Discovery of Novel 2,5-Dioxoimidazolidine-Based P2X7 Receptor Antagonists as Constrained Analogues of KN62
Park, Jin-Hee, Lee, Ga-Eun, Lee, So-Deok, Hien, Tran Thi, Kim, Sujin, Yang, Jin Won, Cho, Joong-Heui, Ko, Hyojin, Lim, Sung-Chul, Kim, Yoon-Gyoon, Kang, Keon-Wook, Kim, Yong-Chul
Published in Journal of medicinal chemistry (12.03.2015)
Published in Journal of medicinal chemistry (12.03.2015)
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Journal Article
Insights of a Lead Optimization Study and Biological Evaluation of Novel 4‑Hydroxytamoxifen Analogs as Estrogen-Related Receptor γ (ERRγ) Inverse Agonists
Kim, Jina, Woo, Seo Yeon, Im, Chun Young, Yoo, Eun Kyung, Lee, Seungmi, Kim, Hyo-Ji, Hwang, Hee-Jong, Cho, Joong-heui, Lee, Won Seok, Yoon, Heeseok, Kim, Shinae, Kwon, Oh-bin, Hwang, Hayoung, Kim, Kyung-Hee, Jeon, Jae-Han, Singh, Thoudam Debraj, Kim, Sang Wook, Hwang, Sung Yeoun, Choi, Hueng-Sik, Lee, In-Kyu, Kim, Seong Heon, Jeon, Yong Hyun, Chin, Jungwook, Cho, Sung Jin
Published in Journal of medicinal chemistry (23.11.2016)
Published in Journal of medicinal chemistry (23.11.2016)
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Journal Article
Synthesis and biological evaluation of novel 4-hydroxytamoxifen analogs as estrogen-related receptor gamma inverse agonists
Kim, Jina, Chin, Jungwook, Im, Chun Young, Yoo, Eun Kyung, Woo, Seoyeon, Hwang, Hee Jong, Cho, Joong-heui, Seo, Kyung-ah, Song, Jaeyoung, Hwang, Hayoung, Kim, Kyung-Hee, Kim, Nam Doo, Yoon, Suk Kyoon, Jeon, Jae-Han, Yoon, Seung-Yun, Jeon, Yong Hyun, Choi, Hueng-Sik, Lee, In-Kyu, Kim, Seong Heon, Cho, Sung Jin
Published in European journal of medicinal chemistry (14.09.2016)
Published in European journal of medicinal chemistry (14.09.2016)
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Journal Article
Design and synthesis of potent and selective P2X3 receptor antagonists derived from PPADS as potential pain modulators
Cho, Joong-Heui, Jung, Kwan-Young, Jung, Younghwan, Kim, Min Hye, Ko, Hyojin, Park, Chul-Seung, Kim, Yong-Chul
Published in European journal of medicinal chemistry (2013)
Published in European journal of medicinal chemistry (2013)
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Journal Article
Structure–Activity Relationships and Optimization of 3,5-Dichloropyridine Derivatives As Novel P2X 7 Receptor Antagonists
Lee, Won-Gil, Lee, So-Deok, Cho, Joong-Heui, Jung, Younghwan, Kim, Jeong-hyun, Hien, Tran T., Kang, Keon-Wook, Ko, Hyojin, Kim, Yong-Chul
Published in Journal of medicinal chemistry (26.04.2012)
Published in Journal of medicinal chemistry (26.04.2012)
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Journal Article
Design and synthesis of 1,4-dihydropyridine derivatives as BACE-1 inhibitors
Choi, Soo-Jeong, Cho, Joong-Heui, Im, Isak, Lee, So-Deok, Jang, Ji-Yeon, Oh, Yu-Min, Jung, Yong-Keun, Jeon, Eun-Seok, Kim, Yong-Chul
Published in European journal of medicinal chemistry (01.06.2010)
Published in European journal of medicinal chemistry (01.06.2010)
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Journal Article
Discovery of Novel 2,5-Dioxoimidazolidine-Based P2X(7) Receptor Antagonists as Constrained Analogues of KN62
Park, Jin-Hee, Lee, Ga-Eun, Lee, So-Deok, Tran Thi Hien, Kim, Sujin, Yang, Jin Won, Cho, Joong-Heui, Ko, Hyojin, Lim, Sung-Chul, Kim, Yoon-Gyoon, Kang, Keon-Wook, Kim, Yong-Chul
Published in Journal of medicinal chemistry (12.03.2015)
Published in Journal of medicinal chemistry (12.03.2015)
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Journal Article
Design and synthesis of potent and selective P2X(3) receptor antagonists derived from PPADS as potential pain modulators
Cho, Joong-Heui, Jung, Kwan-Young, Jung, Younghwan, Kim, Mm Hye, Ko, Hyojin, Park, Chul-Seung, Kim, Yong-Chul
Published in European journal of medicinal chemistry (01.12.2013)
Published in European journal of medicinal chemistry (01.12.2013)
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Journal Article
Structure-Activity Relationships and Optimization of 3,5-Dichloropyridine Derivatives As Novel P2X(7) Receptor Antagonists
Lee, Won-Gil, Lee, So-Deok, Cho, Joong-Heui, Jung, Younghwan, Kim, Jeong-hyun, Hien, Tran T., Kang, Keon-Wook, Ko, Hyojin, Kim, Yong-Chul
Published in Journal of medicinal chemistry (26.04.2012)
Published in Journal of medicinal chemistry (26.04.2012)
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Journal Article
Discovery of Novel 2,5-Dioxoimidazolidine-Based P2X 7 Receptor Antagonists as Constrained Analogues of KN62
Park, Jin-Hee, Lee, Ga-Eun, Lee, So-Deok, Hien, Tran Thi, Kim, Sujin, Yang, Jin Won, Cho, Joong-Heui, Ko, Hyojin, Lim, Sung-Chul, Kim, Yoon-Gyoon, Kang, Keon-Wook, Kim, Yong-Chul
Published in Journal of medicinal chemistry (12.03.2015)
Published in Journal of medicinal chemistry (12.03.2015)
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Journal Article
Structure–Activity Relationships and Optimization of 3,5-Dichloropyridine Derivatives As Novel P2X7 Receptor Antagonists
Lee, Won-Gil, Lee, So-Deok, Cho, Joong-Heui, Jung, Younghwan, Kim, Jeong-hyun, Hien, Tran T, Kang, Keon-Wook, Ko, Hyojin, Kim, Yong-Chul
Published in Journal of medicinal chemistry (26.04.2012)
Published in Journal of medicinal chemistry (26.04.2012)
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Journal Article