Discovery and Optimization of Novel Antagonists to the Human Neurokinin‑3 Receptor for the Treatment of Sex-Hormone Disorders (Part I)
Hoveyda, Hamid R, Fraser, Graeme L, Roy, Marie-Odile, Dutheuil, Guillaume, Batt, Frédéric, El Bousmaqui, Mohamed, Korac, Julien, Lenoir, François, Lapin, Alexey, Noël, Sophie, Blanc, Sébastien
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
Get full text
Journal Article
The role of ChemR23 in the induction and resolution of cigarette smoke-induced inflammation
Demoor, Tine, Bracke, Ken R, Dupont, Lisa L, Plantinga, Maud, Bondue, Benjamin, Roy, Marie-Odile, Lannoy, Vincent, Lambrecht, Bart N, Brusselle, Guy G, Joos, Guy F
Published in The Journal of immunology (1950) (01.05.2011)
Published in The Journal of immunology (1950) (01.05.2011)
Get full text
Journal Article
Proenkephalin A gene products activate a new family of sensory neuron-specific GPCRs
Lembo, Paola M.C, Grazzini, Eric, Groblewski, Thierry, O'Donnell, Dajan, Roy, Marie-Odile, Zhang, Ji, Hoffert, Cyrla, Cao, Jack, Schmidt, Ralf, Pelletier, Manon, Labarre, Maryse, Gosselin, Mylene, Fortin, Yves, Banville, Denis, Shen, S.H, Ström, Peter, Payza, Kemal, Dray, Andy, Walker, Philippe, Ahmad, Sultan
Published in Nature neuroscience (01.03.2002)
Published in Nature neuroscience (01.03.2002)
Get full text
Journal Article
Sensory Neuron-Specific Receptor Activation Elicits Central and Peripheral Nociceptive Effects in Rats
Grazzini, Eric, Puma, Carole, Roy, Marie-Odile, Yu, Xiao Hong, O'Donnell, Dajan, Schmidt, Ralf, Dautrey, Sophie, Ducharme, Julie, Perkins, Martin, Panetta, Rosemarie, Jennifer M. A. Laird, Ahmad, Sultan, Paola M. C. Lembo, Hökfelt, Tomas
Published in Proceedings of the National Academy of Sciences - PNAS (04.05.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (04.05.2004)
Get full text
Journal Article
Oxysterols direct immune cell migration via EBI2
Hannedouche, Sébastien, Zhang, Juan, Yi, Tangsheng, Shen, Weijun, Nguyen, Deborah, Pereira, João P., Guerini, Danilo, Baumgarten, Birgit U., Roggo, Silvio, Wen, Ben, Knochenmuss, Richard, Noël, Sophie, Gessier, Francois, Kelly, Lisa M., Vanek, Mirka, Laurent, Stephane, Preuss, Inga, Miault, Charlotte, Christen, Isabelle, Karuna, Ratna, Li, Wei, Koo, Dong-In, Suply, Thomas, Schmedt, Christian, Peters, Eric C., Falchetto, Rocco, Katopodis, Andreas, Spanka, Carsten, Roy, Marie-Odile, Detheux, Michel, Chen, Yu Alice, Schultz, Peter G., Cho, Charles Y., Seuwen, Klaus, Cyster, Jason G., Sailer, Andreas W.
