Discovery and optimization of 2-pyridinone aminal integrase strand transfer inhibitors for the treatment of HIV
Schreier, John D., Embrey, Mark W., Raheem, Izzat T., Barbe, Guillaume, Campeau, Louis-Charles, Dubost, David, McCabe Dunn, Jamie, Grobler, Jay, Hartingh, Timothy J., Hazuda, Daria J., Klein, Daniel, Miller, Michael D., Moore, Keith P., Nguyen, Natalie, Pajkovic, Natasa, Powell, David A., Rada, Vanessa, Sanders, John M., Sisko, John, Steele, Thomas G., Wai, John, Walji, Abbas, Xu, Min, Coleman, Paul J.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Journal Article
3-Aryl-5-phenoxymethyl-1,3-oxazolidin-2-ones as positive allosteric modulators of mGluR2 for the treatment of schizophrenia: Hit-to-lead efforts
Brnardic, Edward J., Fraley, Mark E., Garbaccio, Robert M., Layton, Mark E., Sanders, John M., Culberson, Chris, Jacobson, Marlene A., Magliaro, Brian C., Hutson, Pete H., O’Brien, Julie A., Huszar, Sarah L., Uslaner, Jason M., Fillgrove, Kerry L., Tang, Cuyue, Kuo, Yuhsin, Sur, Sylvie M., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Journal Article
Crystallographic Structures of Two Bisphosphonate:1-Deoxyxylulose-5-Phosphate Reductoisomerase Complexes
Yajima, Shunsuke, Hara, Kodai, Sanders, John M, Yin, Fenglin, Ohsawa, Kanju, Wiesner, Jochen, Jomaa, Hassan, Oldfield, Eric
Published in Journal of the American Chemical Society (08.09.2004)
Published in Journal of the American Chemical Society (08.09.2004)
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Journal Article
Augmenting Hit Identification by Virtual Screening Techniques in Small Molecule Drug Discovery
Yan, Xin Cindy, Sanders, John M, Gao, Ying-Duo, Tudor, Matthew, Haidle, Andrew M, Klein, Daniel J, Converso, Antonella, Lesburg, Charles A, Zang, Yi, Wood, Harold B
Published in Journal of chemical information and modeling (28.09.2020)
Published in Journal of chemical information and modeling (28.09.2020)
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Journal Article
Potent, selective and orally bioavailable leucine-rich repeat kinase 2 (LRRK2) inhibitors
Greshock, Thomas J., Sanders, John M., Drolet, Robert E., Rajapakse, Hemaka A., Chang, Ronald K., Kim, Boyoung, Rada, Vanessa L., Tiscia, Heather E., Su, Hua, Lai, Ming-Tain, Sur, Sylvie M., Sanchez, Rosa I., Bilodeau, Mark T., Renger, John J., Kern, Jonathan T., McCauley, John A.
Published in Bioorganic & medicinal chemistry letters (01.06.2016)
Published in Bioorganic & medicinal chemistry letters (01.06.2016)
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Journal Article
Solid-State NMR, Crystallographic, and Computational Investigation of Bisphosphonates and Farnesyl Diphosphate Synthase−Bisphosphonate Complexes
Mao, Junhong, Mukherjee, Sujoy, Zhang, Yong, Cao, Rong, Sanders, John M, Song, Yongcheng, Zhang, Yonghui, Meints, Gary A, Gao, Yi Gui, Mukkamala, Dushyant, Hudock, Michael P, Oldfield, Eric
Published in Journal of the American Chemical Society (15.11.2006)
Published in Journal of the American Chemical Society (15.11.2006)
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Journal Article
Synthesis and optimization of N-heterocyclic pyridinones as catechol-O-methyltransferase (COMT) inhibitors
Zhao, Zhijian, Harrison, Scott T., Schubert, Jeffrey W., Sanders, John M., Polsky-Fisher, Stacey, Zhang, Nanyan Rena, McLoughlin, Debra, Gibson, Christopher R., Robinson, Ronald G., Sachs, Nancy A., Kandebo, Monika, Yao, Lihang, Smith, Sean M., Hutson, Pete H., Wolkenberg, Scott E., Barrow, James C.
Published in Bioorganic & medicinal chemistry letters (15.06.2016)
Published in Bioorganic & medicinal chemistry letters (15.06.2016)
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Journal Article
High concentration electrophysiology-based fragment screen: Discovery of novel acid-sensing ion channel 3 (ASIC3) inhibitors
Wolkenberg, Scott E., Zhao, Zhijian, Mulhearn, James J., Harrison, Scott T., Sanders, John M., Cato, Matthew J., Jovanovska, Aneta, Panigel, Jacqueline, Cook, Sean P., Henze, Darrell A., Kane, Stefanie A., Hartman, George D., Barrow, James C.
