Heterocyclic ketones as inhibitors of histone deacetylase
Vasudevan, Anil, Ji, Zhiqin, Frey, Robin R., Wada, Carol K., Steinman, Douglas, Heyman, H.Robin, Guo, Yan, Curtin, Michael L., Guo, Jun, Li, Junling, Pease, Lori, Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Get full text
Journal Article
Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Get full text
Journal Article
Trifluoromethyl ketones as inhibitors of histone deacetylase
Frey, Robin R., Wada, Carol K., Garland, Robert B., Curtin, Michael L., Michaelides, Michael R., Li, Junling, Pease, Lori J., Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Murphy, Shannon S., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Get full text
Journal Article
α-Keto amides as inhibitors of histone deacetylase
Wada, Carol K., Frey, Robin R., Ji, Zhiqin, Curtin, Michael L., Garland, Robert B., Holms, James H., Li, Junling, Pease, Lori J., Guo, Jun, Glaser, Keith B., Marcotte, Patrick A., Richardson, Paul L., Murphy, Shannon S., Bouska, Jennifer J., Tapang, Paul, Magoc, Terrance J., Albert, Daniel H., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Get full text
Journal Article
Biaryl Ether Retrohydroxamates as Potent, Long-lived, Orally Bioavailable MMP Inhibitors
Michaelides, Michael R., Dellaria, Joseph F., Gong, Jane, Holms, James H., Bouska, Jennifer J., Stacey, Jamie, Wada, Carol K., Heyman, H.Robin, Curtin, Michael L., Guo, Yan, Goodfellow, Carole L., Elmore, Ildiko B., Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Get full text
Journal Article
BROMODOMAIN INHIBITORS
WILLIAM J MCCLELLAN, ROBERT A MANTEI, JOHN H HOLMS, GEORGE S SHEPPARD, DAI YUJIA, CAROL K WADA, WARREN M KATI, LE WANG, LISA HASVOLD, LIU DACHUN, STEVEN D FIDANZE, MCDANIEL KEITH F, JOHN K PRATT
Year of Publication 08.11.2018
Get full text
Year of Publication 08.11.2018
Patent
BROMODOMAIN INHIBITORS
WILLIAM J MCCLELLAN, ROBERT A MANTEI, JOHN H HOLMS, GEORGE S SHEPPARD, DAI YUJIA, CAROL K WADA, WARREN M KATI, LE WANG, LISA HASVOLD, LIU DACHUN, STEVEN D FIDANZE, MCDANIEL KEITH F, JOHN K PRATT
Year of Publication 27.07.2017
Get full text
Year of Publication 27.07.2017
Patent
Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770
Curtin, Michael L., Florjancic, Alan S., Heyman, H.Robin, Michaelides, Michael R., Garland, Robert B., Holms, James H., Steinman, Douglas H., Dellaria, Joseph F., Gong, Jane, Wada, Carol K., Guo, Yan, Elmore, Ildiko B., Tapang, Paul, Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Bouska, Jennifer J., Goodfellow, Carole L., Bauch, Joy L., Marsh, Kennan C., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Get full text
Journal Article
Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Get full text
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Journal Article
BROMODOMAIN INHIBITORS
Fidanze, Steven D, Kati, Warren M, Sheppard, George S, Wada, Carol K, Wang, Le, McDaniel, Keith F, Holms, James H, Mantei, Robert A, Pratt, John K, McClellan, William J, Liu, Dachun, Dai, Yujia, Hasvold, Lisa
Year of Publication 25.05.2023
Get full text
Year of Publication 25.05.2023
Patent
BROMODOMAIN INHIBITORS
WADA, CAROL K, MCDANIEL, KEITH F, HASVOLD, LISA, LIU, DACHUN, MANTEI, ROBERT A, SHEPPARD, GEORGE S, HOLMS, JAMES H, MCCLELLAN, WILLIAM J, WANG, LE, PRATT, JOHN K, KATI, WARREN M, DAI, YUJIA, FIDANZE, STEVEN D
Year of Publication 04.01.2022
Get full text
Year of Publication 04.01.2022
Patent
BROMODOMAIN INHIBITORS
Fidanze, Steven D, Kati, Warren M, Sheppard, George S, Wada, Carol K, Wang, Le, McDaniel, Keith F, Holms, James H, Mantei, Robert A, Pratt, John K, McClellan, William J, Liu, Dachun, Dai, Yujia, Hasvold, Lisa
Year of Publication 05.08.2021
Get full text
Year of Publication 05.08.2021
Patent
Bromodomain inhibitors
DAI, Yujia, WANG, Le, SHEPPARD, George S, MANTEI, Robert A, McDANIEL, Keith F, PRATT, John K, HOLMS, James H, LIU, Dachun, HASVOLD, Liza, McCLELLAN, William J, FIDANZE, Steven D, KATI, Warren M, WADA, Carol K
Year of Publication 20.06.2019
Get full text
Year of Publication 20.06.2019
Patent
Bromodomain inhibitors
McClellan, William J, Frey, Robin R, Wada, Carol K, Wang, Le, Hansen, Todd M, McDaniel, Keith F, Liu, Dachun, Pratt, John K
Year of Publication 12.06.2018
Get full text
Year of Publication 12.06.2018
Patent
Bromodomain inhibitors
DAI, Yujia, WANG, Le, SHEPPARD, George S, MANTEI, Robert A, McDANIEL, Keith F, PRATT, John K, HOLMS, James H, LIU, Dachun, HASVOLD, Liza, McCLELLAN, William J, FIDANZE, Steven D, KATI, Warren M, WADA, Carol K
Year of Publication 16.05.2019
Get full text
Year of Publication 16.05.2019
Patent
Bromodomain inhibitors
DAI, Yujia, WANG, Le, SHEPPARD, George S, MANTEI, Robert A, McDANIEL, Keith F, PRATT, John K, HOLMS, James H, LIU, Dachun, HASVOLD, Liza, McCLELLAN, William J, FIDANZE, Steven D, KATI, Warren M, WADA, Carol K
Year of Publication 31.01.2019
Get full text
Year of Publication 31.01.2019
Patent
BROMODOMAIN INHIBITORS
DAI, Yujia, WANG, Le, Kati, Warren M, SHEPPARD, George S, MANTEI, Robert A, Pratt, John K, HOLMS, James H, LIU, Dachun, MCCLELLAN, William J, FIDANZE, Steven D, WADA, Carol K, HASVOLD, Lisa, MCDANIEL, Keith F
Year of Publication 29.10.2018
Get full text
Year of Publication 29.10.2018
Patent
BROMODOMAIN INHIBITORS
DAI, Yujia, WANG, Le, SHEPPARD, George S, MANTEI, Robert A, PRATT, John K, HOLMS, James H, LIU, Dachun, MCCLELLAN, William J, FIDANZE, Steven D, KATI, Warren M, WADA, Carol K, HASVOLD, Lisa, MCDANIEL, Keith F
Year of Publication 20.10.2018
Get full text
Year of Publication 20.10.2018
Patent
BROMODOMAIN INHIBITORS
Fidanze, Steven D, Kati, Warren M, Sheppard, George S, Wada, Carol K, Wang, Le, McDaniel, Keith F, Holms, James H, Mantei, Robert A, Pratt, John K, McClellan, William J, Liu, Dachun, Dai, Yujia, Hasvold, Lisa
Year of Publication 18.10.2018
Get full text
Year of Publication 18.10.2018
Patent