Bicyclic pyridine, pyrazine, and pyrimidine derivatives as PI3K beta inhibitors
Meerpoel, Lieven, Querolle, Olivier Alexis Georges, Berthelot, Didier Jean-Claude, Mercey, Guillaume Jean Maurice, Demestre, Christophe Gabriel Marcel, Pasquier, Elisabeth Thérèse Jeanne, Angibaud, Patrick René, Pilatte, Isabelle Noëlle Constance, Mevellec, Laurence Anne, Poncelet, Virginie Sophie, Coupa, Sophie, Meyer, Christophe
Year of Publication 01.07.2021
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Year of Publication 01.07.2021
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BICYCLIC PYRIDINE, PYRAZINE, AND PYRIMIDINE DERIVATIVES AS PI3K BETA INHIBITORS
Meerpoel, Lieven, Querolle, Olivier Alexis Georges, Berthelot, Didier Jean-Claude, Mercey, Guillaume Jean Maurice, Demestre, Christophe Gabriel Marcel, Pasquier, Elisabeth Thérèse Jeanne, Angibaud, Patrick René, Pilatte, Isabelle Noëlle Constance, Mevellec, Laurence Anne, Poncelet, Virginie Sophie, Coupa, Sophie, Meyer, Christophe
Year of Publication 28.05.2021
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Year of Publication 28.05.2021
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BICYCLIC PYRIDINE, PYRAZINE, AND PYRIMIDINE DERIVATIVES AS PI3K BETA INHIBITORS
MEERPOEL, Lieven, COUPA, Sophie, MERCEY, Guillaume, Jean, Maurice, BERTHELOT, Didier, Jean-Claude, PASQUIER, Elisabeth, Thérèse, Jeanne, MEVELLEC, Laurence, Anne, DEMESTRE, Christophe, Gabriel, Marcel, PONCELET, Virginie, Sophie, PILATTE, Isabelle, Noëlle, Constance, QUEROLLE, Olivier, Alexis, Georges, ANGIBAUD, Patrick, René, MEYER, Christophe
Year of Publication 24.02.2021
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Year of Publication 24.02.2021
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Azabenzimidazole derivatives as PI3K beta inhibitors
Querolle, Olivier Alexis Georges, Meerpoel, Lieven, Berthelot, Didier Jean-Claude, Mercey, Guillaume Jean Maurice, Demestre, Christophe Gabriel Marcel, Pasquier, Elisabeth Thérèse Jeanne, Angibaud, Patrick René, Pilatte, Isabelle Noëlle Constance, Mevellec, Laurence Anne, Poncelet, Virginie Sophie, Coupa, Sophie, Meyer, Christophe
Year of Publication 04.02.2021
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Year of Publication 04.02.2021
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AZABENZIMIDAZOLE DERIVATIVES AS PI3K BETA INHIBITORS
MEERPOEL, Lieven, COUPA, Sophie, MERCEY, Guillaume, Jean, Maurice, BERTHELOT, Didier, Jean-Claude, PASQUIER, Elisabeth, Thérèse, Jeanne, MEVELLEC, Laurence, Anne, DEMESTRE, Christophe, Gabriel, Marcel, PONCELET, Virginie, Sophie, PILATTE, Isabelle, Noëlle, Constance, QUEROLLE, Olivier, Alexis, Georges, ANGIBAUD, Patrick, René, MEYER, Christophe
Year of Publication 17.06.2020
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Year of Publication 17.06.2020
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PYRAZOLYL QUINOXALINE KINASE INHIBITORS
Besong, Gilbert Ebai, Govaerts, Tom Cornelis Hortense, Papanikos, Alexandra, Bonnet, Pascal Ghislain André, Woodhead, Steven John, Weerts, Johan Erwin Edmond, Berdini, Valerio, Perera, Timothy Pietro Suren, Querolle, Olivier Alexis Georges, Gilissen, Ronaldus Arnodus Hendrika Joseph, Pasquier, Elisabeth Thérèse Jeanne, Angibaud, Patrick René, Rees, David Charles, Mevellec, Laurence Anne, Embrechts, Werner Constant Johan, Reader, Michael, SAXTY, Gordon, Hamlett, Christopher Charles Frederick, Wroblowski, Berthold, Lacrampe, Jean Fernand Armand, Akkari, Rhalid, Meerpoel, Lieven, Pilatte, Isabelle Noëlle Constance, Freyne, Eddy Jean Edgard, Johnson, Christopher Norbert, Murray, Christopher William
