A Chemoproteomic Approach to Query the Degradable Kinome Using a Multi-kinase Degrader
Huang, Hai-Tsang, Dobrovolsky, Dennis, Paulk, Joshiawa, Yang, Guang, Weisberg, Ellen L., Doctor, Zainab M., Buckley, Dennis L., Cho, Joong-Heui, Ko, Eunhwa, Jang, Jaebong, Shi, Kun, Choi, Hwan Geun, Griffin, James D., Li, Ying, Treon, Steven P., Fischer, Eric S., Bradner, James E., Tan, Li, Gray, Nathanael S.
Published in Cell chemical biology (18.01.2018)
Published in Cell chemical biology (18.01.2018)
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Journal Article
Discovery of Novel 2,5-Dioxoimidazolidine-Based P2X7 Receptor Antagonists as Constrained Analogues of KN62
Park, Jin-Hee, Lee, Ga-Eun, Lee, So-Deok, Hien, Tran Thi, Kim, Sujin, Yang, Jin Won, Cho, Joong-Heui, Ko, Hyojin, Lim, Sung-Chul, Kim, Yoon-Gyoon, Kang, Keon-Wook, Kim, Yong-Chul
Published in Journal of medicinal chemistry (12.03.2015)
Published in Journal of medicinal chemistry (12.03.2015)
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Journal Article
Nanoparticle-encapsulated P2X7 receptor antagonist in a pH-sensitive polymer as a potential local drug delivery system to acidic inflammatory environments
Lee, Sun-Mi, Cho, Joong-Heui, Lee, So-Deok, Kim, Yong-Chul
Published in Bioorganic & medicinal chemistry letters (01.10.2015)
Published in Bioorganic & medicinal chemistry letters (01.10.2015)
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Journal Article
Benserazide, the first allosteric inhibitor of Coxsackievirus B3 3C protease
Kim, Bo-Kyoung, Cho, Joong-Heui, Jeong, Pyeonghwa, Lee, Youngjin, Lim, Jia Jia, Park, Kyoung Ryoung, Eom, Soo Hyun, Kim, Yong-Chul
Published in FEBS letters (08.07.2015)
Published in FEBS letters (08.07.2015)
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Journal Article
Insights of a Lead Optimization Study and Biological Evaluation of Novel 4‑Hydroxytamoxifen Analogs as Estrogen-Related Receptor γ (ERRγ) Inverse Agonists
Kim, Jina, Woo, Seo Yeon, Im, Chun Young, Yoo, Eun Kyung, Lee, Seungmi, Kim, Hyo-Ji, Hwang, Hee-Jong, Cho, Joong-heui, Lee, Won Seok, Yoon, Heeseok, Kim, Shinae, Kwon, Oh-bin, Hwang, Hayoung, Kim, Kyung-Hee, Jeon, Jae-Han, Singh, Thoudam Debraj, Kim, Sang Wook, Hwang, Sung Yeoun, Choi, Hueng-Sik, Lee, In-Kyu, Kim, Seong Heon, Jeon, Yong Hyun, Chin, Jungwook, Cho, Sung Jin
Published in Journal of medicinal chemistry (23.11.2016)
Published in Journal of medicinal chemistry (23.11.2016)
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Journal Article
Discovery of Potent Antiallodynic Agents for Neuropathic Pain Targeting P2X3 Receptors
Jung, Young-Hwan, Kim, Yeo Ok, Lin, Hai, Cho, Joong-Heui, Park, Jin-Hee, Lee, So-Deok, Bae, Jinsu, Kang, Koon Mook, Kim, Yoon-Gyoon, Pae, Ae Nim, Ko, Hyojin, Park, Chul-Seung, Yoon, Myung Ha, Kim, Yong-Chul
Published in ACS chemical neuroscience (19.07.2017)
Published in ACS chemical neuroscience (19.07.2017)
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Journal Article
Synthesis and biological evaluation of novel 4-hydroxytamoxifen analogs as estrogen-related receptor gamma inverse agonists
Kim, Jina, Chin, Jungwook, Im, Chun Young, Yoo, Eun Kyung, Woo, Seoyeon, Hwang, Hee Jong, Cho, Joong-heui, Seo, Kyung-ah, Song, Jaeyoung, Hwang, Hayoung, Kim, Kyung-Hee, Kim, Nam Doo, Yoon, Suk Kyoon, Jeon, Jae-Han, Yoon, Seung-Yun, Jeon, Yong Hyun, Choi, Hueng-Sik, Lee, In-Kyu, Kim, Seong Heon, Cho, Sung Jin
Published in European journal of medicinal chemistry (14.09.2016)
Published in European journal of medicinal chemistry (14.09.2016)
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Journal Article
Suppression of the metastatic spread of breast cancer by DN10764 (AZD7762)-mediated inhibition of AXL signaling
Park, Joon-Suk, Lee, ChuHee, Kim, Hyun-Kyoung, Kim, Dayea, Son, Jung Beom, Ko, Eunhwa, Cho, Joong-Heui, Kim, Nam-Doo, Nan, Hong-Yan, Kim, Choong-Yong, Yoon, Sukkyoon, Lee, Sun-Hwa, Choi, Hwan Geun
Published in Oncotarget (13.12.2016)
Published in Oncotarget (13.12.2016)
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Journal Article
Design and synthesis of potent and selective P2X3 receptor antagonists derived from PPADS as potential pain modulators
Cho, Joong-Heui, Jung, Kwan-Young, Jung, Younghwan, Kim, Min Hye, Ko, Hyojin, Park, Chul-Seung, Kim, Yong-Chul
Published in European journal of medicinal chemistry (2013)
Published in European journal of medicinal chemistry (2013)
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Journal Article
Structure–Activity Relationships and Optimization of 3,5-Dichloropyridine Derivatives As Novel P2X 7 Receptor Antagonists
Lee, Won-Gil, Lee, So-Deok, Cho, Joong-Heui, Jung, Younghwan, Kim, Jeong-hyun, Hien, Tran T., Kang, Keon-Wook, Ko, Hyojin, Kim, Yong-Chul
Published in Journal of medicinal chemistry (26.04.2012)
Published in Journal of medicinal chemistry (26.04.2012)
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Synthesis of potent chemical inhibitors of dynamin GTPase
Lee, Suho, Jung, Kwan-Young, Park, Joohyun, Cho, Joong-Heui, Kim, Yong-Chul, Chang, Sunghoe
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
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Design and synthesis of 1,4-dihydropyridine derivatives as BACE-1 inhibitors
Choi, Soo-Jeong, Cho, Joong-Heui, Im, Isak, Lee, So-Deok, Jang, Ji-Yeon, Oh, Yu-Min, Jung, Yong-Keun, Jeon, Eun-Seok, Kim, Yong-Chul
Published in European journal of medicinal chemistry (01.06.2010)
Published in European journal of medicinal chemistry (01.06.2010)
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Journal Article
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CHO JOONG HEUI, YOON HONG BIN, HAM YOUNG JIN, KWAK YOUNG SHIN, KIM JUNG JOON
Year of Publication 02.07.2024
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Year of Publication 02.07.2024
Patent
RON Novel compound as RON inhibitors
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KWAK, Young Shin, HAM, Young Jin, CHO, Joong Heui, KIM, Jung Joon, YOON, Hong Bin
Year of Publication 27.06.2024
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Year of Publication 27.06.2024
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NOVEL COMPOUND AS RON INHIBITOR
KWAK, Young Shin, HAM, Young Jin, CHO, Joong Heui, KIM, Jung Joon, YOON, Hong Bin
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Year of Publication 27.06.2024
Patent