P2–P1′ macrocyclization of P2 phenylglycine based HCV NS3 protease inhibitors using ring-closing metathesis
Lampa, Anna, Ehrenberg, Angelica E., Vema, Aparna, Åkerblom, Eva, Lindeberg, Gunnar, Helena Danielson, U., Karlén, Anders, Sandström, Anja
Published in Bioorganic & medicinal chemistry (15.08.2011)
Published in Bioorganic & medicinal chemistry (15.08.2011)
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Discovery of achiral inhibitors of the hepatitis C virus NS3 protease based on 2(1 H)-pyrazinones
Örtqvist, Pernilla, Gising, Johan, Ehrenberg, Angelica E., Vema, Aparna, Borg, Anneli, Karlén, Anders, Larhed, Mats, Danielson, U. Helena, Sandström, Anja
Published in Bioorganic & medicinal chemistry (01.09.2010)
Published in Bioorganic & medicinal chemistry (01.09.2010)
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Journal Article
Improved P2 phenylglycine-based hepatitis C virus NS3 protease inhibitors with alkenylic prime-side substituents
Lampa, Anna, Ehrenberg, Angelica E., Gustafsson, Sofia S., Vema, Aparna, Åkerblom, Eva, Lindeberg, Gunnar, Karlén, Anders, Danielson, U. Helena, Sandström, Anja
Published in Bioorganic & medicinal chemistry (15.07.2010)
Published in Bioorganic & medicinal chemistry (15.07.2010)
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Three-dimensional quantitative structure (3-D QSAR) activity relationship studies on imidazolyl and N-pyrrolyl heptenoates as 3-hydroxy-3-methylglutaryl-CoA reductase (HMGR) inhibitors by comparative molecular similarity indices analysis (CoMSIA)
Thilagavathi, Ramasamy, Kumar, Raj, Aparna, Vema, Sobhia, M. Elizabeth, Gopalakrishnan, Bulusu, Chakraborti, Asit K.
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
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Design of EGFR kinase inhibitors: A ligand-based approach and its confirmation with structure-based studies
Vema, Aparna, Panigrahi, Sunil K., Rambabu, G., Gopalakrishnan, B., Sarma, J.A.R.P., Desiraju, Gautam R.
Published in Bioorganic & medicinal chemistry (15.10.2003)
Published in Bioorganic & medicinal chemistry (15.10.2003)
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