Capsaicin, a novel inhibitor of the NorA efflux pump, reduces the intracellular invasion of Staphylococcus aureus
NITIN PAL KALIA, MAHAJAN, Priya, MEHRA, Rukmankesh, NARGOTRA, Amit, JAI PARKASH SHARMA, KOUL, Surrinder, INSHAD ALI KHAN
Published in Journal of antimicrobial chemotherapy (01.10.2012)
Published in Journal of antimicrobial chemotherapy (01.10.2012)
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Journal Article
Cytochrome bd oxidase: an emerging anti-tubercular drug target
Saha, Pallavi, Das, Samarpita, Indurthi, Harish K, Kumar, Rohit, Roy, Arnab, Kalia, Nitin Pal, Sharma, Deepak K
Published in MedChemComm (20.03.2024)
Published in MedChemComm (20.03.2024)
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Journal Article
Targeting the Mycobacterium ulcerans cytochrome bc 1 :aa 3 for the treatment of Buruli ulcer
Scherr, Nicole, Bieri, Raphael, Thomas, Sangeeta S, Chauffour, Aurélie, Nitin Pal Kalia, Schneide, Paul, Ruf, Marie-Thérèse, Lamelas, Araceli, Manimekalai, Malathy S S, Grüber, Gerhard, Ishii, Norihisa, Suzuki, Koichi, Tanner, Marcel, Moraski, Garrett C, Miller, Marvin J, Witschel, Matthias, Jarlier, Vincent, Pluschke, Gerd, Pethe, Kevin
Published in Nature communications (01.12.2018)
Published in Nature communications (01.12.2018)
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Journal Article
Discovery of a Novel Mycobacterial F‐ATP Synthase Inhibitor and its Potency in Combination with Diarylquinolines
Hotra, Adam, Ragunathan, Priya, Ng, Pearly Shuyi, Seankongsuk, Pattarakiat, Harikishore, Amaravadhi, Sarathy, Jickky Palmae, Saw, Wuan‐Geok, Lakshmanan, Umayal, Sae‐Lao, Patcharaporn, Kalia, Nitin Pal, Shin, Joon, Kalyanasundaram, Revathy, Anbarasu, Sivaraj, Parthasarathy, Krupakar, Pradeep, Chaudhari Namrata, Makhija, Harshyaa, Dröge, Peter, Poulsen, Anders, Tan, Jocelyn Hui Ling, Pethe, Kevin, Dick, Thomas, Bates, Roderick W., Grüber, Gerhard
Published in Angewandte Chemie International Edition (03.08.2020)
Published in Angewandte Chemie International Edition (03.08.2020)
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Journal Article
Exploring rhodanine linked enamine–carbohydrazide derivatives as mycobacterial carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and molecular docking studies
Maddipatla, Sarvan, Bakchi, Bulti, Gadhave, Rutuja Rama, Ammara, Andrea, Sau, Shashikanta, Rani, Bandela, Nanduri, Srinivas, Kalia, Nitin Pal, Supuran, Claudiu T., Yaddanapudi, Venkata Madhavi
Published in Archiv der Pharmazie (Weinheim) (01.07.2024)
Published in Archiv der Pharmazie (Weinheim) (01.07.2024)
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Journal Article
M. tuberculosis relies on trace oxygen to maintain energy homeostasis and survive in hypoxic environments
Kalia, Nitin Pal, Singh, Samsher, Hards, Kiel, Cheung, Chen-Yi, Sviriaeva, Ekaterina, Banaei-Esfahani, Amir, Aebersold, Ruedi, Berney, Michael, Cook, Gregory M., Pethe, Kevin
Published in Cell reports (Cambridge) (30.05.2023)
Published in Cell reports (Cambridge) (30.05.2023)
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Journal Article
Piperine as an inhibitor of the MdeA efflux pump of Staphylococcus aureus
ZAHID MEHMOOD MIRZA, KUMAR, Ashwani, NITIN PAL KALIA, ZARGAR, Afzal, INSHAD ALI KHAN
Published in Journal of medical microbiology (01.10.2011)
Published in Journal of medical microbiology (01.10.2011)
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Journal Article
Tweaking host immune responses for novel therapeutic approaches against Mycobacterium tuberculosis
Roy, Arnab, Kumari Agnivesh, Puja, Sau, Shashikanta, Kumar, Sunil, Pal Kalia, Nitin
Published in Drug discovery today (01.09.2023)
Published in Drug discovery today (01.09.2023)
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Journal Article
Exploration of 3-aryl pyrazole-tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors
Ommi, Ojaswitha, Paoletti, Niccolo, Bonardi, Alessandro, Gratteri, Paola, Bhalerao, Harshada Anil, Sau, Shashikanta, Nanduri, Srinivas, Mohammed, Arifuddin, Kalia, Nitin Pal, Sonti, Rajesh, Supuran, Claudiu T., Yaddanapudi, Venkata Madhavi
