Aglycone exploration of C-arylglucoside inhibitors of renal sodium-dependent glucose transporter SGLT2
Ellsworth, Bruce A., Meng, Wei, Patel, Manorama, Girotra, Ravindar N., Wu, Gang, Sher, Philip M., Hagan, Deborah L., Obermeier, Mary T., Humphreys, William G., Robertson, James G., Wang, Aiying, Han, Songping, Waldron, Thomas L., Morgan, Nathan N., Whaley, Jean M., Washburn, William N.
Published in Bioorganic & medicinal chemistry letters (01.09.2008)
Published in Bioorganic & medicinal chemistry letters (01.09.2008)
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Carboxyl-promoted enhancement of selectivity for the β3 adrenergic receptor. Negative charge of the sulfonic acid BMS-187413 introduces β3 binding selectivity
SHER, P. M, MATHUR, A, FISHER, L. G, WU, G, SKWISH, S, MICHEL, I. M, SEILER, S. M, DICKINSON, K. E. J
Published in Bioorganic & medicinal chemistry letters (01.06.1997)
Published in Bioorganic & medicinal chemistry letters (01.06.1997)
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Carboxyl-promoted enhancement of selectivity for the β 3 adrenergic receptor. Negative charge of the sulfonic acid BMS-187413 introduces-β 3 binding selectivity
Sher, Philip M., Mathur, Arvind, Fisher, Liesl G., Wu, Gang, Skwish, Stephen, Michel, Inge M., Seiler, Steven M., Dickinson, Kenneth E.J.
Published in Bioorganic & medicinal chemistry letters (1997)
Published in Bioorganic & medicinal chemistry letters (1997)
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Thromboxane receptor antagonist BMS-180291: A new pre-clinical lead
Misra, Raj N., Brown, Baerbel R., Sher, Philip M., Patel, Manorama M., Hall, Steven E., Han, Wen-Ching, Barrish, Joel C., Floyd, David M., Sprague, Peter W., Morrison, Richard A., Ridgewell, Richard E., White, Ronald E., DiDonato, Gerald C., Harris, Don N., Hedberg, Anders, Schumacher, William A., Webb, Maria L., Ogletree, Martin L.
Published in Bioorganic & medicinal chemistry letters (1992)
Published in Bioorganic & medicinal chemistry letters (1992)
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Interphenylene 7-oxabicyclo[2.2.1]heptanes. SQ33,961: a new potent, long-acting thromboxane antagonist
Misra, Raj N., Brown, Baerbel R., Sher, Philip M., Patel, Manorama M., Goldenberg, Harold J., Michel, Inge M., Harris, Don N.
Published in Bioorganic & medicinal chemistry letters (1991)
Published in Bioorganic & medicinal chemistry letters (1991)
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