Design, synthesis, and in vitro and in vivo anti-angiogenesis study of a novel vascular endothelial growth factor receptor-2 (VEGFR-2) inhibitor based on 1,2,3-triazole scaffold
Wang, De-pu, Liu, Kai-li, Li, Xin-yang, Lu, Guo-qing, Xue, Wen-han, Qian, Xin-hua, Mohamed O, Kamara, Meng, Fan-hao
Published in European journal of medicinal chemistry (05.02.2021)
Published in European journal of medicinal chemistry (05.02.2021)
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Discovery of (quinazolin-6-yl)benzamide derivatives containing a 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline moiety as potent reversal agents against P-glycoprotein-mediated multidrug resistance
Xue, Wen-han, Liu, Kai-li, Zhang, Ting-jian, Dong, Gang, Wang, Jia-hui, Wang, Jing, Guo, Shuai, Hu, Jie, Zhang, Qing-yu, Li, Xin-yang, Meng, Fan-hao
Published in European journal of medicinal chemistry (15.01.2024)
Published in European journal of medicinal chemistry (15.01.2024)
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Discovery of novel thymidylate synthase (TS) inhibitors that influence cancer angiogenesis and metabolic reprogramming in NSCLC cells
Dong, Gang, Li, Yu-heng, Guo, Jing-si, Lin, Qi-qi, Deng, Mei-yan, Xue, Wen-han, Li, Xin-yang, Meng, Fan-hao
Published in European journal of medicinal chemistry (05.10.2023)
Published in European journal of medicinal chemistry (05.10.2023)
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Novel Allosteric Inhibitors of Deoxyhypusine Synthase against Malignant Melanoma: Design, Synthesis, and Biological Evaluation
Liu, Kai-li, Li, Xin-yang, Wang, De-pu, Xue, Wen-han, Qian, Xin-hua, Li, Yu-heng, Lin, Qi-qi, Li, Shuai, Meng, Fan-hao
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
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2-((1-Phenyl-1H-1,2,3-triazol-4-yl)methyl)-2-azabicyclo[3.2.1]octan-3-one derivatives: Simplification and modification of aconitine scaffold for the discovery of novel anticancer agents
Zhang, Yi, Zhang, Ting-jian, Li, Xin-yang, Liang, Jing-wei, Tu, Shun, Xu, Hai-li, Xue, Wen-han, Qian, Xin-hua, Zhang, Zhen-hao, Zhang, Xu, Meng, Fan-hao
Published in European journal of medicinal chemistry (15.01.2021)
Published in European journal of medicinal chemistry (15.01.2021)
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Synthesis and evaluation of novel HER-2 inhibitors to exert anti-breast cancer ability through epithelial-mesenchymal transition (EMT) pathway
Li, Xin-yang, Qian, Xin-hua, Zhu, Ju, Li, Yu-heng, Lin, Qi-qi, Li, Shuai, Xue, Wen-han, Jian, Ling-yan, Meng, Fan-hao
Published in European journal of medicinal chemistry (05.07.2022)
Published in European journal of medicinal chemistry (05.07.2022)
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Discovery of N-(1,3,4-thiadiazol-2-yl)benzamide derivatives containing a 6,7-methoxyquinoline structure as novel EGFR/HER-2 dual-target inhibitors against cancer growth and angiogenesis
Li, Xin-yang, Wang, De-pu, Li, Shuai, Xue, Wen-han, Qian, Xin-hua, Liu, Kai-li, Li, Yu-heng, Lin, Qi-qi, Dong, Gang, Meng, Fan-hao, Jian, Ling-yan
Published in Bioorganic chemistry (01.02.2022)
Published in Bioorganic chemistry (01.02.2022)
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Design, synthesis and biological evaluation of novel (E)-N-phenyl-4-(pyridine-acylhydrazone) benzamide derivatives as potential antitumor agents for the treatment of multiple myeloma (MM)
Li, Xin-yang, Li, Shuai, Lu, Guo-qing, Wang, De-pu, Liu, Kai-li, Qian, Xin-hua, Xue, Wen-han, Meng, Fan-hao
Published in Bioorganic chemistry (01.10.2020)
Published in Bioorganic chemistry (01.10.2020)
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