Synthesis and use of FSCPX, an irreversible adenosine A1 antagonist, as a 'Receptor knock-down' tool
VAN MUIJLWIJK-KOEZEN, Jacqueline E, TIMMERMAN, Henk, VAN DER SLUIS, Richard P, VAN DE STOLPE, Andrea C, MENGE, Wiro M. P. B, BEUKERS, Margot W, VAN DER GRAAF, Piet H, DE GROOTE, Miriam, IJZERMAN, Adriaan P
Published in Bioorganic & medicinal chemistry letters (26.03.2001)
Published in Bioorganic & medicinal chemistry letters (26.03.2001)
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New high affinity H3 receptor agonists without a basic side chain
KITBUNNADAJ, Ruengwit, HOFFMANN, Marcel, LEURS, Rob, FRATANTONI, Silvina A, BONGERS, Gerold, BAKKER, Remko A, WIELAND, Kerstin, EL JILALI, Ahmed, DE ESCH, Iwan J. P, MENGE, Wiro M. P. B, TIMMERMAN, Henk
Published in Bioorganic & medicinal chemistry (01.12.2005)
Published in Bioorganic & medicinal chemistry (01.12.2005)
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A role for spinal, but not supraspinal, α2 adrenergic receptors in the actions of improgan, a powerful, non-opioid analgesic
SVOKOS, Konstantina, NALWALK, Julia W, LEURS, Rob, MENGE, Wiro M. P. B, TIMMERMAN, Henk, HOUGH, Lindsay B
Published in Brain research (27.12.2001)
Published in Brain research (27.12.2001)
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Cytotoxicity of a series of mono- and di-substituted thiourea in freshly isolated rat hepatocytes: a preliminary structure-toxicity relationship study
Onderwater, Rob C.A, Commandeur, Jan N.M, Groot, Ed J, Sitters, Astrid, Menge, Wiro M.P.B, Vermeulen, Nico P.E
Published in Toxicology (Amsterdam) (06.02.1998)
Published in Toxicology (Amsterdam) (06.02.1998)
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Journal Article
Absence of antinociceptive tolerance to improgan, a cimetidine analog, in rats
Bannoura, Michelle D, Nalwalk, Julia W, Tang, Yuming, Carlile, MaryEllen, Leurs, Rob, Menge, Wiro M.P.B, Timmerman, Henk, Hough, Lindsay B
Published in Brain research (14.12.1998)
Published in Brain research (14.12.1998)
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Journal Article
Identification of 4-(1H-Imidazol-4(5)-ylmethyl)pyridine (Immethridine) as a Novel, Potent, and Highly Selective Histamine H3 Receptor Agonist
Kitbunnadaj, Ruengwit, Zuiderveld, Obbe P, Christophe, Bernard, Hulscher, Saskia, Menge, Wiro M. P. B, Gelens, Edith, Snip, Erwin, Bakker, Remko A, Celanire, Sylvain, Gillard, Michel, Talaga, Patrice, Timmerman, Henk, Leurs, Rob
Published in Journal of medicinal chemistry (06.05.2004)
Published in Journal of medicinal chemistry (06.05.2004)
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Journal Article
Isoquinoline and Quinazoline Urea Analogues as Antagonists for the Human Adenosine A3 Receptor
van Muijlwijk-Koezen, Jacqueline E, Timmerman, Henk, van der Goot, Henk, Menge, Wiro M. P. B, Frijtag von Drabbe Künzel, Jacobien, de Groote, Miriam, IJzerman, Adriaan P
Published in Journal of medicinal chemistry (01.06.2000)
Published in Journal of medicinal chemistry (01.06.2000)
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N-Substituted Piperidinyl Alkyl Imidazoles: Discovery of Methimepip as a Potent and Selective Histamine H3 Receptor Agonist
Kitbunnadaj, Ruengwit, Hashimoto, Takeshi, Poli, Enzo, Zuiderveld, Obbe P, Menozzi, Alessandro, Hidaka, Ryoko, de Esch, Iwan J. P, Bakker, Remko A, Menge, Wiro M. P. B, Yamatodani, Atsushi, Coruzzi, Gabriella, Timmerman, Henk, Leurs, Rob
