Adenosine Analogues as Selective Inhibitors of Glyceraldehyde-3-phosphate Dehydrogenase of Trypanosomatidae via Structure-Based Drug Design
Bressi, Jerome C, Verlinde, Christophe L. M. J, Aronov, Alex M, Shaw, My Le, Shin, Sam S, Nguyen, Lisa N, Suresh, Stephen, Buckner, Frederick S, Van Voorhis, Wesley C, Kuntz, Irwin D, Hol, Wim G. J, Gelb, Michael H
Published in Journal of medicinal chemistry (21.06.2001)
Published in Journal of medicinal chemistry (21.06.2001)
Get full text
Journal Article
Structure of a ribulose 5-phosphate 3-epimerase from Plasmodium falciparum
Caruthers, J., Bosch, J., Buckner, F., Van Voorhis, W., Myler, P., Worthey, E., Mehlin, C., Boni, E., DeTitta, G., Luft, J., Lauricella, A., Kalyuzhniy, O., Anderson, L., Zucker, F., Soltis, M., Hol, Wim G. J.
Published in Proteins, structure, function, and bioinformatics (01.02.2006)
Published in Proteins, structure, function, and bioinformatics (01.02.2006)
Get full text
Journal Article
Adenosine analogues as inhibitors of Trypanosoma brucei phosphoglycerate kinase: elucidation of a novel binding mode for a 2-amino-N(6)-substituted adenosine
Bressi, J C, Choe, J, Hough, M T, Buckner, F S, Van Voorhis, W C, Verlinde, C L, Hol, W G, Gelb, M H
Published in Journal of medicinal chemistry (02.11.2000)
Published in Journal of medicinal chemistry (02.11.2000)
Get full text
Journal Article
Protein farnesyl and N-myristoyl transferases: piggy-back medicinal chemistry targets for the development of antitrypanosomatid and antimalarial therapeutics
Gelb, Michael H., Van Voorhis, Wesley C., Buckner, Frederick S., Yokoyama, Kohei, Eastman, Richard, Carpenter, Elisabeth P., Panethymitaki, Chrysoula, Brown, Katherine A., Smith, Deborah F.
Published in Molecular & Biochemical Parasitology (01.02.2003)
Published in Molecular & Biochemical Parasitology (01.02.2003)
Get full text
Book Review
Journal Article
Trypanosome and Animal Lanosterol Synthases Use Different Catalytic Motifs
Joubert, Bridget M, Buckner, Frederick S, Matsuda, Seiichi P. T
Published in Organic letters (14.06.2001)
Published in Organic letters (14.06.2001)
Get full text
Journal Article
Protein farnesyltransferase from Trypanosoma brucei. A heterodimer of 61- and 65-kDa subunits as a new target for antiparasite therapeutics
Yokoyama, K. (University of Washington, Seattle, WA.), Trobridge, P, Buckner, F.S, Van Voorhis, W.C, Stuart, K.D, Gelb, M.H
Published in The Journal of biological chemistry (09.10.1998)
Published in The Journal of biological chemistry (09.10.1998)
Get full text
Journal Article
Cloning, heterologous expression, and substrate specificities of protein farnesyltransferases from Trypanosoma cruzi and Leishmania major
Buckner, Frederick S, Eastman, Richard T, Nepomuceno-Silva, José L, Speelmon, Emily C, Myler, Peter J, Van Voorhis, Wesley C, Yokoyama, Kohei
Published in Molecular and biochemical parasitology (01.07.2002)
Published in Molecular and biochemical parasitology (01.07.2002)
Get full text
Journal Article
Cloning, Heterologous Expression, and Distinct Substrate Specificity of Protein Farnesyltransferase from Trypanosoma brucei
Buckner, Frederick S., Yokoyama, Kohei, Nguyen, Lisa, Grewal, Anita, Erdjument-Bromage, Hediye, Tempst, Paul, Strickland, Corey L., Xiao, Li, Van Voorhis, Wesley C., Gelb, Michael H.
