Discovery of GSK2193874: An Orally Active, Potent, and Selective Blocker of Transient Receptor Potential Vanilloid 4
Cheung, Mui, Bao, Weike, Behm, David J, Brooks, Carl A, Bury, Michael J, Dowdell, Sarah E, Eidam, Hilary S, Fox, Ryan M, Goodman, Krista B, Holt, Dennis A, Lee, Dennis, Roethke, Theresa J, Willette, Robert N, Xu, Xiaoping, Ye, Guosen, Thorneloe, Kevin S
Published in ACS medicinal chemistry letters (11.05.2017)
Published in ACS medicinal chemistry letters (11.05.2017)
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Journal Article
Discovery of GSK3527497: A Candidate for the Inhibition of Transient Receptor Potential Vanilloid‑4 (TRPV4)
Brooks, Carl A, Barton, Linda S, Behm, David J, Brnardic, Edward J, Costell, Melissa H, Holt, Dennis A, Jolivette, Larry J, Matthews, Jay M, McAtee, John J, McCleland, Brent W, Patterson, Jaclyn R, Pero, Joseph E, Rivero, Ralph A, Roethke, Theresa J, Sanchez, Robert M, Shenje, Raynold, Terrell, Lamont R, Lawhorn, Brian G
Published in Journal of medicinal chemistry (24.10.2019)
Published in Journal of medicinal chemistry (24.10.2019)
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Journal Article
Discovery of GSK2798745: A Clinical Candidate for Inhibition of Transient Receptor Potential Vanilloid 4 (TRPV4)
Brooks, Carl A, Barton, Linda S, Behm, David J, Eidam, Hilary S, Fox, Ryan M, Hammond, Marlys, Hoang, Tram H, Holt, Dennis A, Hilfiker, Mark A, Lawhorn, Brian G, Patterson, Jaclyn R, Stoy, Patrick, Roethke, Theresa J, Ye, Guosen, Zhao, Steve, Thorneloe, Kevin S, Goodman, Krista B, Cheung, Mui
Published in ACS medicinal chemistry letters (08.08.2019)
Published in ACS medicinal chemistry letters (08.08.2019)
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Journal Article
TRPV4 antagonists
Li, Peng, Pero, Joseph E, Matthews, Jay M, Lawhorn, Brian Griffin, Sender, Matthew Robert, Behm, David J, McAtee, John Jeffrey, Brooks, Carl A, Brnardic, Edward J, Terrell, Lamont Roscoe
Year of Publication 01.03.2022
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Year of Publication 01.03.2022
Patent
TRPV4 ANTAGONISTS
BROOKS, Carl A, LAWHORN, Brian Griffin, PERO, Joseph E, LI, Peng, SENDER, Matthew Robert, BRNARDIC, Edward J, McATEE, John Jeffrey, MATTHEWS, Jay M, TERRELL, Lamont Roscoe, BEHM, David J
Year of Publication 30.09.2021
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Year of Publication 30.09.2021
Patent
TRPV4 ANTAGONISTS
MCATEE, John Jeffrey, BROOKS, Carl A, LAWHORN, Brian Griffin, PERO, Joseph E, LI, Peng, SENDER, Matthew Robert, BRNARDIC, Edward J, MATTHEWS, Jay M, TERRELL, Lamont Roscoe, BEHM, David J
Year of Publication 31.03.2021
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Year of Publication 31.03.2021
Patent