Chemical Genetic Analysis and Functional Characterization of Staphylococcal Wall Teichoic Acid 2-Epimerases Reveals Unconventional Antibiotic Drug Targets
Mann, Paul A, Müller, Anna, Wolff, Kerstin A, Fischmann, Thierry, Wang, Hao, Reed, Patricia, Hou, Yan, Li, Wenjin, Müller, Christa E, Xiao, Jianying, Murgolo, Nicholas, Sher, Xinwei, Mayhood, Todd, Sheth, Payal R, Mirza, Asra, Labroli, Marc, Xiao, Li, McCoy, Mark, Gill, Charles J, Pinho, Mariana G, Schneider, Tanja, Roemer, Terry
Published in PLoS pathogens (01.05.2016)
Published in PLoS pathogens (01.05.2016)
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Journal Article
Impact of Antifungal Prophylaxis on Colonization and Azole Susceptibility of Candida Species
MANN, Paul A, MCNICHOLAS, Paul M, CHAU, Andrew S, PATEL, Reena, MENDRICK, Cara, ULLMANN, Andrew J, CORNELY, Oliver A, PATINO, Hernando, BLACK, Todd A
Published in Antimicrobial Agents and Chemotherapy (01.12.2009)
Published in Antimicrobial Agents and Chemotherapy (01.12.2009)
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Chemical Genomics-Based Antifungal Drug Discovery: Targeting Glycosylphosphatidylinositol (GPI) Precursor Biosynthesis
Mann, Paul A, McLellan, Catherine A, Koseoglu, Sandra, Si, Qian, Kuzmin, Elena, Flattery, Amy, Harris, Guy, Sher, Xinwei, Murgolo, Nicholas, Wang, Hao, Devito, Kristine, de Pedro, Nuria, Genilloud, Olga, Kahn, Jennifer Nielsen, Jiang, Bo, Costanzo, Michael, Boone, Charlie, Garlisi, Charles G, Lindquist, Susan, Roemer, Terry
Published in ACS infectious diseases (09.01.2015)
Published in ACS infectious diseases (09.01.2015)
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Journal Article
Multiple Resistance Mechanisms among Aspergillus fumigatus Mutants with High-Level Resistance to Itraconazole
NASCIMENTO, Adriana M, GOLDMAN, Gustavo H, PARK, Steven, MAMAS, Salvatore A. E, DELMAS, Guillaume, OZA, Uma, LOLANS, Karen, DUDLEY, Michael N, MANN, Paul A, PERLIN, David S
Published in Antimicrobial Agents and Chemotherapy (01.05.2003)
Published in Antimicrobial Agents and Chemotherapy (01.05.2003)
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Journal Article
Mapping and characterization of vicriviroc resistance mutations from HIV-1 isolated from treatment-experienced subjects enrolled in a phase II study (VICTOR-E1)
McNicholas, Paul M, Mann, Paul A, Wojcik, Lisa, Qiu, Ping, Lee, Erin, McCarthy, Michael, Shen, Junwu, Black, Todd A, Strizki, Julie M
Published in Journal of acquired immune deficiency syndromes (1999) (01.03.2011)
Published in Journal of acquired immune deficiency syndromes (1999) (01.03.2011)
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Mutations in Aspergillus fumigatus Resulting in Reduced Susceptibility to Posaconazole Appear To Be Restricted to a Single Amino Acid in the Cytochrome P450 14α-Demethylase
MANN, Paul A, PARMEGIANI, Raulo M, WEI, Shui-Qing, MENDRICK, Cara A, XIN LI, LOEBENBERG, David, DIDOMENICO, Beth, HARE, Roberta S, WALKER, Scott S, MCNICHOLAS, Paul M
Published in Antimicrobial Agents and Chemotherapy (01.02.2003)
Published in Antimicrobial Agents and Chemotherapy (01.02.2003)
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Journal Article
Posaconazole Is a Potent Inhibitor of Sterol 14α-Demethylation in Yeasts and Molds
Munayyer, Hanan K, Mann, Paul A, Chau, Andrew S, Yarosh-Tomaine, Taisa, Greene, Jonathan R, Hare, Roberta S, Heimark, Larry, Palermo, Robert E, Loebenberg, David, McNicholas, Paul M
