The Differential Effects of Atypical Antipsychotics on Prolactin Elevation Are Explained by Their Differential Blood-Brain Disposition: A Pharmacological Analysis in Rats
Kapur, S, Langlois, X, Vinken, P, Megens, A A H P, De Coster, R, Andrews, J S
Published in The Journal of pharmacology and experimental therapeutics (01.09.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2002)
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Pharmacological Profile of (2R-trans)-4-[1-[3,5-bis(Trifluoromethyl)benzoyl]-2-(phenylmethyl)-4-piperidinyl]-N-(2,6-dimethylphenyl)-1-acetamide (S)-Hydroxybutanedioate (R116301), an Orally and Centrally Active Neurokinin-1 Receptor Antagonist
Megens, A A H P, Ashton, D, Vermeire, J C A, Vermote, P C M, Hens, K A, Hillen, L C, Fransen, J F, Mahieu, M, Heylen, L, Leysen, J E, Jurzak, M R, Janssens, F
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
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Attentional performance of (C57BL/6J × 129Sv)F2 mice in the five-choice serial reaction time task
de Bruin, N.M.W.J., Fransen, F., Duytschaever, H., Grantham, C., Megens, A.A.H.P.
Published in Physiology & behavior (30.12.2006)
Published in Physiology & behavior (30.12.2006)
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Lipophilic nalmefene prodrugs to achieve a one-month sustained release
Gaekens, Tim, Guillaume, Michel, Borghys, Herman, De Zwart, Loeckie L., de Vries, Ronald, Embrechts, Roger C.A., Vermeulen, An, Megens, Anton A.H.P., Leysen, Josée E., Herdewijn, Piet, Annaert, Pieter P., Atack, John R.
Published in Journal of controlled release (28.06.2016)
Published in Journal of controlled release (28.06.2016)
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Differential interaction of neuroleptics with apomorphine-induced behavior in rats as a function of changing levels of dopamine receptor stimulation
Megens, Anton A H P, Hendrickx, Herman M R, Lavreysen, Hilde, Langlois, Xavier
Published in The Journal of pharmacology and experimental therapeutics (01.12.2013)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2013)
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JNJ-40255293, a Novel Adenosine A2A/A1 Antagonist with Efficacy in Preclinical Models of Parkinson’s Disease
Atack, John R, Shook, Brian C, Rassnick, Stefanie, Jackson, Paul F, Rhodes, Kenneth, Drinkenburg, Wilhelmus H, Ahnaou, Abdallah, te Riele, Paula, Langlois, Xavier, Hrupka, Brian, De Haes, Patrick, Hendrickx, Herman, Aerts, Nancy, Hens, Koen, Wellens, Annemie, Vermeire, Jef, Megens, Anton A. H. P
Published in ACS chemical neuroscience (15.10.2014)
Published in ACS chemical neuroscience (15.10.2014)
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Humanization of Mouse 5-Hydroxytryptamine1B Receptor Gene by Homologous Recombination: In Vitro and In Vivo Characterization
Bonaventure, P, Umans, L, Bakker, M H, Cras, P, Langlois, X, Luyten, W H, Megens, A A, Serneels, L, Van Leuven, F, Leysen, J E
Published in Molecular pharmacology (01.07.1999)
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Published in Molecular pharmacology (01.07.1999)
Journal Article
Survey on the pharmacodynamics of the new antipsychotic risperidone
Megens, A A, Awouters, F H, Schotte, A, Meert, T F, Dugovic, C, Niemegeers, C J, Leysen, J E
Published in Psychopharmacology (01.02.1994)
Published in Psychopharmacology (01.02.1994)
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Pharmacology of JNJ-42314415, a centrally active phosphodiesterase 10A (PDE10A) inhibitor: a comparison of PDE10A inhibitors with D2 receptor blockers as potential antipsychotic drugs
Megens, Anton A H P, Hendrickx, Herman M R, Hens, Koen A, Fonteyn, Ineke, Langlois, Xavier, Lenaerts, Ilse, Somers, Marijke V F, de Boer, Peter, Vanhoof, Greet
Published in The Journal of pharmacology and experimental therapeutics (01.04.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2014)
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Journal Article
Interaction of antipsychotic drugs with neurotransmitter receptor sites in vitro and in vivo in relation to pharmacological and clinical effects: role of 5HT2 receptors
Leysen, J E, Janssen, P M, Schotte, A, Luyten, W H, Megens, A A
Published in Psychopharmacology (01.03.1993)
Published in Psychopharmacology (01.03.1993)
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Pharmacology of risperidone (R 64 766), a new antipsychotic with serotonin-S2 and dopamine-D2 antagonistic properties
JANSSEN, P. A. J, NIEMEGEERS, C. J. E, AWOUTERS, F, SCHELLEKENS, K. H. L, MEGENS, A. A. H. P, MEERT, T. F
Published in The Journal of pharmacology and experimental therapeutics (01.02.1988)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1988)
Journal Article
Comparison of the Analgesic and Intestinal Effects of Fentanyl and Morphine in Rats
Megens, Anton A.H.P., Artois, Kamiel, Vermeire, Jef, Meert, Theo, Awouters, Frans H.L.
Published in Journal of pain and symptom management (01.04.1998)
Published in Journal of pain and symptom management (01.04.1998)
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Conference Proceeding
Functional interaction between serotonin-S2 and dopamine-D2 neurotransmission as revealed by selective antagonism of hyper-reactivity to tryptamine and apomorphine
AWOUTERS, F, NIEMEGEERS, C. J. E, MEGENS, A. A. H. P, JANSSEN, P. A. J
Published in The Journal of pharmacology and experimental therapeutics (01.09.1990)
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Published in The Journal of pharmacology and experimental therapeutics (01.09.1990)
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