An allosteric modulator of alpha7 nicotinic receptors, N-(5-Chloro-2,4-dimethoxyphenyl)-N'-(5-methyl-3-isoxazolyl)-urea (PNU-120596), causes conformational changes in the extracellular ligand binding domain similar to those caused by acetylcholine
Barron, Sean C, McLaughlin, James T, See, Jennifer A, Richards, Vanessa L, Rosenberg, Robert L
Published in Molecular pharmacology (01.08.2009)
Published in Molecular pharmacology (01.08.2009)
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