Year of Publication 05.05.2022
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Year of Publication 05.05.2022
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IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
MEERPOEL, Lieven, COUPA, Sophie, MERCEY, Guillaume, Jean, Maurice, PASQUIER, Elisabeth, Thérèse, Jeanne, BERTHELOT, Didier, Jean-Claude, MEVELLEC, Laurence, Anne, DEMESTRE, Christophe, Gabriel, Marcel, PONCELET, Virginie, Sophie, PILATTE, Isabelle, Noëlle, Constance, QUEROLLE, Olivier, Alexis, Georges, MEYER, Christophe, ANGIBAUD, Patrick, René
Year of Publication 20.04.2020
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Year of Publication 20.04.2020
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PYRAZOLYL QUINOXALINE KINASE INHIBITORS
Besong, Gilbert Ebai, Govaerts, Tom Cornelis Hortense, Papanikos, Alexandra, Bonnet, Pascal Ghislain André, Woodhead, Steven John, Weerts, Johan Erwin Edmond, Berdini, Valerio, Perera, Timothy Pietro Suren, Querolle, Olivier Alexis Georges, Gilissen, Ronaldus Arnodus Hendrika Joseph, Pasquier, Elisabeth Thérèse Jeanne, Angibaud, Patrick René, Rees, David Charles, Mevellec, Laurence Anne, Saxty, Gordon, Embrechts, Werner Constant Johan, Reader, Michael, Hamlett, Christopher Charles Frederick, Wroblowski, Berthold, Lacrampe, Jean Fernand Armand, Akkari, Rhalid, Meerpoel, Lieven, Pilatte, Isabelle Noëlle Constance, Freyne, Eddy Jean Edgard, Johnson, Christopher Norbert, Murray, Christopher William
Year of Publication 18.02.2022
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Year of Publication 18.02.2022
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PYRAZOLYL QUINOXALINE KINASE INHIBITORS
LACRAMPE, JEAN FERNAND ARMAND, JOHNSON, CHRISTOPHER NORBERT, EMBRECHTS, WERNER CONSTANT JOHAN, PAPANIKOS, ALEXANDRA, WOODHEAD, STEVEN JOHN, PASQUIER, ELISABETH THÉRÈSE JEANNE, BONNET, PASCAL GHISLAIN ANDRE, ANGIBAUD, PATRICK RENÉ, WEERTS, JOHAN ERWIN EDMOND, GILISSEN, RONALDUS ARNODUS HENDRIKA JOSEPH, WROBLOWSKI, BERTHOLD, READER, MICHAEL, REES, DAVID CHARLES, AKKARI, RHALID, FREYNE, EDDY JEAN EDGARD, PILATTE, ISABELLE NOËLLE CONSTANCE, BESONG, GILBERT EBAI, MURRAY, CHRISTOPHER WILLIAM, HAMLETT, CHRISTOPHER CHARLES FREDERICK, SAXTY, GORDON, GOVAERTS, TOM CORNELIS HORTENSE, PERERA, TIMOTHY PIETRO SUREN, BERDINI, VALERIO, MEVELLEC, LAURENCE ANNE, QUEROLLE, OLIVIER ALEXIS GEORGES, MEERPOEL, LIEVEN
Year of Publication 07.02.2022
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Year of Publication 07.02.2022
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HETEROCYCLYL LINKED IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
Meerpoel, Lieven, Querolle, Olivier Alexis Georges, Berthelot, Didier Jean-Claude, Mercey, Guillaume Jean Maurice, Demestre, Christophe Gabriel Marcel, Pasquier, Elisabeth Thérèse Jeanne, Angibaud, Patrick René, Pilatte, Isabelle Noëlle Constance, Mevellec, Laurence Anne, Poncelet, Virginie Sophie, Coupa, Sophie, Meyer, Christophe
Year of Publication 21.02.2020
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Year of Publication 21.02.2020