Published in Bioorganic & medicinal chemistry letters (01.05.2011)
Published in Bioorganic & medicinal chemistry letters (01.05.2011)
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Journal Article
HIV SUBSTITUTED QUINOLIZINE DERIVATIVES USEFUL AS HIV INTEGRASE INHIBITORS
WADDELL SHERMAN TIM, COLEMAN PAUL J, WAI JOHN S, SANDERS JOHN M, FERGUSON RONALD, YU TAO, ZHANG YONGLIAN, STAMFORD ANDREW
Year of Publication 05.12.2017
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Year of Publication 05.12.2017
Patent
니코틴산 아세틸콜린 수용체의 알로스테릭 조정제
DUFFY JOSEPH L, GUIADEEN DEODIAL G, SANDERS JOHN M, GRESHOCK THOMAS J, LEAVITT KENNETH J, HUFF BELINDA C, BELL IAN M, SHIPE WILLIAM D, CAMPBELL BRIAN T, RADA VANESSA L, SUEN LINDA M, HARVEY ANDREW JOHN, CROWLEY BRENDAN M
Year of Publication 29.11.2018
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Year of Publication 29.11.2018
Patent
SUBSTITUTED QUINOLIZINE DERIVATIVES USEFUL AS HIV INTEGRASE INHIBITORS
WADDELL SHERMAN TIM, COLEMAN PAUL J, WAI JOHN S, SANDERS JOHN M, FERGUSON RONALD, YU TAO, ZHANG YONGLIAN, STAMFORD ANDREW
Year of Publication 31.05.2016
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Year of Publication 31.05.2016
Patent
Synthesis of chiral phosphoantigens and their activity in gamma delta T cell stimulation
Song, Yongcheng, Zhang, Yonghui, Wang, Hong, Raker, Amy M, Sanders, John M, Broderick, Erin, Clark, Allen, Morita, Craig T, Oldfield, Eric
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
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Journal Article
ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
CAMPBELL, BRIAN, T, SANDERS, JOHN, M, CROWLEY, BRENDAN M, HARVEY, ANDREW JOHN, SHIPE, WILLIAM, D, LEAVITT, KENNETH, J, BELL, IAN, M, RADA, VANESSA, L, GRESHOCK, THOMAS J, GUIADEEN, DEODIAL, G, DUFFY, JOSEPH, L, SUEN, LINDA, M, HUFF, BELINDA, C
Year of Publication 27.02.2023
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Year of Publication 27.02.2023
Patent
Substituted quinolizine derivatives useful as HIV integrase inhibitors
WADDELL Sherman Tim, YU Tao, ZHANG Yonglian, COLEMAN Paul J, STAMFORD Andrew, WAI John S, SANDERS John M, FERGUSON Ronald
Year of Publication 28.02.2022
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Year of Publication 28.02.2022
Patent
ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
LEAVITT, Kenneth, J, BELL, Ian, M, RADA, Vanessa, L, HUFF, Belinda, C, GRESHOCK, Thomas, J, SANDERS, John, M, DUFFY, Joseph, L, HARVEY, Andrew, John, CROWLEY, Brendan, M, CAMPBELL, Brian, T, GUIADEEN, Deodial, G, SHIPE, William, D, SUEN, Linda, M
Year of Publication 06.04.2022
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Year of Publication 06.04.2022
Patent
SUBSTITUTED BICYCLIC HETEROARYL ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
BELL, Ian, M, LEAVITT, Kenneth, J, RADA, Vanessa, L, CROWLEY, Brendan, M, GUIADEEN, Deodial, G, SHIPE, William, D, HARVEY, Andrew John, SUEN, Linda, M, SANDERS, John, M, GRESHOCK, Thomas, J
Year of Publication 06.04.2022
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Year of Publication 06.04.2022
Patent
ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
Crowley, Brendan M, Sanders, John M, Guiadeen, Deodial G, Huff, Belinda C, Shipe, William D, Campbell, Brian T, Greshock, Thomas J, Leavitt, Kenneth J, Suen, Linda M, Bell, Ian M, Duffy, Joseph L, Rada, Vanessa L, Harvey, Andrew John
Year of Publication 18.03.2022
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Year of Publication 18.03.2022
Patent
ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
HUFF Belinda C, GUIADEEN Deodial G, RADA Vanessa L, CAMPBELL Brian T, SUEN Linda M, SHIPE William D, HARVEY Andrew John, LEAVITT Kenneth J, BELL Ian M, CROWLEY Brendan M, GRESHOCK Thomas J, SANDERS John M, DUFFY Joseph L
Year of Publication 31.01.2022
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Year of Publication 31.01.2022
Patent