Inhibition of thioredoxin reductase by auranofin induces apoptosis in cisplatin-resistant human ovarian cancer cells
Marzano, Christine, Gandin, Valentina, Folda, Alessandra, Scutari, Guido, Bindoli, Alberto, Rigobello, Maria Pia
Published in Free radical biology & medicine (15.03.2007)
Published in Free radical biology & medicine (15.03.2007)
Get full text
Journal Article
Anticancer activity, DNA binding and cell mechanistic studies of estrogen-functionalised Cu(II) complexes
Barrett, Stephen, De Franco, Michele, Kellett, Andrew, Dempsey, Eithne, Marzano, Cristina, Erxleben, Andrea, Gandin, Valentina, Montagner, Diego
Published in Journal of biological inorganic chemistry (01.02.2020)
Published in Journal of biological inorganic chemistry (01.02.2020)
Get full text
Journal Article
Oxidative Stress Induced by Pt(IV) Pro-drugs Based on the Cisplatin Scaffold and Indole Carboxylic Acids in Axial Position
Tolan, Dina, Gandin, Valentina, Morrison, Liam, El-Nahas, Ahmed, Marzano, Cristina, Montagner, Diego, Erxleben, Andrea
Published in Scientific reports (11.07.2016)
Published in Scientific reports (11.07.2016)
Get full text
Journal Article
Antiproliferative Homoleptic and Heteroleptic Phosphino Silver(I) Complexes: Effect of Ligand Combination on Their Biological Mechanism of Action
Dammak, Khouloud, Porchia, Marina, De Franco, Michele, Zancato, Mirella, Naïli, Houcine, Gandin, Valentina, Marzano, Cristina
Published in Molecules (Basel, Switzerland) (23.11.2020)
Published in Molecules (Basel, Switzerland) (23.11.2020)
Get full text
Journal Article
Structural Manipulations of Marine Natural Products Inspire a New Library of 3-Amino-1,2,4-Triazine PDK Inhibitors Endowed with Antitumor Activity in Pancreatic Ductal Adenocarcinoma
Carbone, Daniela, De Franco, Michele, Pecoraro, Camilla, Bassani, Davide, Pavan, Matteo, Cascioferro, Stella, Parrino, Barbara, Cirrincione, Girolamo, Dall'Acqua, Stefano, Sut, Stefania, Moro, Stefano, Gandin, Valentina, Diana, Patrizia
Published in Marine drugs (04.05.2023)
Published in Marine drugs (04.05.2023)
Get full text
Journal Article
Cancer cell death induced by phosphine gold(I) compounds targeting thioredoxin reductase
Gandin, Valentina, Fernandes, Aristi Potamitou, Rigobello, Maria Pia, Dani, Barbara, Sorrentino, Francesca, Tisato, Francesco, Björnstedt, Mikael, Bindoli, Alberto, Sturaro, Alberto, Rella, Rocco, Marzano, Cristina
Published in Biochemical pharmacology (15.01.2010)
Published in Biochemical pharmacology (15.01.2010)
Get full text
Journal Article
Platinum(IV) Complexes of trans -1,2-diamino-4-cyclohexene: Prodrugs Affording an Oxaliplatin Analogue that Overcomes Cancer Resistance
Papadia, Paride, Micoli, Katia, Barbanente, Alessandra, Ditaranto, Nicoletta, Hoeschele, James D, Natile, Giovanni, Marzano, Cristina, Gandin, Valentina, Margiotta, Nicola
Published in International journal of molecular sciences (27.03.2020)
Published in International journal of molecular sciences (27.03.2020)
Get full text
Journal Article
Synthesis and Cytotoxic Activity Evaluation of New Cu(I) Complexes of Bis(pyrazol-1-yl) Acetate Ligands Functionalized with an NMDA Receptor Antagonist
Pellei, Maura, Bagnarelli, Luca, Luciani, Lorenzo, Del Bello, Fabio, Giorgioni, Gianfabio, Piergentili, Alessandro, Quaglia, Wilma, De Franco, Michele, Gandin, Valentina, Marzano, Cristina, Santini, Carlo
Published in International journal of molecular sciences (09.04.2020)
Published in International journal of molecular sciences (09.04.2020)
Get full text
Journal Article
Hydroxyapatite nanocrystals as a smart, pH sensitive, delivery system for kiteplatin
Lelli, Marco, Roveri, Norberto, Marzano, Cristina, Hoeschele, James D, Curci, Alessandra, Margiotta, Nicola, Gandin, Valentina, Natile, Giovanni
Published in Dalton transactions : an international journal of inorganic chemistry (16.08.2016)
Published in Dalton transactions : an international journal of inorganic chemistry (16.08.2016)
Get full text
Journal Article
