Regional brain uptake of the muscarinic ligand, [ 18F]FP-TZTP, is greatly decreased in M2 receptor knockout mice but not in M1, M3 and M4 receptor knockout mice
Jagoda, E.M., Kiesewetter, D.O., Shimoji, K., Ravasi, L., Yamada, M., Gomeza, J., Wess, J., Eckelman, W.C.
Published in Neuropharmacology (01.04.2003)
Published in Neuropharmacology (01.04.2003)
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Journal Article
Biologically stable [ 18F]-labeled benzylfluoride derivatives
Magata, Yasuhiro, Lang, Lixin, Kiesewetter, Dale O, Jagoda, Elaine M, Channing, Michael A, Eckelman, William C
Published in Nuclear medicine and biology (01.02.2000)
Published in Nuclear medicine and biology (01.02.2000)
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Journal Article
A review of new oncotropic tracers for pet imaging
Lang, L., Aloj, L., Kiesewetter, D.O., Jagoda, E., Lee, J.T., Paik, C.H., Carrasquillo, J.A., Eckelman, W.C.
Published in Nuclear medicine and biology (01.08.1996)
Published in Nuclear medicine and biology (01.08.1996)
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Journal Article
Conference Proceeding
Evaluation of stereoisomers of 4-fluoroalkyl analogues of 3-quinuclidinyl benzilate in in vivo competition studies for the M1, M2, and M3 muscarinic receptor subtypes in brain
Lee, Jaetae, Paik, Chang H., Kiesewetter, Dale O., Park, Seok G., Eckelman, William C.
Published in Nuclear medicine and biology (01.08.1995)
Published in Nuclear medicine and biology (01.08.1995)
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Journal Article
Syntheses and D2 receptor affinities of derivatives of spiperone containing aliphatic halogens
Kiesewetter, D O, Eckelman, W C, Cohen, R M, Finn, R D, Larson, S M
Published in International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes (1986)
Published in International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes (1986)
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Journal Article
Chronic neuropathic pain reduces opioid receptor availability with associated anhedonia in rat
Thompson, Scott J, Pitcher, Mark H, Stone, Laura S, Tarum, Farid, Niu, Gang, Chen, Xiaoyuan, Kiesewetter, Dale O, Schweinhardt, Petra, Bushnell, M Catherine
Published in Pain (Amsterdam) (01.09.2018)
Published in Pain (Amsterdam) (01.09.2018)
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Journal Article
Using single photon emission tomography (SPECT) and positron emission tomography (PET) to trace the distribution of muscarinic acetylcholine receptor (MACHR) binding radioligands
Kiesewetter, Dale O., Carson, Richard E., Jagoda, Elaine M., Herscovitch, Peter, Eckelman, William C.
Published in Life sciences (1973) (1999)
Published in Life sciences (1973) (1999)
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Journal Article
In vivo muscarinic binding selectivity of (R,S)- and (R,R)-[18F]-fluoromethyl QNB
Kiesewetter, D O, Carson, R E, Jagoda, E M, Endres, C J, Der, M G, Herscovitch, P, Eckelman, W C
Published in Bioorganic & medicinal chemistry (01.08.1997)
Published in Bioorganic & medicinal chemistry (01.08.1997)
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Journal Article
Characterization of the uptake of 16 alpha-([18F]fluoro)-17 beta-estradiol in DMBA-induced mammary tumors
Mathias, C J, Welch, M J, Katzenellenbogen, J A, Brodack, J W, Kilbourn, M R, Carlson, K E, Kiesewetter, D O
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1987)
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1987)
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Journal Article
Fluoro-, bromo-, and iodopaclitaxel derivatives: synthesis and biological evaluation
Kiesewetter, Dale O, Jagoda, Elaine M, Kao, Chih-Hao K, Ma, Ying, Ravasi, Laura, Shimoji, Kazuaki, Szajek, Lawrence P, Eckelman, William C
Published in Nuclear medicine and biology (2003)
Published in Nuclear medicine and biology (2003)
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Journal Article
Liquid chromatography–tandem mass spectrometry identification of metabolites of three phenylcarboxyl derivatives of the 5-HT1A antagonist, N-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-N-(2-pyridyl) trans-4-fluorocyclohexanecarboxamide (FCWAY), produced by human and rat hepatocytes
Ma, Ying, Lang, Lixin, Kiesewetter, Dale O, Eckelman, William C
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.11.2002)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (15.11.2002)
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Journal Article
The automated radiosynthesis of [ 18F]FP-TZTP
Kiesewetter, Dale O, Vuong, Bik-kee, Channing, Michael A
Published in Nuclear medicine and biology (2003)
Published in Nuclear medicine and biology (2003)
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Journal Article
Purification of the precursor for the automated radiosynthesis of [ [formula omitted]]FCWAY by counter-current chromatography
Ma, Ying, Lang, Lixin, Kiesewetter, Dale O, Vuong, Bik-Kee, Channing, Michael, Ito, Yoichiro, Eckelman, William C
Published in Journal of Chromatography A (23.04.2004)
Published in Journal of Chromatography A (23.04.2004)
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Journal Article
Determination of [ 18F]FCWAY, [ 18F]FP-TZTP, and their metabolites in plasma using rapid and efficient liquid-liquid and solid phase extractions
Ma, Ying, Kiesewetter, Dale O, Lang, Lixin, Der, Margaret, Huang, Bill, Carson, Richard E, Eckelman, William C
Published in Nuclear medicine and biology (01.04.2003)
Published in Nuclear medicine and biology (01.04.2003)
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Journal Article
Identification of metabolites of fluorine-18-labeled M2 muscarinic receptor agonist, 3-(3-[(3-fluoropropyl)thio]-1,2,5-thiadiazol-4-yl)-1,2,5,6-tetrahydro-1-methylpyridine, produced by human and rat hepatocytes
Ma, Ying, Kiesewetter, Dale O, Jagoda, Elaine M, Huang, Bill X, Eckelman, William C
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (25.01.2002)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (25.01.2002)
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Journal Article
Routine quality control of recycled target [ 18O]water by capillary electrophoresis and gas chromatography
Huang, Bill X., Channing, Michael A., Plascjak, Paul S., Kiesewetter, Dale O., Der, Margaret, Ma, Ying, Eckelman, William C.
Published in Nuclear medicine and biology (01.10.2003)
Published in Nuclear medicine and biology (01.10.2003)
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Journal Article
Radiochemical synthesis and biodistribution of a novel maxi-K potassium channel opener
Kiesewetter, Dale O, Jagoda, Elaine M, Starrett, John E, Gribkoff, Valentin K, Hewawasam, Piyasena, Srinivas, Nugahally, Salazar, Daniel, Eckelman, William C
Published in Nuclear medicine and biology (2002)
Published in Nuclear medicine and biology (2002)
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Journal Article
Characterization of the uptake of 16α-([ 18F]fluoro)-17β-estradiol in DMBA-induced mammary tumors
Mathias, Carla J., Welch, Michael J., Katzenellenbogen, John A., Brodack, James W., Kilbourn, Michael R., Carlson, Kathryn E., Kiesewetter, Dale O.
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1987)
Published in International journal of radiation applications and instrumentation. Part B, Nuclear medicine and biology (1987)
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Journal Article