A Three-Site Mechanism for Agonist/Antagonist Selective Binding to Vasopressin Receptors
Saleh, Noureldin, Saladino, Giorgio, Gervasio, Francesco L., Haensele, Elke, Banting, Lee, Whitley, David C., Sopkova-de Oliveira Santos, Jana, Bureau, Ronan, Clark, Timothy
Published in Angewandte Chemie (International ed.) (04.07.2016)
Published in Angewandte Chemie (International ed.) (04.07.2016)
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Room-Temperature ortho-Alkoxylation and -Halogenation of N-Tosylbenzamides by Using Palladium(II)-Catalyzed CH Activation
Péron, Florent, Fossey, Christine, Sopkova-de Oliveira Santos, Jana, Cailly, Thomas, Fabis, Frédéric
Published in Chemistry : a European journal (10.06.2014)
Published in Chemistry : a European journal (10.06.2014)
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Effect of oral exposure to the acaricide pirimicarb, a new varroacide candidate, on Apis mellifera feeding rate
Riva, Clémence, Sokolowski, Michel BC, Normand, Julien, Santos, Jana Sopkova‐de Oliveira, Halm‐Lemeille, Marie‐Pierre
Published in Pest management science (01.08.2018)
Published in Pest management science (01.08.2018)
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Synthesis and Physicochemical Properties of Cryptophazane—A Soluble and Functionalizable C1‐Symmetrical Cryptophane
Vigier, Clément, Fayolle, Dimitri, El Siblani, Hussein, Sopkova ‐ de Oliveira Santos, Jana, Fabis, Frederic, Cailly, Thomas, Dubost, Emmanuelle
Published in Angewandte Chemie International Edition (14.11.2022)
Published in Angewandte Chemie International Edition (14.11.2022)
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Selecting the first chemical molecule inhibitor of HSP110 for colorectal cancer therapy
Gozzi, Gustavo J., Gonzalez, Daniel, Boudesco, Christophe, Dias, Alexandre M. M., Gotthard, Guillaume, Uyanik, Burhan, Dondaine, Lucile, Marcion, Guillaume, Hermetet, François, Denis, Camille, Hardy, Laurianne, Suzanne, Peggy, Douhard, Romain, Jego, Gaetan, Dubrez, Laurence, Demidov, Oleg N., Neiers, Fabrice, Briand, Loïc, Sopková-de Oliveira Santos, Jana, Voisin-Chiret, Anne-Sophie, Garrido, Carmen
Published in Cell death and differentiation (01.01.2020)
Published in Cell death and differentiation (01.01.2020)
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Web Resource
Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer's Disease
Toublet, François-Xavier, Lecoutey, Cédric, Lalut, Julien, Hatat, Bérénice, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopkova de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in Molecules (Basel, Switzerland) (31.07.2019)
Published in Molecules (Basel, Switzerland) (31.07.2019)
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Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5‑HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers
Dubost, Emmanuelle, Dumas, Noé, Fossey, Christine, Magnelli, Rosa, Butt-Gueulle, Sabrina, Ballandonne, Céline, Caignard, Daniel H, Dulin, Fabienne, Sopkova de-Oliveira Santos, Jana, Millet, Philippe, Charnay, Yves, Rault, Sylvain, Cailly, Thomas, Fabis, Frederic
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
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Journal Article
An Efficient and Straightforward Access to Sulfur Substituted [2.2]Paracyclophanes: Application to Stereoselective Sulfenate Salt Alkylation
Lohier, Jean-François, Foucoin, Florian, Jaffrès, Paul-Alain, Garcia, José I, Sopková−de Oliveira Santos, Jana, Perrio, Stéphane, Metzner, Patrick
Published in Organic letters (20.03.2008)
Published in Organic letters (20.03.2008)
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Journal Article
Structure-guided design of pyridoclax derivatives based on Noxa / Mcl-1 interaction mode
Hedir, Siham, De Giorgi, Marcella, Fogha, Jade, De Pascale, Martina, Weiswald, Louis-Bastien, Brotin, Emilie, Marekha, Bogdan, Denoyelle, Christophe, Denis, Camille, Suzanne, Peggy, Gautier, Fabien, Juin, Philippe, Ligat, Laetitia, Lopez, Frédéric, Carlier, Ludovic, Legay, Rémi, Bureau, Ronan, Rault, Sylvain, Poulain, Laurent, Oliveira Santos, Jana Sopková-de, Voisin-Chiret, Anne Sophie
Published in European journal of medicinal chemistry (05.11.2018)
Published in European journal of medicinal chemistry (05.11.2018)
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Journal Article
Synthesis of Pyridoclax Analogues: Insight into Their Druggability by Investigating Their Physicochemical Properties and Interactions with Membranes
De Pascale, Martina, Iacopetta, Domenico, Since, Marc, Corvaisier, Sophie, Vie, Véronique, Paboeuf, Gilles, Hennequin, Didier, Perato, Serge, De Giorgi, Marcella, Sinicropi, Maria Stefania, Sopkova‐De Oliveira Santos, Jana, Voisin‐Chiret, Anne‐Sophie, Malzert‐Freon, Aurélie
