Regional brain uptake of the muscarinic ligand, [ 18F]FP-TZTP, is greatly decreased in M2 receptor knockout mice but not in M1, M3 and M4 receptor knockout mice
Jagoda, E.M., Kiesewetter, D.O., Shimoji, K., Ravasi, L., Yamada, M., Gomeza, J., Wess, J., Eckelman, W.C.
Published in Neuropharmacology (01.04.2003)
Published in Neuropharmacology (01.04.2003)
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Journal Article
Muscarinic Cholinergic Receptor Measurements With [ F]FP-TZTP: Control and Competition Studies
Carson, Richard E., Kiesewetter, Dale O., Jagoda, Elaine, Der, Margaret G., Herscovitch, Peter, Eckelman, William C.
Published in Journal of cerebral blood flow and metabolism (01.10.1998)
Published in Journal of cerebral blood flow and metabolism (01.10.1998)
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Journal Article
Biologically stable [ 18F]-labeled benzylfluoride derivatives
Magata, Yasuhiro, Lang, Lixin, Kiesewetter, Dale O, Jagoda, Elaine M, Channing, Michael A, Eckelman, William C
Published in Nuclear medicine and biology (01.02.2000)
Published in Nuclear medicine and biology (01.02.2000)
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Journal Article
Syntheses and Biological Properties of Chiral Fluoroalkyl Quinuclidinyl Benzilates
Kiesewetter, Dale O, Silverton, James V, Eckelman, William C
Published in Journal of medicinal chemistry (01.05.1995)
Published in Journal of medicinal chemistry (01.05.1995)
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Journal Article
A review of new oncotropic tracers for pet imaging
Lang, L., Aloj, L., Kiesewetter, D.O., Jagoda, E., Lee, J.T., Paik, C.H., Carrasquillo, J.A., Eckelman, W.C.
Published in Nuclear medicine and biology (01.08.1996)
Published in Nuclear medicine and biology (01.08.1996)
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Journal Article
Conference Proceeding
Evaluation of stereoisomers of 4-fluoroalkyl analogues of 3-quinuclidinyl benzilate in in vivo competition studies for the M1, M2, and M3 muscarinic receptor subtypes in brain
Lee, Jaetae, Paik, Chang H., Kiesewetter, Dale O., Park, Seok G., Eckelman, William C.
Published in Nuclear medicine and biology (01.08.1995)
Published in Nuclear medicine and biology (01.08.1995)
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Journal Article
Preparation of 18F-Labeled Muscarinic Agonist with M2 Selectivity
Kiesewetter, Dale O, Lee, JaeTae, Lang, Lixin, Park, Seok Gun, Paik, Chang H, Eckelman, William C
Published in Journal of medicinal chemistry (01.01.1995)
Published in Journal of medicinal chemistry (01.01.1995)
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Journal Article
A single column, rapid quality control procedure for 6-[ 18F]fluoro- l-dopa and 6-[ 18F]fluorodopamine PET imaging agents
Dunn, Bonnie B., Channing, Michael A., Adams, H.Richard, Goldstein, David S., Kirk, Kenneth L., Kiesewetter, Dale O.
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1991)
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1991)
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Journal Article
Fluoro-, bromo-, and iodopaclitaxel derivatives: synthesis and biological evaluation
Kiesewetter, Dale O, Jagoda, Elaine M, Kao, Chih-Hao K, Ma, Ying, Ravasi, Laura, Shimoji, Kazuaki, Szajek, Lawrence P, Eckelman, William C
Published in Nuclear medicine and biology (2003)
Published in Nuclear medicine and biology (2003)
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Journal Article
The automated radiosynthesis of [ 18F]FP-TZTP
Kiesewetter, Dale O, Vuong, Bik-kee, Channing, Michael A
Published in Nuclear medicine and biology (2003)
Published in Nuclear medicine and biology (2003)
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Journal Article
Purification of the precursor for the automated radiosynthesis of [ [formula omitted]]FCWAY by counter-current chromatography
Ma, Ying, Lang, Lixin, Kiesewetter, Dale O, Vuong, Bik-Kee, Channing, Michael, Ito, Yoichiro, Eckelman, William C
Published in Journal of Chromatography A (23.04.2004)
Published in Journal of Chromatography A (23.04.2004)
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Journal Article
Determination of [ 18F]FCWAY, [ 18F]FP-TZTP, and their metabolites in plasma using rapid and efficient liquid-liquid and solid phase extractions
Ma, Ying, Kiesewetter, Dale O, Lang, Lixin, Der, Margaret, Huang, Bill, Carson, Richard E, Eckelman, William C
Published in Nuclear medicine and biology (01.04.2003)
Published in Nuclear medicine and biology (01.04.2003)
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Journal Article
Routine quality control of recycled target [ 18O]water by capillary electrophoresis and gas chromatography
Huang, Bill X., Channing, Michael A., Plascjak, Paul S., Kiesewetter, Dale O., Der, Margaret, Ma, Ying, Eckelman, William C.
Published in Nuclear medicine and biology (01.10.2003)
Published in Nuclear medicine and biology (01.10.2003)
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Journal Article
Radiochemical synthesis and biodistribution of a novel maxi-K potassium channel opener
Kiesewetter, Dale O, Jagoda, Elaine M, Starrett, John E, Gribkoff, Valentin K, Hewawasam, Piyasena, Srinivas, Nugahally, Salazar, Daniel, Eckelman, William C
Published in Nuclear medicine and biology (2002)
Published in Nuclear medicine and biology (2002)
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Journal Article
Characterization of the uptake of 16α-([ 18F]fluoro)-17β-estradiol in DMBA-induced mammary tumors
Mathias, Carla J., Welch, Michael J., Katzenellenbogen, John A., Brodack, James W., Kilbourn, Michael R., Carlson, Kathryn E., Kiesewetter, Dale O.
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1987)
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1987)
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Journal Article
Synthesis of a fluorinated fatty acid, dl-erthro-9,10-[18F]difluoropalmitic acid, and biodistribution studies in rats
SCHMALL, B, FINN, R. D, RAPOPORT, S. I, NORONHA, J. G, DEGEORGE, J. J, KIESEWETTER, D. O, SIMPSON, N. R, LARSON, S. M
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1990)
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Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1990)
Journal Article
Liquid chromatography-tandem mass spectrometry identification of metabolites of two 5-HT1A antagonists, N-{2-[4-(2-methoxylphenyl)piperazino]ethyl}-N-(2-pyridyl) trans-and cis-4-fluorocyclohexanecarboxamide, produced by human and rat hepatocytes
YING MA, LIXIN LANG, KIESEWETTER, Dale O, JAGODA, Elaine, SASSAMAN, Mark B, DER, Margaret, ECKELMAN, William C
Published in Journal of chromatography. B, Biomedical sciences and applications (05.05.2001)
Published in Journal of chromatography. B, Biomedical sciences and applications (05.05.2001)
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