ATR kinase inhibitor AZD6738 potentiates CD8+ T cell-dependent antitumor activity following radiation
Vendetti, Frank P, Karukonda, Pooja, Clump, David A, Teo, Troy, Lalonde, Ronald, Nugent, Katriana, Ballew, Matthew, Kiesel, Brian F, Beumer, Jan H, Sarkar, Saumendra N, Conrads, Thomas P, O'Connor, Mark J, Ferris, Robert L, Tran, Phuoc T, Delgoffe, Greg M, Bakkenist, Christopher J
Published in The Journal of clinical investigation (31.08.2018)
Published in The Journal of clinical investigation (31.08.2018)
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Journal Article
Safety and Efficacy of T-DM1 Plus Neratinib in Patients With Metastatic HER2-Positive Breast Cancer: NSABP Foundation Trial FB-10
Abraham, Jame, Montero, Albert J, Jankowitz, Rachel C, Salkeni, Mohamad Adham, Beumer, Jan H, Kiesel, Brian F, Piette, Fanny, Adamson, Laura M, Nagy, Rebecca J, Lanman, Richard B, Sperinde, Jeff, Huang, Weidong, Allegra, Carmen J, Srinivasan, Ashok, Wang, Ying, Pogue-Geile, Katherine L, Lucas, Peter C, Jacobs, Samuel A
Published in Journal of clinical oncology (10.10.2019)
Published in Journal of clinical oncology (10.10.2019)
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Journal Article
Phase I Study of Veliparib (ABT-888) Combined with Cisplatin and Vinorelbine in Advanced Triple-Negative Breast Cancer and/or BRCA Mutation-Associated Breast Cancer
Rodler, Eve T, Kurland, Brenda F, Griffin, Melissa, Gralow, Julie R, Porter, Peggy, Yeh, Rosa F, Gadi, Vijayakrishna K, Guenthoer, Jamie, Beumer, Jan H, Korde, Larissa, Strychor, Sandra, Kiesel, Brian F, Linden, Hannah M, Thompson, John A, Swisher, Elizabeth, Chai, Xiaoyu, Shepherd, Stacie, Giranda, Vincent, Specht, Jennifer M
Published in Clinical cancer research (15.06.2016)
Published in Clinical cancer research (15.06.2016)
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Journal Article
Non-linear IV pharmacokinetics of the ATR inhibitor berzosertib (M6620) in mice
Deppas, Joshua J., Kiesel, Brian F., Guo, Jianxia, Parise, Robert A., Clump, D. Andy, D’Argenio, David Z., Bakkenist, Christopher J., Beumer, Jan H.
Published in Cancer chemotherapy and pharmacology (01.08.2024)
Published in Cancer chemotherapy and pharmacology (01.08.2024)
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Journal Article
Dose-dependent bioavailability and tissue distribution of the ATR inhibitor AZD6738 (ceralasertib) in mice
Kiesel, Brian F., Guo, Jianxia, Parise, Robert A., Venkataramanan, Raman, Clump, David A., Bakkenist, Christopher J., Beumer, Jan H.
Published in Cancer chemotherapy and pharmacology (01.02.2022)
Published in Cancer chemotherapy and pharmacology (01.02.2022)
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Journal Article
Quantitation of the ataxia‐telangiectasia‐mutated and Rad3‐related inhibitor elimusertib (BAY‐1895344) in human plasma using LC–MS/MS
Kiesel, Brian F., Parise, Robert A., Krishnamurthy, Anuradha, Gore, Steven, Beumer, Jan H.
