A Charge‐Switchable Zwitterionic Peptide for Rapid Detection of SARS‐CoV‐2 Main Protease
Jin, Zhicheng, Mantri, Yash, Retout, Maurice, Cheng, Yong, Zhou, Jiajing, Jorns, Alec, Fajtova, Pavla, Yim, Wonjun, Moore, Colman, Xu, Ming, Creyer, Matthew N., Borum, Raina M., Zhou, Jingcheng, Wu, Zhuohong, He, Tengyu, Penny, William F., O'Donoghue, Anthony J., Jokerst, Jesse V.
Published in Angewandte Chemie International Edition (21.02.2022)
Published in Angewandte Chemie International Edition (21.02.2022)
Get full text
Journal Article
Cathepsin B in neurodegeneration of Alzheimer's disease, traumatic brain injury, and related brain disorders
Hook, Vivian, Yoon, Michael, Mosier, Charles, Ito, Gen, Podvin, Sonia, Head, Brian P., Rissman, Robert, O'Donoghue, Anthony J., Hook, Gregory
Published in Biochimica et biophysica acta. Proteins and proteomics (01.08.2020)
Published in Biochimica et biophysica acta. Proteins and proteomics (01.08.2020)
Get full text
Journal Article
Structure- and function-based design of Plasmodium-selective proteasome inhibitors
Li, Hao, O’Donoghue, Anthony J., van der Linden, Wouter A., Xie, Stanley C., Yoo, Euna, Foe, Ian T., Tilley, Leann, Craik, Charles S., da Fonseca, Paula C. A., Bogyo, Matthew
Published in Nature (London) (11.02.2016)
Published in Nature (London) (11.02.2016)
Get full text
Journal Article
A Clinical-Stage Cysteine Protease Inhibitor blocks SARS-CoV‑2 Infection of Human and Monkey Cells
Mellott, Drake M, Tseng, Chien-Te, Drelich, Aleksandra, Fajtová, Pavla, Chenna, Bala C, Kostomiris, Demetrios H, Hsu, Jason, Zhu, Jiyun, Taylor, Zane W, Kocurek, Klaudia I, Tat, Vivian, Katzfuss, Ardala, Li, Linfeng, Giardini, Miriam A, Skinner, Danielle, Hirata, Ken, Yoon, Michael C, Beck, Sungjun, Carlin, Aaron F, Clark, Alex E, Beretta, Laura, Maneval, Daniel, Hook, Vivian, Frueh, Felix, Hurst, Brett L, Wang, Hong, Raushel, Frank M, O’Donoghue, Anthony J, de Siqueira-Neto, Jair Lage, Meek, Thomas D, McKerrow, James H
Published in ACS chemical biology (16.04.2021)
Published in ACS chemical biology (16.04.2021)
Get full text
Journal Article
Selective Neutral pH Inhibitor of Cathepsin B Designed Based on Cleavage Preferences at Cytosolic and Lysosomal pH Conditions
Yoon, Michael C, Solania, Angelo, Jiang, Zhenze, Christy, Mitchell P, Podvin, Sonia, Mosier, Charles, Lietz, Christopher B, Ito, Gen, Gerwick, William H, Wolan, Dennis W, Hook, Gregory, O’Donoghue, Anthony J, Hook, Vivian
Published in ACS chemical biology (17.09.2021)
Published in ACS chemical biology (17.09.2021)
Get full text
Journal Article
Development of a Potent Inhibitor of the Plasmodium Proteasome with Reduced Mammalian Toxicity
LaMonte, Gregory M, Almaliti, Jehad, Bibo-Verdugo, Betsaida, Keller, Lena, Zou, Bing Yu, Yang, Jennifer, Antonova-Koch, Yevgeniya, Orjuela-Sanchez, Pamela, Boyle, Colleen A, Vigil, Edgar, Wang, Lawrence, Goldgof, Gregory M, Gerwick, Lena, O’Donoghue, Anthony J, Winzeler, Elizabeth A, Gerwick, William H, Ottilie, Sabine
Published in Journal of medicinal chemistry (10.08.2017)
Published in Journal of medicinal chemistry (10.08.2017)
Get full text
Journal Article
Skin Commensal Malassezia globosa Secreted Protease Attenuates Staphylococcus aureus Biofilm Formation
Li, Hao, Goh, Bee Na, Teh, Wooi Keong, Jiang, Zhenze, Goh, Joleen Pei Zhen, Goh, Amelia, Wu, Guangxi, Hoon, Shawn S., Raida, Manfred, Camattari, Andrea, Yang, Liang, O’Donoghue, Anthony J., Dawson, Thomas L.
