Exploiting an Asp-Glu "switch" in glycogen synthase kinase 3 to design paralog-selective inhibitors for use in acute myeloid leukemia
Wagner, Florence F, Benajiba, Lina, Campbell, Arthur J, Weïwer, Michel, Sacher, Joshua R, Gale, Jennifer P, Ross, Linda, Puissant, Alexandre, Alexe, Gabriela, Conway, Amy, Back, Morgan, Pikman, Yana, Galinsky, Ilene, DeAngelo, Daniel J, Stone, Richard M, Kaya, Taner, Shi, Xi, Robers, Matthew B, Machleidt, Thomas, Wilkinson, Jennifer, Hermine, Olivier, Kung, Andrew, Stein, Adam J, Lakshminarasimhan, Damodharan, Hemann, Michael T, Scolnick, Edward, Zhang, Yan-Ling, Pan, Jen Q, Stegmaier, Kimberly, Holson, Edward B
Published in Science translational medicine (07.03.2018)
Published in Science translational medicine (07.03.2018)
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Journal Article
Dual targeting of the androgen receptor and PI3K/AKT/mTOR pathways in prostate cancer models improves antitumor efficacy and promotes cell apoptosis
Sugawara, Tatsuo, Nevedomskaya, Ekaterina, Heller, Simon, Böhme, Annika, Lesche, Ralf, Ahsen, Oliver, Grünewald, Sylvia, Nguyen, Holly M., Corey, Eva, Baumgart, Simon J., Georgi, Victoria, Pütter, Vera, Fernández‐Montalván, Amaury, Vasta, James D., Robers, Matthew B., Politz, Oliver, Mumberg, Dominik, Haendler, Bernard
Published in Molecular oncology (01.03.2024)
Published in Molecular oncology (01.03.2024)
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Journal Article
Resistance to kinase inhibition through shortened target engagement
Rangwala, Aziz M., Berger, Benedict-Tilman, Robers, Matthew B., Knapp, Stefan, Seeliger, Markus A.
Published in Molecular & cellular oncology (31.12.2022)
Published in Molecular & cellular oncology (31.12.2022)
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Journal Article
Small-molecule inhibition of the archetypal UbiB protein COQ8
Murray, Nathan H., Asquith, Christopher R. M., Fang, Zixiang, East, Michael P., Ptak, Naomi, Smith, Robert W., Vasta, James D., Zimprich, Chad A., Corona, Cesear R., Robers, Matthew B., Johnson, Gary L., Bingman, Craig A., Pagliarini, David J.
Published in Nature chemical biology (01.02.2023)
Published in Nature chemical biology (01.02.2023)
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Journal Article
Tumor-suppressor role of Notch3 in medullary thyroid carcinoma revealed by genetic and pharmacological induction
Jaskula-Sztul, Renata, Eide, Jacob, Tesfazghi, Sara, Dammalapati, Ajitha, Harrison, April D, Yu, Xiao-Min, Scheinebeck, Casi, Winston-McPherson, Gabrielle, Kupcho, Kevin R, Robers, Matthew B, Hundal, Amrit K, Tang, Weiping, Chen, Herbert
Published in Molecular cancer therapeutics (01.02.2015)
Published in Molecular cancer therapeutics (01.02.2015)
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Journal Article
OPLOPHORUS-DERIVED LUCIFERASES, NOVEL COELENTERAZINE SUBSTRATES, AND METHODS OF USE
WOOD MONIKA G, BINKOWSKI BROCK, SLATER MICHAEL R, WOOD KEITH V, HALL MARY, ENCELL LANCE P, ROBERS MATTHEW B
Year of Publication 24.07.2013
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Year of Publication 24.07.2013
Patent
Abstract 160: High target binding affinity with long lasting cellular target engagement and high dose intermittent schedule of PI3K inhibitor copanlisib contribute to the potent anti-tumor activity and good safety profile
Fernández-Montalván, Amaury E., Georgi, Victoria, Vasta, James, Glaeske, Sarah, Puetter, Vera, Robers, Matthew B., Moenning, Ursula, Sturz, Andrea, Lefranc, Julien, Ziegelbauer, Karl, Brands, Michael, Stegmann, Christian, Scott, William J., Liu, Ningshu
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 3512: Measuring intracellular target engagement and drug residence time with nanoBRET
Robers, Matthew B., Dart, Melanie, Zimprich, Chad, Kirkland, Thomas, Levin, Sergiy, Machleidt, Thomas, Hartnett, Jim, Zimmerman, Kris, Ohana, Rachel, Daniels, Danette, Cong, Mei, Fan, Frank, Wood, Keith
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Journal Article
Abstract 151: Advancing pathway analysis using bioluminescent reporters
Robers, Matthew B., Binkowski, Brock, Karassina, Natasha, Stecha, Pete, Eggers, Chris, Cheng, Jey, Zimmerman, Kris, Fan, Frank, Cong, Mei
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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Journal Article
OPLOPHORUS-DERIVED LUCIFERASES, NOVEL COELENTERAZINE SUBSTRATES, AND METHODS OF USE
Wood, Keith V, Binkowski, Brock, Slater, Michael R, Wood, Monika G, Encell, Lance P, Robers, Matthew B, Hall, Mary
Year of Publication 16.05.2024
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Year of Publication 16.05.2024
Patent
FUNCTIONALIZED NANOLUC INHIBITORS
MACHLEIDT, Thomas, MEISENHEIMER, Poncho, HALL, Mary, NATH, Nidhi, ROBERS, Matthew B, ZHOU, Wenhui, WALKER, Joel R, FLEMMING, Roderick, G
Year of Publication 08.02.2023
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Year of Publication 08.02.2023
Patent
OPLOPHORUS-DERIVED LUCIFERASES, NOVEL COELENTERAZINE SUBSTRATES, AND METHODS OF USE
Wood, Keith V, Binkowski, Brock, Slater, Michael R, Wood, Monika G, Encell, Lance P, Robers, Matthew B, Hall, Mary
Year of Publication 03.11.2022
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Year of Publication 03.11.2022
Patent
Oplophorus-derived luciferases, novel coelenterazine substrates, and methods of use
Wood, Keith V, Klaubert, Dieter, Binkowski, Brock, Slater, Michael R, Unch, James, Valley, Michael P, Wood, Monika G, Encell, Lance P, Robers, Matthew B, Hall, Mary, Meisenheimer, Poncho
Year of Publication 30.05.2023
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Year of Publication 30.05.2023
Patent
AKTIVERING AF BIOLUMINESCENS VIA STRUKTUREL KOMPLEMENTERING
BINKOWSKI, Brock, SCHWINN, Marie, DIXON, Andrew S, NATH, Nidhi, DART, Melanie, ROBERS, Matthew B, ENCELL, Lance P, ZEGZOUTI, Hicham, UNCH, James, MEISENHEIMER, Poncho, MACHLEIDT, Thomas, GOUELI, Said, PULUKKUNAT, Dileep K, WOOD, Keith V, WOOD, Monika G, MONDAL, Subhanjan, Kirkland, Thomas, Hall, Mary P
Year of Publication 19.08.2024
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Year of Publication 19.08.2024
Patent