Glutamate and GABA synthesis, release, transport and metabolism as targets for seizure control
Rowley, Nicole M., Madsen, Karsten K., Schousboe, Arne, Steve White, H.
Published in Neurochemistry international (01.09.2012)
Published in Neurochemistry international (01.09.2012)
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Journal Article
Selective mGAT2 (BGT-1) GABA Uptake Inhibitors: Design, Synthesis, and Pharmacological Characterization
Vogensen, Stine B, Jørgensen, Lars, Madsen, Karsten K, Borkar, Nrupa, Wellendorph, Petrine, Skovgaard-Petersen, Jonas, Schousboe, Arne, White, H. Steve, Krogsgaard-Larsen, Povl, Clausen, Rasmus P
Published in Journal of medicinal chemistry (14.03.2013)
Published in Journal of medicinal chemistry (14.03.2013)
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Journal Article
Cyclic analogs of galanin and neuropeptide Y by hydrocarbon stapling
Green, Brad R., Klein, Brian D., Lee, Hee-Kyoung, Smith, Misty D., Steve White, H., Bulaj, Grzegorz
Published in Bioorganic & medicinal chemistry (01.01.2013)
Published in Bioorganic & medicinal chemistry (01.01.2013)
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Journal Article
A tribute to Arne Schousboe's contributions to neurochemistry and his innovative and enduring research in GABA, glutamate, and brain energy metabolism
McKenna, Mary C, Sonnewald, Ursula, Waageptersen, Helle S, White, H Steve
Published in Journal of neurochemistry (26.08.2024)
Published in Journal of neurochemistry (26.08.2024)
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Journal Article
Conantokins: Peptide Antagonists of NMDA Receptors
Layer, Richard T, Wagstaff, John D, White, H Steve
Published in Current medicinal chemistry (01.12.2004)
Published in Current medicinal chemistry (01.12.2004)
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Journal Article
NAX 810-2, A Novel Galanin-Based Therapy for Epilepsy
Metcalf, Cameron, Klein, Brian, McDougle, Daniel, Zhang, Liuyin, Bulaj, Grzegorz, Steve White, H.
Published in Neuropeptides (Edinburgh) (01.10.2017)
Published in Neuropeptides (Edinburgh) (01.10.2017)
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Journal Article
Anticonvulsant neuropeptides as drug leads for neurological diseases
Robertson, Charles R, Flynn, Sean P, White, H Steve, Bulaj, Grzegorz
Published in Natural product reports (01.04.2011)
Published in Natural product reports (01.04.2011)
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Journal Article
Anticonvulsant effects of a galanin receptor 3 (galr3) antagonist SNAP 37889 in mouse models of seizures
Gagangras, Saurabh, Jill Dahle, E., Thomson, Kyle, Zhang, Luiyin, Metcalf, Cameron, Bulaj, Grzegorz, Steve White, H.
Published in Neuropeptides (Edinburgh) (01.10.2017)
Published in Neuropeptides (Edinburgh) (01.10.2017)
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Journal Article
Engineering Galanin Analogues That Discriminate between GalR1 and GalR2 Receptor Subtypes and Exhibit Anticonvulsant Activity following Systemic Delivery
Robertson, Charles R, Scholl, Erika Adkins, Pruess, Timothy H, Green, Brad R, White, H. Steve, Bulaj, Grzegorz
Published in Journal of medicinal chemistry (25.02.2010)
Published in Journal of medicinal chemistry (25.02.2010)
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Journal Article
Design, Synthesis, and Characterization of High-Affinity, Systemically-Active Galanin Analogues with Potent Anticonvulsant Activities
Bulaj, Grzegorz, Green, Brad R, Lee, Hee-Kyoung, Robertson, Charles R, White, Karen, Zhang, Liuyin, Sochanska, Marianna, Flynn, Sean P, Scholl, Erika Adkins, Pruess, Timothy H, Smith, Misty D, White, H. Steve
Published in Journal of medicinal chemistry (25.12.2008)
Published in Journal of medicinal chemistry (25.12.2008)
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Journal Article
Novel, Broad-Spectrum Anticonvulsants Containing a Sulfamide Group: Pharmacological Properties of (S)‑N‑[(6-Chloro-2,3-dihydrobenzo[1,4]dioxin-2-yl)methyl]sulfamide (JNJ-26489112)
McComsey, David F, Smith-Swintosky, Virginia L, Parker, Michael H, Brenneman, Douglas E, Malatynska, Ewa, White, H. Steve, Klein, Brian D, Wilcox, Karen S, Milewski, Michael E, Herb, Mark, Finley, Michael F. A, Liu, Yi, Lubin, Mary Lou, Qin, Ning, Reitz, Allen B, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (27.11.2013)
Published in Journal of medicinal chemistry (27.11.2013)
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Journal Article
Stapling Mimics Noncovalent Interactions of γ-Carboxyglutamates in Conantokins, Peptidic Antagonists of N-Methyl-d-Aspartic Acid Receptors
Platt, Randall J., Han, Tiffany S., Green, Brad R., Smith, Misty D., Skalicky, Jack, Gruszczyński, Paweł, White, H. Steve, Olivera, Baldomero, Bulaj, Grzegorz, Gajewiak, Joanna
Published in The Journal of biological chemistry (08.06.2012)
Published in The Journal of biological chemistry (08.06.2012)
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Journal Article
GABA transporters as drug targets for modulation of GABAergic activity
Schousboe, Arne, Sarup, Alan, Larsson, Orla M., White, H. Steve
Published in Biochemical pharmacology (15.10.2004)
Published in Biochemical pharmacology (15.10.2004)
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Journal Article
Conference Proceeding
Structural Requirements for a Lipoamino Acid in Modulating the Anticonvulsant Activities of Systemically Active Galanin Analogues
Zhang, Liuyin, Robertson, Charles R, Green, Brad R, Pruess, Timothy H, White, H. Steve, Bulaj, Grzegorz
Published in Journal of medicinal chemistry (12.03.2009)
Published in Journal of medicinal chemistry (12.03.2009)
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Journal Article
Conantokins Derived from the Asprella Clade Impart conRl-B, an N-Methyl d-Aspartate Receptor Antagonist with a Unique Selectivity Profile for NR2B Subunits
Gowd, Konkallu Hanumae, Han, Tiffany S, Twede, Vernon, Gajewiak, Joanna, Smith, Misty D, Watkins, Maren, Platt, Randall J, Toledo, Gabriela, White, H. Steve, Olivera, Baldomero M, Bulaj, Grzegorz
Published in Biochemistry (Easton) (12.06.2012)
Published in Biochemistry (Easton) (12.06.2012)
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Journal Article
Novel, Broad-Spectrum Anticonvulsants Containing a Sulfamide Group: Advancement of N-((Benzo[b]thien-3-yl)methyl)sulfamide (JNJ-26990990) into Human Clinical Studies
Parker, Michael H, Smith-Swintosky, Virginia L, McComsey, David F, Huang, Yifang, Brenneman, Douglas, Klein, Brian, Malatynska, Ewa, White, H. Steve, Milewski, Michael E, Herb, Mark, Finley, Michael F. A, Liu, Yi, Lubin, Mary Lou, Qin, Ning, Iannucci, Robert, Leclercq, Laurent, Cuyckens, Filip, Reitz, Allen B, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (10.12.2009)
Published in Journal of medicinal chemistry (10.12.2009)
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Journal Article