Published in Biomedical chromatography (01.11.2022)
Published in Biomedical chromatography (01.11.2022)
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Journal Article
Phase I and pharmacokinetic study of veliparib, a PARP inhibitor, and pegylated liposomal doxorubicin (PLD) in recurrent gynecologic cancer and triple negative breast cancer with long-term follow-up
Pothuri, Bhavana, Brodsky, Allison L., Sparano, Joseph A., Blank, Stephanie V., Kim, Mimi, Hershman, Dawn L., Tiersten, Amy, Kiesel, Brian F., Beumer, Jan H., Liebes, Leonard, Muggia, Franco
Published in Cancer chemotherapy and pharmacology (01.04.2020)
Published in Cancer chemotherapy and pharmacology (01.04.2020)
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Journal Article
Neratinib-Plus-Cetuximab in Quadruple-WT ( KRAS, NRAS, BRAF, PIK3CA ) Metastatic Colorectal Cancer Resistant to Cetuximab or Panitumumab: NSABP FC-7, A Phase Ib Study
Jacobs, Samuel A, Lee, James J, George, Thomas J, Wade, 3rd, James L, Stella, Philip J, Wang, Ding, Sama, Ashwin R, Piette, Fanny, Pogue-Geile, Katherine L, Kim, Rim S, Gavin, Patrick G, Lipchik, Corey, Feng, Huichen, Wang, Ying, Finnigan, Melanie, Kiesel, Brian F, Beumer, Jan H, Wolmark, Norman, Lucas, Peter C, Allegra, Carmen J, Srinivasan, Ashok
Published in Clinical cancer research (15.03.2021)
Published in Clinical cancer research (15.03.2021)
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Journal Article
Phase 1 study of the Aurora kinase A inhibitor alisertib (MLN8237) combined with the histone deacetylase inhibitor vorinostat in lymphoid malignancies
Siddiqi, Tanya, Frankel, Paul, Beumer, Jan H., Kiesel, Brian F., Christner, Susan, Ruel, Chris, Song, Joo Y., Chen, Robert, Kelly, Kevin R., Ailawadhi, Sikander, Kaesberg, Paul, Popplewell, Leslie, Puverel, Sandrine, Piekarz, Richard, Forman, Stephen J., Newman, Edward M.
Published in Leukemia & lymphoma (28.01.2020)
Published in Leukemia & lymphoma (28.01.2020)
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Journal Article
Dose-dependent bioavailability, absorption-rate limited elimination, and tissue distribution of the ATR inhibitor BAY-1895344 (elimusertib) in mice
Kiesel, Brian F., Deppas, Joshua J., Guo, Jianxia, Parise, Robert. A., Clump, David A., Bakkenist, Christopher J., Beumer, Jan H.
Published in Cancer chemotherapy and pharmacology (01.06.2022)
Published in Cancer chemotherapy and pharmacology (01.06.2022)
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Journal Article
In vitro evaluation of the metabolic enzymes and drug interaction potential of triapine
Joshi, Anand, Kiesel, Brian F., Chaphekar, Nupur, Jones, Reyna, Guo, Jianxia, Kunos, Charles A., Taylor, Sarah, Chu, Edward, Venkataramanan, Raman, Beumer, Jan H.
Published in Cancer chemotherapy and pharmacology (01.11.2020)
Published in Cancer chemotherapy and pharmacology (01.11.2020)
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Journal Article
A phase 1 study of veliparib (ABT-888) plus weekly carboplatin and paclitaxel in advanced solid malignancies, with an expansion cohort in triple negative breast cancer (TNBC) (ETCTN 8620)
Malhotra, Monica K., Pahuja, Shalu, Kiesel, Brian F., Appleman, Leonard J., Ding, Fei, Lin, Yan, Tawbi, Hussein A., Stoller, Ronald G., Lee, James J., Belani, Chandra P., Chen, Alice P., Giranda, Vincent L., Shepherd, Stacie Peacock, Emens, Leisha A., Ivy, S. Percy, Chu, Edward, Beumer, Jan H., Puhalla, Shannon
Published in Breast cancer research and treatment (01.04.2023)
Published in Breast cancer research and treatment (01.04.2023)
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Journal Article
A phase I study of veliparib with cyclophosphamide and veliparib combined with doxorubicin and cyclophosphamide in advanced malignancies
Tan, Antoinette R., Chan, Nancy, Kiesel, Brian F., Stein, Mark N., Moss, Rebecca A., Malhotra, Jyoti, Aisner, Joseph, Shah, Mansi, Gounder, Murugesan, Lin, Hongxia, Kane, Michael P., Lin, Yong, Ji, Jiuping, Chen, Alice, Beumer, Jan H., Mehnert, Janice M.