Published in Nature (London) (28.07.2011)
Published in Nature (London) (28.07.2011)
Get full text
Journal Article
A truncated form of CKβ8‐1 is a potent agonist for human formyl peptide‐receptor‐like 1 receptor
Elagoz, Aram, Henderson, Duncan, Babu, Poda Suresh, Salter, Sylvia, Grahames, Caroline, Bowers, Lorna, Roy, Marie‐Odile, Laplante, Patricia, Grazzini, Eric, Ahmad, Sultan, Lembo, Paola M C
Published in British journal of pharmacology (01.01.2004)
Published in British journal of pharmacology (01.01.2004)
Get full text
Journal Article
Annexin-I expression modulates drug resistance in tumor cells
Wang, Ying, Serfass, Lucile, Roy, Marie-Odile, Wong, Judy, Bonneau, Anne-Marie, Georges, Elias
Published in Biochemical and biophysical research communications (06.02.2004)
Published in Biochemical and biophysical research communications (06.02.2004)
Get full text
Journal Article
Protein interactions in concentrated ribonuclease solutions
Boyer, Mireille, Roy, Marie-Odile, Jullien, Magali, Bonneté, Françoise, Tardieu, Annette
Published in Journal of crystal growth (01.01.1999)
Published in Journal of crystal growth (01.01.1999)
Get full text
Journal Article
Conference Proceeding
NK-3 N--5678---[124][43-a] NK-3 NOVEL CHIRAL N-ACYL-5678-SUBSTITUTED-TETRAHYDRO-[124]TRIAZOLO[43-a]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS PHARMACEUTICAL COMPOSITION METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
DUTHEUIL GUILLAUME, ROY MARIE ODILE, FRASER GRAEME, EL BOUSMAQUI MOHAMED, BATT FREDERIC, HOVEYDA HAMID
Year of Publication 28.11.2019
Get full text
Year of Publication 28.11.2019
Patent
Does fusion of domains from unrelated proteins affect their folding pathways and the structural changes involved in their function? A case study with the diphtheria toxin T domain
Chenal, Alexandre, Nizard, Philippe, Forge, Vincent, Pugnière, Martine, Roy, Marie-Odile, Mani, Jean-Claude, Guillain, Florent, Gillet, Daniel
Published in Protein engineering, design and selection (01.05.2002)
Published in Protein engineering, design and selection (01.05.2002)
Get full text
Journal Article
NOVEL CHIRAL N-ACYL-5,6,7,(8-SUBSTITUTED)-TETRAHYDRO-[1,2,4]TRIAZOLO[4,3-A]PYRAZINES AS SELECTIVE NK-3 RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR USE IN NK-3 RECEPTOR MEDIATED DISORDERS AND CHIRAL SYNTHESIS THEREOF
DUTHEUIL GUILLAUME, ROY MARIE ODILE, FRASER GRAEME, EL BOUSMAQUI MOHAMED, BATT FREDERIC, HOVEYDA HAMID
Year of Publication 13.06.2014
Get full text
Year of Publication 13.06.2014
Patent
Crystallization of monoacylated proteins: influence of acyl chain length
Roy, M O, Uppenberg, J, Robert, S, Boyer, M, Chopineau, J, Jullien, M
Published in European biophysics journal (01.01.1997)
Published in European biophysics journal (01.01.1997)
Get full text
Journal Article
A truncated form of CK β 8‐1 is a potent agonist for human formyl peptide‐receptor‐like 1 receptor
Elagoz, Aram, Henderson, Duncan, Babu, Poda Suresh, Salter, Sylvia, Grahames, Caroline, Bowers, Lorna, Roy, Marie‐Odile, Laplante, Patricia, Grazzini, Eric, Ahmad, Sultan, Lembo, Paola M C
Published in British journal of pharmacology (02.02.2009)
Published in British journal of pharmacology (02.02.2009)
Get full text
Journal Article
Corrigendum to “Discovery of 3-aryl-5-acylpiperazinyl-pyrazoles as antagonists to the NK3 receptor” [Bioorg. Med. Chem. Lett. 21 (2011) 1991–1996]
Hoveyda, Hamid R., Roy, Marie-Odile, Blanc, Sebastien, Noël, Sophie, Salvino, Joseph M., Ator, Mark A., Fraser, Graeme
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Get full text
Journal Article
Discovery of 3-aryl-5-acylpiperazinyl-pyrazoles as antagonists to the NK sub(3 receptor)
Hoveyda, Hamid R, Roy, Marie-Odile, Blanc, Sebastien, Noel, Sophie, Salvino, Joseph M, Ator, Mark A, Fraser, Graeme
Published in Bioorganic & medicinal chemistry letters (01.04.2011)
Published in Bioorganic & medicinal chemistry letters (01.04.2011)
Get full text
Journal Article