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Chu, Guo-Hua, Gu, Minghua, Cassel, Joel A., Belanger, Serge, Graczyk, Thomas M., DeHaven, Robert N., Conway-James, Nathalie, Koblish, Mike, Little, Patrick J., DeHaven-Hudkins, Diane L., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
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High-performance liquid chromatographic enantioseparation of methanobenzazocines
Barker, William M., Worm, Karin, Dolle, Roland E.
Published in Journal of Chromatography A (06.11.2009)
Published in Journal of Chromatography A (06.11.2009)
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Nascent structure–activity relationship study of a diastereomeric series of kappa opioid receptor antagonists derived from CJ-15,208
Dolle, Roland E., Michaut, Mathieu, Martinez-Teipel, Blanca, Seida, Pamela R., Ajello, Christopher W., Muller, Alison L., DeHaven, Robert N., Carroll, Patrick J.
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
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General and efficient synthetic approach to novel tricyclic spiroketones
Chu, Guo-Hua, Le Bourdonnec, Bertrand, Gu, Minghua, Saeui, Christopher T., Dolle, Roland E.
Published in Tetrahedron (04.07.2009)
Published in Tetrahedron (04.07.2009)
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Novel pyridine derivatives as potent and selective CB2 cannabinoid receptor agonists
CHU, Guo-Hua, SAEUI, Christopher T, BROGDON, Bernice, SMITH, Steve, LE BOURDONNEC, Bertrand, DOLLE, Roland E, WORM, Karin, WEAVER, Damian G, GOODMAN, Allan J, BROADRUP, Robert L, CASSE, Joel A, DEHAVEN, Robert N, LABUDA, Christopher J, KOBLISH, Michael
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
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Novel malonamide derivatives as potent κ opioid receptor agonists
Chu, Guo-Hua, Gu, Minghua, Cassel, Joel A., Belanger, Serge, Graczyk, Thomas M., DeHaven, Robert N., Conway-James, Nathalie, Koblish, Michael, Little, Patrick J., DeHaven-Hudkins, Diane L., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
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Sulfamoyl benzamides as novel CB2 cannabinoid receptor ligands
WORM, Karin, ZHOU, Q. Jean, LITTLE, Patrick J, DOLLE, Roland E, SAEUI, Christopher T, GREEN, Rosalyn C, CASSEL, Joel A, STABLEY, Gabriel J, DEHAVEN, Robert N, CONWAY-JAMES, Nathalie, LABUDA, Christopher J, KOBLISH, Michael
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
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Novel sulfamoyl benzamides as selective CB2 agonists with improved in vitro metabolic stability
SELLITTO, Ian, LE BOURDONNEC, Bertrand, DEHAVEN, Robert N, LABUDA, Christopher J, KOBLISH, Michael, LITTLE, Patrick J, BROGDON, Bernice L, SMITH, Steven A, DOLLE, Roland E, WORM, Karin, GOODMAN, Allan, SAVOLAINEN, Markku A, CHU, Guo-Hua, AJELLO, Christopher W, SAEUI, Christopher T, LEISTER, Lara K, CASSEL, Joel A
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Discovery of N-(3-(morpholinomethyl)-phenyl)-amides as potent and selective CB2 agonists
WORM, Karin, WEAVER, Damian G, KOBLISH, Michael, BROGDON, Bernice L, SMITH, Steven A, DOLLE, Roland E, GREEN, Rosalyn C, SAEUI, Christopher T, DULAY, Doreen-Marie S, BARKER, William M, CASSEL, Joel A, STABLEY, Gabriel J, DEHAVEN, Robert N, LABUDA, Christopher J
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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Biaryl cannabinoid mimetics—Synthesis and structure–activity relationship
Worm, Karin, Zhou, Q. Jean, Stabley, Gabriel J., DeHaven, Robert N., Dolle, Roland E.
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
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5,7-Dimethoxy-3-(4-Pyridinyl)Quinoline Is a Potent and Selective Inhibitor of Human Vascular .beta.-Type Platelet-Derived Growth Factor Receptor Tyrosine Kinase
Dolle, Roland E, Dunn, Joseph A, Bobko, Mark, Singh, Baldev, Kuster, Joan E, Baizman, Eugene, Harris, Alex L, Sawutz, David G, Miller, Deborah, Wang, Su, Faltynek, Connie R, Xie, Wen, Sarup, Jay, Bode, D. Christopher, Pagani, Edward D, Silver, Paul J
Published in Journal of medicinal chemistry (19.08.1994)
Published in Journal of medicinal chemistry (19.08.1994)
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