Heterocyclic ketones as inhibitors of histone deacetylase
Vasudevan, Anil, Ji, Zhiqin, Frey, Robin R., Wada, Carol K., Steinman, Douglas, Heyman, H.Robin, Guo, Yan, Curtin, Michael L., Guo, Jun, Li, Junling, Pease, Lori, Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
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Trifluoromethyl ketones as inhibitors of histone deacetylase
Frey, Robin R., Wada, Carol K., Garland, Robert B., Curtin, Michael L., Michaelides, Michael R., Li, Junling, Pease, Lori J., Glaser, Keith B., Marcotte, Patrick A., Bouska, Jennifer J., Murphy, Shannon S., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
Published in Bioorganic & medicinal chemistry letters (02.12.2002)
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α-Keto amides as inhibitors of histone deacetylase
Wada, Carol K., Frey, Robin R., Ji, Zhiqin, Curtin, Michael L., Garland, Robert B., Holms, James H., Li, Junling, Pease, Lori J., Guo, Jun, Glaser, Keith B., Marcotte, Patrick A., Richardson, Paul L., Murphy, Shannon S., Bouska, Jennifer J., Tapang, Paul, Magoc, Terrance J., Albert, Daniel H., Davidsen, Steven K., Michaelides, Michael R.
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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Biaryl Ether Retrohydroxamates as Potent, Long-lived, Orally Bioavailable MMP Inhibitors
Michaelides, Michael R., Dellaria, Joseph F., Gong, Jane, Holms, James H., Bouska, Jennifer J., Stacey, Jamie, Wada, Carol K., Heyman, H.Robin, Curtin, Michael L., Guo, Yan, Goodfellow, Carole L., Elmore, Ildiko B., Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770
Curtin, Michael L., Florjancic, Alan S., Heyman, H.Robin, Michaelides, Michael R., Garland, Robert B., Holms, James H., Steinman, Douglas H., Dellaria, Joseph F., Gong, Jane, Wada, Carol K., Guo, Yan, Elmore, Ildiko B., Tapang, Paul, Albert, Daniel H., Magoc, Terrance J., Marcotte, Patrick A., Bouska, Jennifer J., Goodfellow, Carole L., Bauch, Joy L., Marsh, Kennan C., Morgan, Douglas W., Davidsen, Steven K.
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
Published in Bioorganic & medicinal chemistry letters (18.06.2001)
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Journal Article
Methylpyrrole inhibitors of BET bromodomains
Hasvold, Lisa A., Sheppard, George S., Wang, Le, Fidanze, Steven D., Liu, Dachun, Pratt, John K., Mantei, Robert A., Wada, Carol K., Hubbard, Robbert, Shen, Yu, Lin, Xiaoyu, Huang, Xiaoli, Warder, Scott E., Wilcox, Denise, Li, Leiming, Buchanan, F. Greg, Smithee, Lauren, Albert, Daniel H., Magoc, Terrance J., Park, Chang H., Petros, Andrew M., Panchal, Sanjay C., Sun, Chaohong, Kovar, Peter, Soni, Nirupama B., Elmore, Steven W., Kati, Warren M., McDaniel, Keith F.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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