Sophie, Sopkova-de Oliveira Santos, Jana
Published in Journal of chemical information and modeling (22.06.2020)
Published in Journal of chemical information and modeling (22.06.2020)
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Novel Multitarget-Directed Ligands (MTDLs) with Acetylcholinesterase (AChE) Inhibitory and Serotonergic Subtype 4 Receptor (5-HT4R) Agonist Activities As Potential Agents against Alzheimer’s Disease: The Design of Donecopride
Rochais, Christophe, Lecoutey, Cédric, Gaven, Florence, Giannoni, Patrizia, Hamidouche, Katia, Hedou, Damien, Dubost, Emmanuelle, Genest, David, Yahiaoui, Samir, Freret, Thomas, Bouet, Valentine, Dauphin, François, Sopkova de Oliveira Santos, Jana, Ballandonne, Céline, Corvaisier, Sophie, Malzert-Fréon, Aurélie, Legay, Remi, Boulouard, Michel, Claeysen, Sylvie, Dallemagne, Patrick
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
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Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer’s disease
Toublet, François-Xavier, Lalut, Julien, Hatat, Bérénice, Lecoutey, Cédric, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopková-de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in European journal of medicinal chemistry (15.01.2021)
Published in European journal of medicinal chemistry (15.01.2021)
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Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine “bio-oxidizable” prodrugs: Synthesis, biological evaluation and structure-activity relationship
Azzouz, Rabah, Peauger, Ludovic, Gembus, Vincent, Ţînţaş, Mihaela-Liliana, Sopková-de Oliveira Santos, Jana, Papamicaël, Cyril, Levacher, Vincent
Published in European journal of medicinal chemistry (10.02.2018)
Published in European journal of medicinal chemistry (10.02.2018)
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Design, synthesis and biological evaluation of novel indano- and thiaindano-pyrazoles with potential interest for Alzheimer's disease
Genest, David, Rochais, Christophe, Lecoutey, Cédric, Oliveira Santos, Jana Sopkova-de, Ballandonne, Céline, Butt-Gueulle, Sabrina, Legay, Remi, Since, Marc, Dallemagne, Patrick
Published in MedChemComm (01.06.2013)
Published in MedChemComm (01.06.2013)
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First Synthesis of Racemic Trans Propargylamino-Donepezil, a Pleiotrope Agent Able to Both Inhibit AChE and MAO-B, with Potential Interest against Alzheimer's Disease
Guieu, Benjamin, Lecoutey, Cedric, Legay, Rémi, Davis, Audrey, Sopkova de Oliveira Santos, Jana, Altomare, Cosimo Damiano, Catto, Marco, Rochais, Christophe, Dallemagne, Patrick
Published in Molecules (Basel, Switzerland) (01.01.2021)
Published in Molecules (Basel, Switzerland) (01.01.2021)
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Discovery of Bis-Imidazoline Derivatives as New CXCR4 Ligands
Zhou, Zhicheng, Staropoli, Isabelle, Brelot, Anne, Suzanne, Peggy, Lesnard, Aurélien, Fontaine, Fanny, Perato, Serge, Rault, Sylvain, Helynck, Olivier, Arenzana-Seisdedos, Fernando, Sopkova-de Oliveira Santos, Jana, Lagane, Bernard, Munier-Lehmann, Hélène, Colin, Philippe
Published in Molecules (Basel, Switzerland) (24.01.2023)
Published in Molecules (Basel, Switzerland) (24.01.2023)
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Three-dimensional model of the human urotensin-II receptor: Docking of human urotensin-II and nonpeptide antagonists in the binding site and comparison with an antagonist pharmacophore model
Lescot, Elodie, Sopkova-de Oliveira Santos, Jana, Colloc'h, Nathalie, Rodrigo, Jordi, Milazzo-Segalas, Isabelle, Bureau, Ronan, Rault, Sylvain
Published in Proteins, structure, function, and bioinformatics (01.10.2008)
Published in Proteins, structure, function, and bioinformatics (01.10.2008)
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Drug Repurposing: Deferasirox Inhibits the Anti-Apoptotic Activity of Mcl-1
Bourafai-Aziez, Asma, Benabderrahmane, Mohammed, Paysant, Hippolyte, Weiswald, Louis-Bastien, Poulain, Laurent, Carlier, Ludovic, Ravault, Delphine, Jouanne, Marie, Coadou, Gaël, Oulyadi, Hassan, Voisin-Chiret, Anne-Sophie, Sopková-de Oliveira Santos, Jana, Sebban, Muriel
Published in Drug design, development and therapy (01.01.2021)
Published in Drug design, development and therapy (01.01.2021)
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Definition of New Pharmacophores for Nonpeptide Antagonists of Human Urotensin-II. Comparison with the 3D-structure of Human Urotensin-II and URP
Lescot, Elodie, Sopkova-de Oliveira Santos, Jana, Dubessy, Christophe, Oulyadi, Hassan, Lesnard, Aurélien, Vaudry, Hubert, Bureau, Ronan, Rault, Sylvain
Published in Journal of chemical information and modeling (01.03.2007)
Published in Journal of chemical information and modeling (01.03.2007)
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