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IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
MEVELLEC, LAURENCE ANNE, PASQUIER, ELISABETH THÉRÈSE JEANNE, QUEROLLE, OLIVIER ALEXIS GEORGES, ANGIBAUD, PATRICK RENÉ, BERTHELOT, DIDIER JEAN-CLAUDE, PILATTE, ISABELLE NOËLLE CONSTANCE, MERCEY, GUILLAUME JEAN MAURICE, PONCELET, VIRGINIE SOPHIE, MEERPOEL, LIEVEN, COUPA, SOPHIE, DEMESTRE, CHRISTOPHE GABRIEL MARCEL, MEYER, CHRISTOPHE
Year of Publication 31.01.2020
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Year of Publication 31.01.2020
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PYRAZOLYL QUINOXALINE KINASE INHIBITORS
FREYNE, EDDY, JEAN, EDGARD, MEVELLEC, LAURENCE, ANNE, MURRAY, CHRISTOPHER, WILLIAM, GOVAERTS, TOM, CORNELIS, HORTENSE, PAPANIKOS, ALEXANDRA, ANGIBAUD, PATRICK, RENÉ, PERERA, TIMOTHY, PIETRO, SUREN, WROBLOWSKI, BERTHOLD, PILATTE, ISABELLE, NOËLLE, CONSTANCE, READER, MICHAEL, REES, DAVID, CHARLES, AKKARI, RHALID, HAMLETT, CHRISTOPHER, CHARLES, FREDERICK, SAXTY, GORDON, WEERTS, JOHAN, ERWIN, EDMOND, BERDINI, VALERIO, GILISSEN, RONALDUS, ARNODUS, HENDRIKA, JOSEPH, QUEROLLE, OLIVIER, ALEXIS, GEORGES, JOHNSON, CHRISTOPHER, NORBERT, WOODHEAD, STEVEN, JOHN, EMBRECHTS, WERNER, CONSTANT, JOHAN, BESONG, GILBERT, EBAI, PASQUIER, ELISABETH, THÉRÈSE, JEANNE, LACRAMPE, JEAN, FERNAND, ARMAND, MEERPOEL, LIEVEN, BONNET, PASCAL, GHISLAIN, ANDRE
Year of Publication 31.12.2021
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Year of Publication 31.12.2021
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PYRAZOLYL QUINOXALINE KINASE INHIBITORS
MEERPOEL, Lieven, PAPANIKOS, Alexandra, JOHNSON, Christopher Norbert, WROBLOWSKI, Berthold, READER, Michael, PILATTE, Isabelle Noëlle Constance, FREYNE, Eddy Jean Edgard, LACRAMPE, Jean Fernand Armand, EMBRECHTS, Werner Constant Johan, BONNET, Pascal Ghislain Andre, PASQUIER, Elisabeth Thérèse Jeanne, BERDINI, Valerio, HAMLETT, Christopher Charles Frederick, BESONG, Gilbert Ebai, REES, David Charles, GILISSEN, Ronaldus Arnodus Hendrika Joseph, WOODHEAD, Steven John, AKKARI, Rhalid, MURRAY, Christopher William, SAXTY, Gordon, PERERA, Timothy Pietro Suren, MEVELLEC, Laurence Anne, GOVAERTS, Tom Cornelis Hortense, QUEROLLE, Olivier Alexis Georges, WEERTS, Johan Erwin Edmond, ANGIBAUD, Patrick René
Year of Publication 27.12.2021
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Year of Publication 27.12.2021
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SUBSTITUTED 4,5,6,7-TETRAHYDRO-PYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AND 5,6,7,8-TETRAHYDRO-4H-PYRAZOLO[1,5-A][1,4]DIAZEPINE DERIVATIVES AS ROS1 INHIBITORS
DESCAMPS, Sophie, MEERPOEL, Lieven, MERCEY, Guillaume, Jean, Maurice, JEANTY, Matthieu, Ludovic, PASQUIER, Elisabeth, Thérèse, Jeanne, VIALARD, Jorge, Eduardo, WROBLOWSKI, Berthold, MEVELLEC, Laurence, Anne, JOUSSEAUME, Thierry, François, Alain, Jean
Year of Publication 26.12.2018
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Year of Publication 26.12.2018
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IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
Meerpoel, Lieven, Querolle, Olivier Alexis Georges, Berthelot, Didier Jean-Claude, Mercey, Guillaume Jean Maurice, Demestre, Christophe Gabriel Marcel, Pasquier, Elisabeth Thérèse Jeanne, Angibaud, Patrick René, Pilatte, Isabelle Noëlle Constance, Mevellec, Laurence Anne, Poncelet, Virginie Sophie, Coupa, Sophie, Meyer, Christophe