Published in Journal of investigative dermatology (01.05.2018)
Published in Journal of investigative dermatology (01.05.2018)
Get full text
Journal Article
A Dual‐Color Fluorescent Probe Allows Simultaneous Imaging of Main and Papain‐like Proteases of SARS‐CoV‐2‐Infected Cells for Accurate Detection and Rapid Inhibitor Screening
Cheng, Yong, Borum, Raina M., Clark, Alex E., Jin, Zhicheng, Moore, Colman, Fajtová, Pavla, O'Donoghue, Anthony J., Carlin, Aaron F., Jokerst, Jesse V.
Published in Angewandte Chemie International Edition (21.02.2022)
Published in Angewandte Chemie International Edition (21.02.2022)
Get full text
Journal Article
Chemoproteomic identification of a DPP4 homolog in Bacteroides thetaiotaomicron
Keller, Laura J., Nguyen, Taylor H., Liu, Lawrence J., Hurysz, Brianna M., Lakemeyer, Markus, Guerra, Matteo, Gelsinger, Danielle J., Chanin, Rachael, Ngo, Nhi, Lum, Kenneth M., Faucher, Franco, Ipock, Phillip, Niphakis, Micah J., Bhatt, Ami S., O’Donoghue, Anthony J., Huang, Kerwyn Casey, Bogyo, Matthew
Published in Nature chemical biology (01.12.2023)
Published in Nature chemical biology (01.12.2023)
Get full text
Journal Article
Global substrate profiling of proteases in human neutrophil extracellular traps reveals consensus motif predominantly contributed by elastase
O'Donoghue, Anthony J, Jin, Ye, Knudsen, Giselle M, Perera, Natascha C, Jenne, Dieter E, Murphy, John E, Craik, Charles S, Hermiston, Terry W
Published in PloS one (20.09.2013)
Published in PloS one (20.09.2013)
Get full text
Journal Article
Structural elucidation of recombinant Trichomonas vaginalis 20S proteasome bound to covalent inhibitors
Silhan, Jan, Fajtova, Pavla, Bartosova, Jitka, Hurysz, Brianna M., Almaliti, Jehad, Miyamoto, Yukiko, Eckmann, Lars, Gerwick, William H., O’Donoghue, Anthony J., Boura, Evzen
Published in Nature communications (04.10.2024)
Published in Nature communications (04.10.2024)
Get full text
Journal Article
A novel class of TMPRSS2 inhibitors potently block SARS-CoV-2 and MERS-CoV viral entry and protect human epithelial lung cells
Mahoney, Matthew, Damalanka, Vishnu C, Tartell, Michael A, Chung, Dong Hee, Lourenço, André Luiz, Pwee, Dustin, Mayer Bridwell, Anne E, Hoffmann, Markus, Voss, Jorine, Karmakar, Partha, Azouz, Nurit P, Klingler, Andrea M, Rothlauf, Paul W, Thompson, Cassandra E, Lee, Melody, Klampfer, Lidija, Stallings, Christina L, Rothenberg, Marc E, Pöhlmann, Stefan, Whelan, Sean P J, O'Donoghue, Anthony J, Craik, Charles S, Janetka, James W
Published in Proceedings of the National Academy of Sciences - PNAS (26.10.2021)
Published in Proceedings of the National Academy of Sciences - PNAS (26.10.2021)
Get full text
Journal Article
Potent Anti-SARS-CoV‑2 Activity by the Natural Product Gallinamide A and Analogues via Inhibition of Cathepsin L
Ashhurst, Anneliese S., Tang, Arthur H., Fajtová, Pavla, Yoon, Michael C., Aggarwal, Anupriya, Bedding, Max J., Stoye, Alexander, Beretta, Laura, Pwee, Dustin, Drelich, Aleksandra, Skinner, Danielle, Li, Linfeng, Meek, Thomas D., McKerrow, James H., Hook, Vivian, Tseng, Chien-Te, Larance, Mark, Turville, Stuart, Gerwick, William H., O’Donoghue, Anthony J., Payne, Richard J.
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
Get full text
Journal Article
Protease-Responsive Peptide-Conjugated Mitochondrial-Targeting AIEgens for Selective Imaging and Inhibition of SARS-CoV-2-Infected Cells
Cheng, Yong, Clark, Alex E., Zhou, Jiajing, He, Tengyu, Li, Yi, Borum, Raina M., Creyer, Matthew N., Xu, Ming, Jin, Zhicheng, Zhou, Jingcheng, Yim, Wonjun, Wu, Zhuohong, Fajtová, Pavla, O’Donoghue, Anthony J., Carlin, Aaron F., Jokerst, Jesse V.
