Identification of a novel allosteric GLP-1R antagonist HTL26119 using structure-based drug design
O'Brien, Alistair, Andrews, Stephen P., Baig, Asma H., Bortolato, Andrea, Brown, Alastair J.H., Brown, Giles A., Brown, Sue H., Christopher, John A., Congreve, Miles, Cooke, Robert M., De Graaf, Chris, Errey, James C., Fieldhouse, Charlotte, Jazayeri, Ali, Marshall, Fiona H., Mason, Jonathan S., Mobarec, Juan Carlos, Okrasa, Krzysztof, Steele, Kelly N., Southall, Stacey M., Teobald, Iryna, Watson, Steve P., Weir, Malcolm
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
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Agonists and Antagonists of Protease-Activated Receptor 2 Discovered within a DNA-Encoded Chemical Library Using Mutational Stabilization of the Target
Brown, Dean G., Brown, Giles A., Centrella, Paolo, Certel, Kaan, Cooke, Robert M., Cuozzo, John W., Dekker, Niek, Dumelin, Christoph E., Ferguson, Andrew, Fiez-Vandal, Cédric, Geschwindner, Stefan, Guié, Marie-Aude, Habeshian, Sevan, Keefe, Anthony D., Schlenker, Oliver, Sigel, Eric A., Snijder, Arjan, Soutter, Holly T., Sundström, Linda, Troast, Dawn M., Wiggin, Giselle, Zhang, Jing, Zhang, Ying, Clark, Matthew A.
Published in SLAS discovery (01.06.2018)
Published in SLAS discovery (01.06.2018)
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Sequenced Reactions with Samarium(II) Iodide. Sequential Intramolecular Reformatsky/Nucleophilic Acyl Substitution Reactions for the Synthesis of Medium-Sized Carbocycles
Molander, Gary A, Brown, Giles A, Storch de Gracia, Isabel
Published in Journal of organic chemistry (17.05.2002)
Published in Journal of organic chemistry (17.05.2002)
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사이클릭 아펠린 수용체 효능제
SCULLY CONOR, PAUL REBECCA, CONGREVE MILES STUART, BROWN GILES ALBERT
Year of Publication 15.06.2023
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Year of Publication 15.06.2023
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선형 아펠린 수용체 효능제
SCULLY CONOR, PAUL REBECCA, CONGREVE MILES STUART, BROWN GILES ALBERT
Year of Publication 15.06.2023
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GPR35 효능제 화합물
SWAIN NIGEL ALAN, FLANAGAN NEIL JOHN, WHITEHURST BENJAMIN, CONGREVE MILES STUART, BROWN GILES ALBERT
Year of Publication 29.12.2023
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Year of Publication 29.12.2023
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Aldehydes and ketones as dipolarophiles: application to the synthesis of oxapenams
Andrews, MD, Brown, GA, Charmant, JPH, Peakman, TM, Rebello, A, Walsh, KE, Gallagher, T, Hales, NJ
Published in Chemical communications (Cambridge, England) (07.02.1999)
Published in Chemical communications (Cambridge, England) (07.02.1999)
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경구 GLP 수용체 작용제
SCULLY CONOR, PAUL REBECCA, CONGREVE MILES STUART, BROWN GILES ALBERT, MUTO SUSUMU, NUKUI SEIJI, WADA HIROKI
Year of Publication 22.11.2022
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Year of Publication 22.11.2022
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GLP 수용체 작용제
SCULLY CONOR, PAUL REBECCA, BORTOLATO ANDREA, CONGREVE MILES STUART, BROWN GILES ALBERT
Year of Publication 22.11.2022
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Year of Publication 22.11.2022
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암에 대해 사용하기 위한 5-아미노-8--[1,2,4]트리아졸로[4,3-c]피리미딘-3-온 화합물
PAUL REBECCA, ANDREWS STEPHEN PHILIPPE, MASON JONATHAN STEPHEN, CONGREVE MILES STUART, RICHARDSON CHRISTINE MARY, BROWN GILES ALBERT
Year of Publication 13.04.2023
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Year of Publication 13.04.2023
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DEFLORIAN FRANCESCA, SWAIN NIGEL ALAN, ANDREWS STEPHEN PHILIPPE, MASON JONATHAN STEPHEN, CONGREVE MILES STUART, BROWN GILES ALBERT
Year of Publication 13.04.2023
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FIELDHOUSE CHARLOTTE, SWAIN NIGEL ALAN, BEAUDION DANIEL, CONGREVE MILES STUART, PICKWORTH MARK, BAYRAKDARIAN MALKEN, BROWN GILES ALBERT, TEOBALD BARRY, KARILA DELPHINE
Year of Publication 14.08.2023
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Year of Publication 14.08.2023
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FIELDHOUSE CHARLOTTE, TEOBALD BARRY JOHN, SWAIN NIGEL ALAN, CONGREVE MILES STUART, PICKWORTH MARK, BOTTEGONI GIOVANNI, BROWN GILES ALBERT
Year of Publication 29.06.2021
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Year of Publication 29.06.2021
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O'BRIEN MICHAEL ALISTAIR, DEFLORIAN FRANCESCA, SWAIN NIGEL ALAN, WATSON STEPHEN PAUL, OTT GREGORY R, CONGREVE MILES STUART, CANSFIELD ANDREW DAVID, CANSFIELD JULIE, BROWN GILES ALBERT
Year of Publication 21.02.2022
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Year of Publication 21.02.2022
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약제학적 화합물
TEOBALD BARRY JOHN, CONGREVE MILES STUART, CANSFIELD JULIE, BROWN GILES ALBERT, TEHAN BENJAMIN GERALD
Year of Publication 13.02.2020
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Year of Publication 13.02.2020
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Trapping highly reactive dipolarophiles. Exploiting the mechanism associated with the azomethine ylide strategy for beta-lactam synthesis
Brown, GA, Anderson, KM, Large, JM, Planchenault, D, Urban, D, Hales, NJ, Gallagher, T
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (2001)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (2001)
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The azomethine ylide strategy for beta-lactam synthesis. An evaluation of alternative pathways for azomethine ylide generation
Brown, GA, Martel, Wisedale, R, Charmant, JPH, Hales, NJ, Fishwick, CWG, Gallagher, T
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2001)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2001)
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