Year of Publication 29.11.2019
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Year of Publication 29.11.2019
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IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
QUEROLLE, OLIVIER, ALEXIS, GEORGES, MEVELLEC, LAURENCE, ANNE, PONCELET, VIRGINIE, SOPHIE, PASQUIER, ELISABETH, THÉRÈSE, JEANNE, MERCEY, GUILLAUME, JEAN, MAURICE, BERTHELOT, DIDIER, JEAN-CLAUDE, MEERPOEL, LIEVEN, ANGIBAUD, PATRICK, RENÉ, COUPA, SOPHIE, PILATTE, ISABELLE, NOËLLE, CONSTANCE, DEMESTRE, CHRISTOPHE, GABRIEL, MARCEL, MEYER, CHRISTOPHE
Year of Publication 31.10.2019
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Year of Publication 31.10.2019
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IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
LIEVEN MEERPOEL, GUILLAUME JEAN MAURICE MERCEY, SOPHIE COUPA, CHRISTOPHE MEYER, PATRICK RENÉ ANGIBAUD, OLIVIER ALEXIS GEORGES QUEROLLE, CHRISTOPHE GABRIEL MARCEL DEMESTRE, ELISABETH THÉRÈSE JEANNE PASQUIER, DIDIE JEAN-CLAUDE BERTHELOT, LAURENCE ANNE MEVELLEC, VIRGINIE SOPHIE PONCELET, ISABELLE, NOËLLE CONSTANCE PILATTE
Year of Publication 09.10.2019
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Year of Publication 09.10.2019
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HETEROCYCLYL LINKED IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
MEERPOEL, Lieven, COUPA, Sophie, MERCEY, Guillaume, Jean, Maurice, PASQUIER, Elisabeth, Thérèse, Jeanne, BERTHELOT, Didier, Jean-Claude, MEVELLEC, Laurence, Anne, DEMESTRE, Christophe, Gabriel, Marcel, PONCELET, Virginie, Sophie, PILATTE, Isabelle, Noëlle, Constance, QUEROLLE, Olivier, Alexis, Georges, MEYER, Christophe, ANGIBAUD, Patrick, René
Year of Publication 25.09.2019
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Year of Publication 25.09.2019
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PYRAZOLYL QUINOXALINE KINASE INHIBITORS
MEERPOEL, Lieven, PAPANIKOS, Alexandra, JOHNSON, Christopher Norbert, WROBLOWSKI, Berthold, READER, Michael, PILATTE, Isabelle Noëlle Constance, FREYNE, Eddy Jean Edgard, LACRAMPE, Jean Fernand Armand, EMBRECHTS, Werner Constant Johan, BONNET, Pascal Ghislain Andre, PASQUIER, Elisabeth Thérèse Jeanne, BERDINI, Valerio, HAMLETT, Christopher Charles Frederick, BESONG, Gilbert Ebai, REES, David Charles, GILISSEN, Ronaldus Arnodus Hendrika Joseph, WOODHEAD, Steven John, AKKARI, Rhalid, MURRAY, Christopher William, SAXTY, Gordon, PERERA, Timothy Pietro Suren, MEVELLEC, Laurence Anne, GOVAERTS, Tom Cornelis Hortense, QUEROLLE, Olivier Alexis Georges, WEERTS, Johan Erwin Edmond, ANGIBAUD, Patrick René
Year of Publication 25.08.2021
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Year of Publication 25.08.2021
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IMIDAZOPYRIDAZINE DERIVATIVES AS PI3KBETA INHIBITORS
MEERPOEL, Lieven, COUPA, Sophie, MERCEY, Guillaume, Jean, Maurice, PASQUIER, Elisabeth, Thérèse, Jeanne, BERTHELOT, Didier, Jean-Claude, MEVELLEC, Laurence, Anne, DEMESTRE, Christophe, Gabriel, Marcel, PONCELET, Virginie, Sophie, PILATTE, Isabelle, Noëlle, Constance, QUEROLLE, Olivier, Alexis, Georges, MEYER, Christophe, ANGIBAUD, Patrick, René
Year of Publication 03.07.2019
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Year of Publication 03.07.2019
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