Published in The Journal of biological chemistry (21.07.2000)
Published in The Journal of biological chemistry (21.07.2000)
Get full text
Journal Article
The effects of protein farnesyltransferase inhibitors on trypanosomatids: inhibition of protein farnesylation and cell growth
Yokoyama, Kohei, Trobridge, Patty, Buckner, Frederick S, Scholten, Jeffrey, Stuart, Kenneth D, Van Voorhis, Wesley C, Gelb, Michael H
Published in Molecular and biochemical parasitology (01.07.1998)
Published in Molecular and biochemical parasitology (01.07.1998)
Get full text
Journal Article
Structures of Substrate- and Inhibitor-Bound Adenosine Deaminase from a Human Malaria Parasite Show a Dramatic Conformational Change and Shed Light on Drug Selectivity
Larson, Eric T., Deng, Wei, Krumm, Brian E., Napuli, Alberto, Mueller, Natascha, Van Voorhis, Wesley C., Buckner, Frederick S., Fan, Erkang, Lauricella, Angela, DeTitta, George, Luft, Joseph, Zucker, Frank, Hol, Wim G.J., Verlinde, Christophe L.M.J., Merritt, Ethan A.
Published in Journal of molecular biology (12.09.2008)
Published in Journal of molecular biology (12.09.2008)
Get full text
Journal Article
Expression of mammalian cytokines by Trypanosoma cruzi indicates unique signal sequence requirements and processing
La Flamme, Anne C., Buckner, Frederick S., Swindle, John, Ajioka, Janet, Van Voorhis, Wesley C.
Published in Molecular and biochemical parasitology (01.12.1995)
Published in Molecular and biochemical parasitology (01.12.1995)
Get full text
Journal Article
Crystal structures and proposed structural/functional classification of three protozoan proteins from the isochorismatase superfamily
Caruthers, Jonathan, Zucker, Frank, Worthey, Elizabeth, Myler, Peter J., Buckner, Fred, Van Voorhuis, Wes, Mehlin, Chris, Boni, Erica, Feist, Tiffany, Luft, Joseph, Gulde, Stacey, Lauricella, Angela, Kaluzhniy, Oleksandr, Anderson, Lori, Le Trong, Isolde, Holmes, Margaret A., Earnest, Thomas, Soltis, Michael, Hodgson, Keith O., Hol, Wim G.J., Merritt, Ethan A.
Published in Protein science (01.11.2005)
Published in Protein science (01.11.2005)
Get full text
Journal Article
TcRho1, a farnesylated Rho family homologue from Trypanosoma cruzi: cloning, trans-splicing, and prenylation studies
Nepomuceno-Silva, J L, Yokoyama, K, de Mello, L D, Mendonca, S M, Paixão, J C, Baron, R, Faye, J C, Buckner, F S, Van Voorhis, W C, Gelb, M H, Lopes, U G
Published in The Journal of biological chemistry (10.08.2001)
Published in The Journal of biological chemistry (10.08.2001)
Get full text
Journal Article
Protein Farnesyltransferase Inhibitors Exhibit Potent Antimalarial Activity
Nallan, Laxman, Bauer, Kevin D, Bendale, Pravin, Rivas, Kasey, Yokoyama, Kohei, Hornéy, Carolyn P, Pendyala, Prakash Rao, Floyd, David, Lombardo, Louis J, Williams, David K, Hamilton, Andrew, Sebti, Said, Windsor, William T, Weber, Patricia C, Buckner, Frederick S, Chakrabarti, Debopam, Gelb, Michael H, Van Voorhis, Wesley C
Published in Journal of medicinal chemistry (02.06.2005)
Published in Journal of medicinal chemistry (02.06.2005)
Get full text
Journal Article
Cloning and functional characterization of a Trypanosoma brucei lanosterol 14alpha-demethylase gene
Joubert, B M, Nguyen, L N, Matsuda, S P, Buckner, F S
Published in Molecular and biochemical parasitology (28.09.2001)
Get full text
Published in Molecular and biochemical parasitology (28.09.2001)
Journal Article