Double Strain-Promoted Macrocyclization for the Rapid Selection of Cell-Active Stapled Peptides
Lau, Yu Heng, Wu, Yuteng, Rossmann, Maxim, Tan, Ban Xiong, de Andrade, Peterson, Tan, Yaw Sing, Verma, Chandra, McKenzie, Grahame J., Venkitaraman, Ashok R., Hyvönen, Marko, Spring, David R.
Published in Angewandte Chemie (International ed.) (14.12.2015)
Published in Angewandte Chemie (International ed.) (14.12.2015)
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Journal Article
Development of Cell‐Permeable, Non‐Helical Constrained Peptides to Target a Key Protein–Protein Interaction in Ovarian Cancer
Wiedmann, Mareike M., Tan, Yaw Sing, Wu, Yuteng, Aibara, Shintaro, Xu, Wenshu, Sore, Hannah F., Verma, Chandra S., Itzhaki, Laura, Stewart, Murray, Brenton, James D., Spring, David R.
Published in Angewandte Chemie International Edition (09.01.2017)
Published in Angewandte Chemie International Edition (09.01.2017)
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Journal Article
A strategy for the diversity-oriented synthesis of macrocyclic scaffolds using multidimensional coupling
Beckmann, Henning S. G., Nie, Feilin, Hagerman, Caroline E., Johansson, Henrik, Tan, Yaw Sing, Wilcke, David, Spring, David R.
Published in Nature chemistry (01.10.2013)
Published in Nature chemistry (01.10.2013)
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Journal Article
Targeted covalent inhibitors of MDM2 using electrophile-bearing stapled peptides
Charoenpattarapreeda, Jiraborrirak, Tan, Yaw Sing, Iegre, Jessica, Walsh, Stephen J, Fowler, Elaine, Eapen, Rohan S, Wu, Yuteng, Sore, Hannah F, Verma, Chandra S, Itzhaki, Laura, Spring, David R
Published in Chemical communications (Cambridge, England) (14.07.2019)
Published in Chemical communications (Cambridge, England) (14.07.2019)
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Journal Article
The Use of Chlorobenzene as a Probe Molecule in Molecular Dynamics Simulations
Tan, Yaw Sing, Spring, David R, Abell, Chris, Verma, Chandra
Published in Journal of chemical information and modeling (28.07.2014)
Published in Journal of chemical information and modeling (28.07.2014)
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Journal Article
Incorporation of Putative Helix-Breaking Amino Acids in the Design of Novel Stapled Peptides: Exploring Biophysical and Cellular Permeability Properties
Partridge, Anthony W, Kaan, Hung Yi Kristal, Juang, Yu-Chi, Sadruddin, Ahmad, Lim, Shuhui, Brown, Christopher J, Ng, Simon, Thean, Dawn, Ferrer, Fernando, Johannes, Charles, Yuen, Tsz Ying, Kannan, Srinivasaraghavan, Aronica, Pietro, Tan, Yaw Sing, Pradhan, Mohan R, Verma, Chandra S, Hochman, Jerome, Chen, Shiying, Wan, Hui, Ha, Sookhee, Sherborne, Brad, Lane, David P, Sawyer, Tomi K
Published in Molecules (Basel, Switzerland) (20.06.2019)
Published in Molecules (Basel, Switzerland) (20.06.2019)
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Journal Article
Stereoisomerism of stapled peptide inhibitors of the p53-Mdm2 interaction: an assessment of synthetic strategies and activity profiles
Yuen, Tsz Ying, Brown, Christopher J, Xue, Yuezhen, Tan, Yaw Sing, Ferrer Gago, Fernando J, Lee, Xue Er, Neo, Jin Yong, Thean, Dawn, Kaan, Hung Yi Kristal, Partridge, Anthony W, Verma, Chandra S, Lane, David P, Johannes, Charles W
Published in Chemical science (Cambridge) (14.07.2019)
Published in Chemical science (Cambridge) (14.07.2019)
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Journal Article
Inhibiting S100B(ββ) for Activating Wild-Type p53: Design of Stapled Peptides
Kannan, Srinivasaraghavan, Aronica, Pietro G. A, Tan, Yaw Sing, Verma, Chandra S
Published in ACS omega (31.03.2019)
Published in ACS omega (31.03.2019)
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Journal Article
Using Ligand-Mapping Simulations to Design a Ligand Selectively Targeting a Cryptic Surface Pocket of Polo-Like Kinase 1
Tan, Yaw Sing, Śledź, Paweł, Lang, Steffen, Stubbs, Christopher J., Spring, David R., Abell, Chris, Best, Robert B.
Published in Angewandte Chemie (International ed.) (01.10.2012)
Published in Angewandte Chemie (International ed.) (01.10.2012)
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Journal Article
Macrocyclized Extended Peptides: Inhibiting the Substrate-Recognition Domain of Tankyrase
Xu, Wenshu, Lau, Yu Heng, Fischer, Gerhard, Tan, Yaw Sing, Chattopadhyay, Anasuya, de la Roche, Marc, Hyvönen, Marko, Verma, Chandra, Spring, David R, Itzhaki, Laura S
Published in Journal of the American Chemical Society (15.02.2017)
Published in Journal of the American Chemical Society (15.02.2017)
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Journal Article
Ultralong recovery time in nanosecond electroporation systems enabled by orientational-disordering processes
Lee, Denise, Naikar, J Shamita, Chan, Sophia S. Y, Meivita, Maria Prisca, Li, Lunna, Tan, Yaw Sing, Bajalovic, Natasa, Loke, Desmond K
Published in Nanoscale (01.06.2022)
Published in Nanoscale (01.06.2022)
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Journal Article
Efficient development of stable and highly functionalised peptides targeting the CK2α/CK2β protein-protein interaction
Iegre, Jessica, Brear, Paul, Baker, David J, Tan, Yaw Sing, Atkinson, Eleanor L, Sore, Hannah F, O' Donovan, Daniel H, Verma, Chandra S, Hyvönen, Marko, Spring, David R
Published in Chemical science (Cambridge) (21.05.2019)
Published in Chemical science (Cambridge) (21.05.2019)
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Journal Article
Macrocyclization of an all-d linear alpha-helical peptide imparts cellular permeability
Kannan, Srinivasaraghavan, Aronica, Pietro G. A., Ng, Simon, Lian, Dawn Thean Gek, Frosi, Yuri, Chee, Sharon, Jiang, Shimin, Yuen, Tsz Ying, Sadruddin, Ahmad, Kaan, Hung Yi Kristal, Chandramohan, Arun, Wong, Jin Huei, Tan, Yaw Sing, Chang, Zi Wei, Ferrer-Gago, Fernando J., Arumugam, Prakash, Han, Yi, Chen, Shiying, Renia, Laurent, Brown, Christopher J., Johannes, Charles W., Henry, Brian, Lane, David P., Sawyer, Tomi K., Verma, Chandra S., Partridge, Anthony W.
Published in Chemical science (Cambridge) (07.06.2020)
Published in Chemical science (Cambridge) (07.06.2020)
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Journal Article
Stapled peptides as a new technology to investigate protein-protein interactions in human platelets
Iegre, Jessica, Ahmed, Niaz S., Gaynord, Josephine S., Wu, Yuteng, Herlihy, Kara M., Tan, Yaw Sing, Lopes-Pires, Maria E., Jha, Rupam, Lau, Yu Heng, Sore, Hannah F., Verma, Chandra, O'Donovan, Daniel H., Pugh, Nicholas, Spring, David R.
Published in Chemical science (Cambridge) (28.05.2018)
Published in Chemical science (Cambridge) (28.05.2018)
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Journal Article