Advances in high‐throughput mass spectrometry in drug discovery
Dueñas, Maria Emilia, Peltier‐Heap, Rachel E, Leveridge, Melanie, Annan, Roland S, Büttner, Frank H, Trost, Matthias
Published in EMBO molecular medicine (11.01.2023)
Published in EMBO molecular medicine (11.01.2023)
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Journal Article
A high-throughput MALDI-TOF MS biochemical screen for small molecule inhibitors of the antigen aminopeptidase ERAP1
Müller, Leonie, Burton, Amy K, Tayler, Chloe L, Rowedder, James E, Hutchinson, Jonathan P, Peace, Simon, Quayle, Julie M, Leveridge, Melanie V, Annan, Roland S, Trost, Matthias, Peltier-Heap, Rachel E, Dueñas, Maria Emilia
Published in SLAS discovery (01.01.2023)
Published in SLAS discovery (01.01.2023)
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Journal Article
Identifying Inhibitors of Inflammation: A Novel High-Throughput MALDI-TOF Screening Assay for Salt-Inducible Kinases (SIKs)
Heap, Rachel E., Hope, Anthony G., Pearson, Lesley-Anne, Reyskens, Kathleen M. S. E., McElroy, Stuart P., Hastie, C. James, Porter, David W., Arthur, J. Simon C., Gray, David W., Trost, Matthias
Published in SLAS discovery (01.12.2017)
Published in SLAS discovery (01.12.2017)
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Journal Article
A MALDI-TOF assay identifies nilotinib as an inhibitor of inflammation in acute myeloid leukaemia
Marin-Rubio, José Luis, Heap, Rachel E, Heunis, Tiaan, Dueñas, Maria Emilia, Inns, Joseph, Scott, Jonathan, Simpson, A John, James Mark Allan, Blair, Helen, Heidenreich, Olaf, Saxty, Barbara, Trost, Matthias
Published in bioRxiv (29.03.2022)
Published in bioRxiv (29.03.2022)
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