Nanocrystalline carbonate-apatites: role of Ca/P ratio on the upload and release of anticancer platinum bisphosphonates
Iafisco, Michele, Palazzo, Barbara, Martra, Gianmario, Margiotta, Nicola, Piccinonna, Sara, Natile, Giovanni, Gandin, Valentina, Marzano, Cristina, Roveri, Norberto
Published in Nanoscale (01.01.2012)
Published in Nanoscale (01.01.2012)
Get full text
Journal Article
Glucose-coated superparamagnetic iron oxide nanoparticles prepared by metal vapour synthesis are electively internalized in a pancreatic adenocarcinoma cell line expressing GLUT1 transporter
Barbaro, Daniele, Di Bari, Lorenzo, Gandin, Valentina, Evangelisti, Claudio, Vitulli, Giovanni, Schiavi, Eleonora, Marzano, Cristina, Ferretti, Anna M, Salvadori, Piero
Published in PloS one (15.04.2015)
Published in PloS one (15.04.2015)
Get full text
Journal Article
In Vitro Antitumor Activity of the Water Soluble Copper(I) Complexes Bearing the Tris(hydroxymethyl)phosphine Ligand
Marzano, Cristina, Gandin, Valentina, Pellei, Maura, Colavito, Davide, Papini, Grazia, Lobbia, Giancarlo Gioia, Del Giudice, Elda, Porchia, Marina, Tisato, Francesco, Santini, Carlo
Published in Journal of medicinal chemistry (28.02.2008)
Published in Journal of medicinal chemistry (28.02.2008)
Get full text
Journal Article
Methylselenol formed by spontaneous methylation of selenide is a superior selenium substrate to the thioredoxin and glutaredoxin systems
Fernandes, Aristi P, Wallenberg, Marita, Gandin, Valentina, Misra, Sougat, Tisato, Francesco, Marzano, Cristina, Rigobello, Maria Pia, Kumar, Sushil, Björnstedt, Mikael
Published in PloS one (30.11.2012)
Published in PloS one (30.11.2012)
Get full text
Journal Article
Synthesis, Characterization and Biological Activity of Novel Cu(II) Complexes of 6-Methyl-2-Oxo-1,2-Dihydroquinoline-3-Carbaldehyde-4n-Substituted Thiosemicarbazones
Ramachandran, Eswaran, Gandin, Valentina, Bertani, Roberta, Sgarbossa, Paolo, Natarajan, Karuppannan, Bhuvanesh, Nattamai S P, Venzo, Alfonso, Zoleo, Alfonso, Mozzon, Mirto, Dolmella, Alessandro, Albinati, Alberto, Castellano, Carlo, Reis Conceição, Nuno, C Guedes da Silva, M Fátima, Marzano, Cristina
Published in Molecules (Basel, Switzerland) (17.04.2020)
Published in Molecules (Basel, Switzerland) (17.04.2020)
Get full text
Journal Article
In Vitro and in Vivo Anticancer Activity of Copper(I) Complexes with Homoscorpionate Tridentate Tris(pyrazolyl)borate and Auxiliary Monodentate Phosphine Ligands
Gandin, Valentina, Tisato, Francesco, Dolmella, Alessandro, Pellei, Maura, Santini, Carlo, Giorgetti, Marco, Marzano, Cristina, Porchia, Marina
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
Get full text
Journal Article
A Quadruple‐Action Platinum(IV) Prodrug with Anticancer Activity Against KRAS Mutated Cancer Cell Lines
Petruzzella, Emanuele, Braude, Jeremy Phillip, Aldrich‐Wright, Janice R., Gandin, Valentina, Gibson, Dan
Published in Angewandte Chemie International Edition (11.09.2017)
Published in Angewandte Chemie International Edition (11.09.2017)
Get full text
Journal Article
Novel design of dual-action Pt() anticancer pro-drugs based on cisplatin and derivatives of the tyrosine kinase inhibitors imatinib and nilotinib
Beirne, Darren Fergal, Farkaš, Barbara, Donati, Chiara, Gandin, Valentina, Rozas, Isabel, Velasco-Torrijos, Trinidad, Montagner, Diego
Published in Dalton transactions : an international journal of inorganic chemistry (10.10.2023)
Published in Dalton transactions : an international journal of inorganic chemistry (10.10.2023)
Get full text
Journal Article
Anticancer activity of new water-soluble sulfonated thiosemicarbazone copper(II) complexes targeting disulfide isomerase
Miglioli, Francesca, De Franco, Michele, Bartoli, Jennifer, Scaccaglia, Mirco, Pelosi, Giorgio, Marzano, Cristina, Rogolino, Dominga, Gandin, Valentina, Carcelli, Mauro
Published in European journal of medicinal chemistry (05.10.2024)
Published in European journal of medicinal chemistry (05.10.2024)
Get full text
Journal Article