Published in ACS nano (23.08.2022)
Published in ACS nano (23.08.2022)
Get full text
Journal Article
Tutuilamides A–C: Vinyl-Chloride-Containing Cyclodepsipeptides from Marine Cyanobacteria with Potent Elastase Inhibitory Properties
Keller, Lena, Canuto, Kirley Marques, Liu, Chenxi, Suzuki, Brian M, Almaliti, Jehad, Sikandar, Asfandyar, Naman, C. Benjamin, Glukhov, Evgenia, Luo, Danmeng, Duggan, Brendan M, Luesch, Hendrik, Koehnke, Jesko, O’Donoghue, Anthony J, Gerwick, William H
Published in ACS chemical biology (20.03.2020)
Published in ACS chemical biology (20.03.2020)
Get full text
Journal Article
Peptide Amphiphile Mediated Co‐assembly for Nanoplasmonic Sensing
Jin, Zhicheng, Li, Yi, Li, Ke, Zhou, Jiajing, Yeung, Justin, Ling, Chuxuan, Yim, Wonjun, He, Tengyu, Cheng, Yong, Xu, Ming, Creyer, Matthew N., Chang, Yu‐Ci, Fajtová, Pavla, Retout, Maurice, Qi, Baiyan, Li, Shuzhou, O'Donoghue, Anthony J., Jokerst, Jesse V.
Published in Angewandte Chemie International Edition (23.01.2023)
Published in Angewandte Chemie International Edition (23.01.2023)
Get full text
Journal Article
Global landscape of HIV–human protein complexes
Jäger, Stefanie, Cimermancic, Peter, Gulbahce, Natali, Johnson, Jeffrey R., McGovern, Kathryn E., Clarke, Starlynn C., Shales, Michael, Mercenne, Gaelle, Pache, Lars, Li, Kathy, Hernandez, Hilda, Jang, Gwendolyn M., Roth, Shoshannah L., Akiva, Eyal, Marlett, John, Stephens, Melanie, D’Orso, Iván, Fernandes, Jason, Fahey, Marie, Mahon, Cathal, O’Donoghue, Anthony J., Todorovic, Aleksandar, Morris, John H., Maltby, David A., Alber, Tom, Cagney, Gerard, Bushman, Frederic D., Young, John A., Chanda, Sumit K., Sundquist, Wesley I., Kortemme, Tanja, Hernandez, Ryan D., Craik, Charles S., Burlingame, Alma, Sali, Andrej, Frankel, Alan D., Krogan, Nevan J.
Published in Nature (London) (19.01.2012)
Published in Nature (London) (19.01.2012)
Get full text
Journal Article
Spacer Matters: All-Peptide-Based Ligand for Promoting Interfacial Proteolysis and Plasmonic Coupling
Jin, Zhicheng, Ling, Chuxuan, Li, Yi, Zhou, Jiajing, Li, Ke, Yim, Wonjun, Yeung, Justin, Chang, Yu-Ci, He, Tengyu, Cheng, Yong, Fajtová, Pavla, Retout, Maurice, O’Donoghue, Anthony J, Jokerst, Jesse V.
Published in Nano letters (23.11.2022)
Published in Nano letters (23.11.2022)
Get full text
Journal Article
Dysregulation of Exosome Cargo by Mutant Tau Expressed in Human-induced Pluripotent Stem Cell (iPSC) Neurons Revealed by Proteomics Analyses
Podvin, Sonia, Jones, Alexander, Liu, Qing, Aulston, Brent, Ransom, Linnea, Ames, Janneca, Shen, Gloria, Lietz, Christopher B., Jiang, Zhenze, O'Donoghue, Anthony J., Winston, Charisse, Ikezu, Tsuneya, Rissman, Robert A., Yuan, Shauna, Hook, Vivian
Published in Molecular & cellular proteomics (01.06.2020)
Published in Molecular & cellular proteomics (01.06.2020)
Get full text
Journal Article
Multiplex substrate profiling by mass spectrometry for proteases
Rohweder, Peter J, Jiang, Zhenze, Hurysz, Brianna M, O'Donoghue, Anthony J, Craik, Charles S
Published in Methods in enzymology (01.01.2023)
Published in Methods in enzymology (01.01.2023)
Get more information
Journal Article