Published in Archiv der Pharmazie (Weinheim) (01.11.2023)
Published in Archiv der Pharmazie (Weinheim) (01.11.2023)
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Journal Article
Synthesis and pharmacological evaluation of 1,3-diaryl substituted pyrazole based (thio)urea derivatives as potent antimicrobial agents against multi-drug resistant Staphylococcus aureus and Mycobacterium tuberculosis
Ommi, Ojaswitha, Ahmad, Mohammad Naiyaz, Gajula, Siva Nageswara Rao, Wanjari, Parita, Sau, Shashikanta, Agnivesh, Puja Kumari, Sahoo, Santosh Kumar, Kalia, Nitin Pal, Sonti, Rajesh, Nanduri, Srinivas, Dasgupta, Arunava, Chopra, Sidharth, Yaddanapudi, Venkata Madhavi
Published in MedChemComm (20.07.2023)
Published in MedChemComm (20.07.2023)
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Journal Article
GaMF1.39's antibiotic efficacy and its enhanced antitubercular activity in combination with clofazimine, Telacebec, ND-011992, or TBAJ-876
Ragunathan, Priya, Shuyi Ng, Pearly, Singh, Samsher, Poh, Wee Han, Litty, Dennis, Kalia, Nitin Pal, Larsson, Simon, Harikishore, Amaravadhi, Rice, Scott A, Ingham, Philip W, Müller, Volker, Moraski, Garrett, Miller, Marvin J, Dick, Thomas, Pethe, Kevin, Grüber, Gerhard
Published in Microbiology spectrum (12.12.2023)
Published in Microbiology spectrum (12.12.2023)
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Journal Article
Discovery of a Novel Mycobacterial F‐ATP Synthase Inhibitor and its Potency in Combination with Diarylquinolines
Hotra, Adam, Ragunathan, Priya, Ng, Pearly Shuyi, Seankongsuk, Pattarakiat, Harikishore, Amaravadhi, Sarathy, Jickky Palmae, Saw, Wuan‐Geok, Lakshmanan, Umayal, Sae‐Lao, Patcharaporn, Kalia, Nitin Pal, Shin, Joon, Kalyanasundaram, Revathy, Anbarasu, Sivaraj, Parthasarathy, Krupakar, Pradeep, Chaudhari Namrata, Makhija, Harshyaa, Dröge, Peter, Poulsen, Anders, Tan, Jocelyn Hui Ling, Pethe, Kevin, Dick, Thomas, Bates, Roderick W., Grüber, Gerhard
Published in Angewandte Chemie (03.08.2020)
Published in Angewandte Chemie (03.08.2020)
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Journal Article
Synthesis and Antitubercular Activity of Berberine Derivatives
Mahapatra, Anita, Maheswari, Vijay, Kalia, Nitin Pal, Rajput, Vikrant S, Khan, Inshad Ali
Published in Chemistry of natural compounds (01.05.2014)
Published in Chemistry of natural compounds (01.05.2014)
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Journal Article
P-glycoprotein inhibitors as an adjunct therapy for TB
Parida, Kishan Kumar, Lahiri, Monali, Ghosh, Mainak, Dalal, Aman, Kalia, Nitin Pal
Published in Drug discovery today (01.09.2024)
Published in Drug discovery today (01.09.2024)
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Journal Article
Role of transcription termination factor Rho in anti-tuberculosis drug discovery
Kumar, Sunil, Sau, Shashikanta, Agnivesh, Puja Kumari, Roy, Arnab, Kalia, Nitin Pal
Published in Drug discovery today (01.03.2023)
Published in Drug discovery today (01.03.2023)
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Journal Article
Exploring and exploiting the host cell autophagy during Mycobacterium tuberculosis infection
Nagdev, Pavan Kumar, Agnivesh, Puja Kumari, Roy, Arnab, Sau, Shashikanta, Kalia, Nitin Pal
Published in European journal of clinical microbiology & infectious diseases (01.11.2023)
Published in European journal of clinical microbiology & infectious diseases (01.11.2023)
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Journal Article
Design, Synthesis, Evaluation of Antitubercular Activity and Insilco Studies of Novel 1,5-Naphthyridin-2(1H)-one Pendent 1,2,3-Triazoles
Chilakala, Nagendra Babu, Roy, Arnab, Kalia, Nitin Pal, Thumma, Vishnu, B, Raju, Etnoori, Sharada, K, Premalatha
Published in Chemistry & biodiversity (21.08.2024)
Published in Chemistry & biodiversity (21.08.2024)
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Journal Article