Published in Antimicrobial Agents and Chemotherapy (01.10.2004)
Published in Antimicrobial Agents and Chemotherapy (01.10.2004)
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Journal Article
Dual-Targeting Small-Molecule Inhibitors of the Staphylococcus aureus FMN Riboswitch Disrupt Riboflavin Homeostasis in an Infectious Setting
Wang, Hao, Mann, Paul A., Xiao, Li, Gill, Charles, Galgoci, Andrew M., Howe, John A., Villafania, Artjohn, Barbieri, Christopher M., Malinverni, Juliana C., Sher, Xinwei, Mayhood, Todd, McCurry, Megan D., Murgolo, Nicholas, Flattery, Amy, Mack, Matthias, Roemer, Terry
Published in Cell chemical biology (18.05.2017)
Published in Cell chemical biology (18.05.2017)
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Journal Article
Evernimicin Binds Exclusively to the 50S Ribosomal Subunit and Inhibits Translation in Cell-Free Systems Derived from both Gram-Positive and Gram-Negative Bacteria
MCNICHOLAS, P. M, NAJARIAN, D. J, MANN, P. A, HESK, D, HARE, R. S, SHAW, K. J, BLACK, T. A
Published in Antimicrobial Agents and Chemotherapy (01.05.2000)
Published in Antimicrobial Agents and Chemotherapy (01.05.2000)
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Journal Article
Murgocil is a Highly Bioactive Staphylococcal-Specific Inhibitor of the Peptidoglycan Glycosyltransferase Enzyme MurG
Mann, Paul A, Müller, Anna, Xiao, Li, Pereira, Pedro M, Yang, Christine, Ho Lee, Sang, Wang, Hao, Trzeciak, Joanna, Schneeweis, Jonathan, dos Santos, Margarida Moreira, Murgolo, Nicholas, She, Xinwei, Gill, Charles, Balibar, Carl J, Labroli, Marc, Su, Jing, Flattery, Amy, Sherborne, Brad, Maier, Richard, Tan, Christopher M, Black, Todd, Önder, Kamil, Kargman, Stacia, Monsma, Frederick J, Pinho, Mariana G, Schneider, Tanja, Roemer, Terry
Published in ACS chemical biology (15.11.2013)
Published in ACS chemical biology (15.11.2013)
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Cerastecins inhibit membrane lipooligosaccharide transport in drug-resistant Acinetobacter baumannii
Wang, Hao, Ishchenko, Andrii, Skudlarek, Jason, Shen, Pamela, Dzhekieva, Liudmila, Painter, Ronald E., Chen, Yun-Ting, Bukhtiyarova, Marina, Leithead, Andrew, Tracy, Rodger, Babaoglu, Kerim, Bahnck-Teets, Carolyn, Buevich, Alexei, Cabalu, Tamara D., Labroli, Marc, Lange, Henry, Lei, Ying, Li, Wei, Liu, Jian, Mann, Paul A., Meng, Tao, Mitchell, Helen J., Mulhearn, James, Scapin, Giovanna, Sha, Deyou, Shaw, Anthony W., Si, Qian, Tong, Ling, Wu, Chengwei, Wu, Zhe, Xiao, Jing Chen, Xu, Min, Zhang, Li-Kang, McKenney, David, Miller, Randy R., Black, Todd A., Cooke, Andrew, Balibar, Carl J., Klein, Daniel J., Raheem, Izzat, Walker, Scott S.
Published in Nature microbiology (01.05.2024)
Published in Nature microbiology (01.05.2024)
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Journal Article
EmtA, a rRNA methyltransferase conferring high‐level evernimicin resistance
Mann, Paul A., Xiong, Liqun, Mankin, Alexander S., Chau, Andrew S., Mendrick, Cara A., Najarian, David J., Cramer, Christina A., Loebenberg, David, Coates, Elizabeth, Murgolo, Nicholas J., Aarestrup, Frank M., Goering, Richard V., Black, Todd A., Hare, Roberta S., McNicholas, Paul M.
Published in Molecular microbiology (01.09.2001)
Published in Molecular microbiology (01.09.2001)
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