Published in Cancer chemotherapy and pharmacology (01.01.2022)
Published in Cancer chemotherapy and pharmacology (01.01.2022)
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Journal Article
Quantitation of iohexol, a glomerular filtration marker, in human plasma by LC–MS/MS
Holleran, Julianne L., Parise, Robert A., Guo, Jianxia, Kiesel, Brian F., Taylor, Sarah E., Ivy, S. Percy, Chu, Edward, Beumer, Jan H.
Published in Journal of pharmaceutical and biomedical analysis (10.09.2020)
Published in Journal of pharmaceutical and biomedical analysis (10.09.2020)
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Journal Article
Phase I trial of belinostat in combination with 13-cis-retinoic acid in advanced solid tumor malignancies: a California Cancer Consortium NCI/CTEP sponsored trial
Luu, Thehang, Frankel, Paul, Beumer, Jan H., Lim, Dean, Cristea, Mihaela, Appleman, Leonard J., Lenz, Heinz J., Gandara, David R., Kiesel, Brian F., Piekarz, Richard L., Newman, Edward M.
Published in Cancer chemotherapy and pharmacology (01.12.2019)
Published in Cancer chemotherapy and pharmacology (01.12.2019)
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Journal Article
A phase I pharmacokinetic study of belinostat in patients with advanced cancers and varying degrees of liver dysfunction
Takebe, Naoko, Beumer, Jan H., Kummar, Shivaani, Kiesel, Brian F., Dowlati, Afshin, O'Sullivan Coyne, Geraldine, Piekarz, Richard, Rubinstein, Lawrence, Fogli, Laura K., Vaishampayan, Ulka, Goel, Sanjay, O'Bryant, Cindy L., El‐Rayes, Bassel F., Chung, Vincent, Lenz, Heinz‐Josef, Kim, Richard, Belani, Chandra P., Tuscano, Joseph M., Schelman, William, Moore, Nancy, Doroshow, James H., Chen, Alice P.
Published in British journal of clinical pharmacology (01.11.2019)
Published in British journal of clinical pharmacology (01.11.2019)
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Journal Article
A phase 1 and pharmacodynamic study of chronically-dosed, single-agent veliparib (ABT-888) in patients with BRCA1- or BRCA2-mutated cancer or platinum-refractory ovarian or triple-negative breast cancer
Manzo, Julia, Puhalla, Shannon, Pahuja, Shalu, Ding, Fei, Lin, Yan, Appleman, Leonard, Tawbi, Hussein, Stoller, Ronald, Lee, James J., Diergaarde, Brenda, Kiesel, Brian F., Yu, Jing, Tan, Antoinette R., Belani, Chandra P., Chew, Helen, Garcia, Agustin A., Morgan, Robert J., Wahner Hendrickson, Andrea E., Visscher, Daniel W., Hurley, Rachel M., Kaufmann, Scott H., Swisher, Elizabeth M., Oesterreich, Steffi, Katz, Tiffany, Ji, Jiuping, Zhang, Yiping, Parchment, Ralph E., Chen, Alice, Duan, Wenrui, Giranda, Vincent, Shepherd, Stacie P., Ivy, S. Percy, Chu, Edward, Beumer, Jan H.
Published in Cancer chemotherapy and pharmacology (01.05.2022)
Published in Cancer chemotherapy and pharmacology (01.05.2022)
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Journal Article
Population pharmacokinetics and exposure–response assessment of veliparib co-administered with temozolomide in patients with myeloid leukemias
Singh, Renu, Mehrotra, Shailly, Gopalakrishnan, Mathangi, Gojo, Ivana, Karp, Judith E., Greer, Jacqueline M., Chen, Alice, Piekarz, Richard, Kiesel, Brian F., Gobburu, Jogarao, Rudek, Michelle A., Beumer, Jan H.
Published in Cancer chemotherapy and pharmacology (01.02.2019)
Published in Cancer chemotherapy and pharmacology (01.02.2019)
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Journal Article
LC–MS/MS assay for the quantitation of the ATR kinase inhibitor VX-970 in human plasma
Kiesel, Brian F., Scemama, Jonas, Parise, Robert A., Villaruz, Liza, Iffland, Andre, Doyle, Austin, Ivy, Percy, Chu, Edward, Bakkenist, Christopher J., Beumer, Jan H.
Published in Journal of pharmaceutical and biomedical analysis (30.11.2017)
Published in Journal of pharmaceutical and biomedical analysis (30.11.2017)
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