Published in ChemMedChem (07.01.2020)
Published in ChemMedChem (07.01.2020)
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Journal Article
Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation
Peauger, Ludovic, Azzouz, Rabah, Gembus, Vincent, Ţînţaş, Mihaela-Liliana, Sopková-de Oliveira Santos, Jana, Bohn, Pierre, Papamicaël, Cyril, Levacher, Vincent
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
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Journal Article
Benzylphenylpyrrolizinones with Anti‐amyloid and Radical Scavenging Effects, Potentially Useful in Alzheimer's Disease Treatment
Jourdan, Jean‐Pierre, Since, Marc, El Kihel, Laïla, Lecoutey, Cédric, Corvaisier, Sophie, Legay, Rémi, Sopková‐de Oliveira Santos, Jana, Cresteil, Thierry, Malzert‐Fréon, Aurélie, Rochais, Christophe, Dallemagne, Patrick
Published in ChemMedChem (21.06.2017)
Published in ChemMedChem (21.06.2017)
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Protein Crystallography under Xenon and Nitrous Oxide Pressure: Comparison with In Vivo Pharmacology Studies and Implications for the Mechanism of Inhaled Anesthetic Action
Colloc’h, Nathalie, Sopkova-de Oliveira Santos, Jana, Retailleau, Pascal, Vivarès, Denis, Bonneté, Françoise, Langlois d’Estainto, Béatrice, Gallois, Bernard, Brisson, Alain, Risso, Jean-Jacques, Lemaire, Marc, Prangé, Thierry, Abraini, Jacques H.
Published in Biophysical journal (01.01.2007)
Published in Biophysical journal (01.01.2007)
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Insights into Mcl-1 Conformational States and Allosteric Inhibition Mechanism from Molecular Dynamics Simulations, Enhanced Sampling, and Pocket Crosstalk Analysis
Benabderrahmane, Mohammed, Bureau, Ronan, Voisin-Chiret, Anne Sophie, Sopkova-de Oliveira Santos, Jana
Published in Journal of chemical information and modeling (22.06.2020)
Published in Journal of chemical information and modeling (22.06.2020)
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Journal Article
Novel Multitarget-Directed Ligands (MTDLs) with Acetylcholinesterase (AChE) Inhibitory and Serotonergic Subtype 4 Receptor (5-HT4R) Agonist Activities As Potential Agents against Alzheimer’s Disease: The Design of Donecopride
Rochais, Christophe, Lecoutey, Cédric, Gaven, Florence, Giannoni, Patrizia, Hamidouche, Katia, Hedou, Damien, Dubost, Emmanuelle, Genest, David, Yahiaoui, Samir, Freret, Thomas, Bouet, Valentine, Dauphin, François, Sopkova de Oliveira Santos, Jana, Ballandonne, Céline, Corvaisier, Sophie, Malzert-Fréon, Aurélie, Legay, Remi, Boulouard, Michel, Claeysen, Sylvie, Dallemagne, Patrick
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
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Journal Article
Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer’s disease
Toublet, François-Xavier, Lalut, Julien, Hatat, Bérénice, Lecoutey, Cédric, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopková-de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in European journal of medicinal chemistry (15.01.2021)
Published in European journal of medicinal chemistry (15.01.2021)
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Journal Article
Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine “bio-oxidizable” prodrugs: Synthesis, biological evaluation and structure-activity relationship
Azzouz, Rabah, Peauger, Ludovic, Gembus, Vincent, Ţînţaş, Mihaela-Liliana, Sopková-de Oliveira Santos, Jana, Papamicaël, Cyril, Levacher, Vincent
Published in European journal of medicinal chemistry (10.02.2018)
Published in European journal of medicinal chemistry (10.02.2018)
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Journal Article
Synthesis, Crystal Structure and Thermal Properties of Phosphorylated Cyclotriphosphazenes
Lejeune, Nicolas, Dez, Isabelle, Jaffrès, Paul-Alain, Lohier, Jean-Fançois, Madec, Pierre-Jean, Sopkova-de Oliveira Santos, Jana
Published in European Journal of Inorganic Chemistry (01.01.2008)
Published in European Journal of Inorganic Chemistry (01.01.2008)
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Rational design of novel benzisoxazole derivatives with acetylcholinesterase inhibitory and serotoninergic 5-HT4 receptors activities for the treatment of Alzheimer’s disease
Lalut, Julien, Payan, Hugo, Davis, Audrey, Lecoutey, Cédric, Legay, Rémi, Sopkova-de Oliveira Santos, Jana, Claeysen, Sylvie, Dallemagne, Patrick, Rochais, Christophe
Published in Scientific reports (20.02.2020)
Published in Scientific reports (20.02.2020)
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