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Published in Bioorganic & medicinal chemistry letters (01.08.2017)
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
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Imidazo[2,1- b]thiazoles: Multitargeted inhibitors of both the insulin-like growth factor receptor and members of the epidermal growth factor family of receptor tyrosine kinases
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Published in Bioorganic & medicinal chemistry letters (15.04.2010)
Published in Bioorganic & medicinal chemistry letters (15.04.2010)
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Biaryl amide glucagon receptor antagonists
KURUKULASURIYA, Ravi, SORENSEN, Bryan K, ADLER, Andrew L, COLLINS, Christine A, LINK, James T, PATEL, Jyoti R, JAE, Hwan-Soo, WINN, Marty X, ROHDE, Jeffrey R, GRIHALDE, Nelson D, LIN, Chun W, OGIELA, Christopher A
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Discovery of novel nonsteroidal glucocorticoid receptor modulators
LINK, J. T, SORENSEN, Bryan K, PATEL, Jyoti, EMERY, Maurice, GRYNFARB, Marlena, GOOS-NILSSON, Annika
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Synthesis, activity, metabolic stability, and pharmacokinetics of glucocorticoid receptor modulator–statin hybrids
Link, J.T, Sorensen, Bryan K, Lai, Chunqiu, Wang, Jiahong, Fung, Steven, Deng, Daisy, Emery, Maurice, Carroll, Sherry, Grynfarb, Marlena, Goos-Nilsson, Annika, von Geldern, Thomas
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Optimization and metabolic stabilization of a class of nonsteroidal glucocorticoid modulators
Link, J.T, Sorensen, Bryan K, Patel, Jyoti, Arendsen, David, Li, Gaoquan, Swanson, Susan, Nguyen, Bach, Emery, Maurice, Grynfarb, Marlena, Goos-Nilsson, Annika
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Bile acid conjugates of a nonsteroidal glucocorticoid receptor modulator
Tu, Noah, Link, J.T, Sorensen, Bryan K, Emery, Maurice, Grynfarb, Marlena, Goos-Nilsson, Annika, Nguyen, Bach
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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An Evaluation of a C-Glucuronide as a liver targeting group: conjugate of a glucocorticoid antagonist
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Published in Bioorganic & medicinal chemistry letters (21.07.2003)
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
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Discovery of a series of pyrrolidine-based endothelin receptor antagonists with enhanced ET A receptor selectivity
Boyd, Steven A, Mantei, Robert A, Tasker, Andrew S, Liu, Gang, Sorensen, Bryan K, Henry Jr, Kenneth J, von Geldern, Thomas W, Winn, Martin, Wu-Wong, Jinshyun R, Chiou, William J, Dixon, Douglas B, Hutchins, Charles W, Marsh, Kennan C, Nguyen, Bach, Opgenorth, Terry J
Published in Bioorganic & medicinal chemistry (01.06.1999)
Published in Bioorganic & medicinal chemistry (01.06.1999)
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Discovery of a series of pyrrolidine-based endothelin receptor antagonists with enhanced ETA receptor selectivity
BOYD, S. A, MANTEI, R. A, DIXON, D. B, HUTCHINS, C. W, MARSH, K. C, NGUYEN, B, OPGENORTH, T. J, TASKER, A. S, GANG LIU, SORENSEN, B. K, HENRY, K. J, VON GELDERN, T. W, WINN, M, WU-WONG, J. R, CHIOU, W. J
Published in Bioorganic & medicinal chemistry (01.06.1999)
Published in Bioorganic & medicinal chemistry (01.06.1999)
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Synthesis and In Vitro evaluation of fused ring heterocyle-containing angiotensin II antagonists
Zydowsky, Thomas M., Winn, Martin, De, Biswanath, Condon, Stephen L., Altenbach, Robert J., Basha, Fatima Z., Boyd, Steven A., Buckner, Steven A., Hancock, Arthur A., Lee, Jang Y., Mantei, Robert A., Novosad, Eugene I., Sorensen, Bryan K., Tasker, Andrew S., Shiosaki, Kazumi, Kerkman, Daniel J., Opgenorth, Terry J., DeBernardis, John F.
Published in Bioorganic & medicinal chemistry letters (1994)
Published in Bioorganic & medicinal chemistry letters (1994)
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[ 3H]A-81988, a potent, selective, competitive antagonist radioligand for angiotensin AT 1 receptors
Hancock, Arthur A., Surber, Bruce W., Rotert, Gary, Thomas, Samuel, Tasker, Andrew S., Sorensen, Bryan K., Vodenlich, Alex D., Opgenorth, Terry J., Kerkman, Daniel J., DeBernardis, John F.
Published in European journal of pharmacology. Molecular pharmacology section (1994)
Published in European journal of pharmacology. Molecular pharmacology section (1994)
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[3H]A-81988, a potent, selective, competitive antagonist radioligand for angiotensin AT1 receptors
HANCOCK, A. A, SURBER, B. W, ROTERT, G, THOMAS, S, TASKER, A. S, SORENSEN, B. K, VODENLICH, A. D, OPGENORTH, T. J, KERKMAN, D. J, DEBERNARDIS, J. F
Published in European journal of pharmacology. Molecular pharmacology section (15.03.1994)
Published in European journal of pharmacology. Molecular pharmacology section (15.03.1994)
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