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Journal Article
Synthesis and Structure−Activity Relationships of Conformationally Constrained Histamine H3 Receptor Agonists
Kitbunnadaj, Ruengwit, Zuiderveld, Obbe P, De Esch, Iwan J. P, Vollinga, Roeland C, Bakker, Remko, Lutz, Martin, Spek, Anthony L, Cavoy, Emile, Deltent, Marie-France, Menge, Wiro M. P. B, Timmerman, Henk, Leurs, Rob
Published in Journal of medicinal chemistry (04.12.2003)
Published in Journal of medicinal chemistry (04.12.2003)
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Journal Article
Synthesis and Structure−Activity Relationship of the First Nonpeptidergic Inverse Agonists for the Human Cytomegalovirus Encoded Chemokine Receptor US28
Hulshof, Janneke W, Casarosa, Paola, Menge, Wiro M. P. B, Kuusisto, Leena M. S, van der Goot, Henk, Smit, Martine J, de Esch, Iwan J. P, Leurs, Rob
Published in Journal of medicinal chemistry (06.10.2005)
Published in Journal of medicinal chemistry (06.10.2005)
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A Chemical Switch for the Modulation of the Functional Activity of Higher Homologues of Histamine on the Human Histamine H3 Receptor: Effect of Various Substitutions at the Primary Amino Function
Govoni, Marinella, Lim, Herman D., El-Atmioui, Dris, Menge, Wiro M. P. B., Timmerman, Henk, Bakker, Remko A., Leurs, Rob, De Esch, Iwan J. P.
Published in Journal of medicinal chemistry (20.04.2006)
Published in Journal of medicinal chemistry (20.04.2006)
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Journal Article
New high affinity H 3 receptor agonists without a basic side chain
Kitbunnadaj, Ruengwit, Hoffmann, Marcel, Fratantoni, Silvina A., Bongers, Gerold, Bakker, Remko A., Wieland, Kerstin, Jilali, Ahmed el, De Esch, Iwan J.P., Menge, Wiro M.P.B., Timmerman, Henk, Leurs, Rob
Published in Bioorganic & medicinal chemistry (01.12.2005)
Published in Bioorganic & medicinal chemistry (01.12.2005)
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Journal Article
Synthesis of Novel Se-Substituted Selenocysteine Derivatives as Potential Kidney Selective Prodrugs of Biologically Active Selenol Compounds: Evaluation of Kinetics of β-Elimination Reactions in Rat Renal Cytosol
Andreadou, Ioanna, Menge, Wiro M. P. B, Commandeur, Jan N. M, Worthington, Eduard A, Vermeulen, Nico P. E
Published in Journal of medicinal chemistry (10.05.1996)
Published in Journal of medicinal chemistry (10.05.1996)
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Journal Article
Evaluation of [ 18 F]VUF 5000 as a potential PET ligand for brain imaging of the histamine H 3 receptor
Windhorst, Albert D., Timmerman, Henk, Klok, Rob P., Menge, Wiro M.P.B., Leurs, Rob, Herscheid, Jacobus D.M.
Published in Bioorganic & medicinal chemistry (01.09.1999)
Published in Bioorganic & medicinal chemistry (01.09.1999)
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Journal Article
A Third Life for Burimamide: Discovery and Characterization of a Novel Class of Non-Opioid Analgesics Derived from Histamine Antagonists
HOUGH, LINDSAY B., NALWALK, JULIA W., BARNES, WILLIAM G., LEURS, ROB, MENGE, WIRO M. P. B., TIMMERMAN, HENK, WENTLAND, MARK
Published in Annals of the New York Academy of Sciences (01.01.2000)
Published in Annals of the New York Academy of Sciences (01.01.2000)
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