Microwave assisted synthesis: a new technology in drug discovery
Santagada, V, Frecentese, F, Perissutti, E, Fiorino, F, Severino, B, Caliendo, G
Published in Mini reviews in medicinal chemistry (01.03.2009)
Published in Mini reviews in medicinal chemistry (01.03.2009)
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Journal Article
Derivatives as 5HT1A Receptor Ligands-Past and Present
CALIENDO, G, SANTAGADA, V, PERISSUTTI, E, FIORINO, F
Published in Current medicinal chemistry (2005)
Published in Current medicinal chemistry (2005)
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Journal Article
Synthesis of phenylpyrimidinones as guanylyl cyclase C inhibitors
Magli, E., Fiorino, F., Severino, B., Corvino, A., Perissutti, E., Frecentese, F., Giordano, F., Saccone, Luciano, P., Zaminelli, T., Santagada, Caliendo, G., de Nucci, G.
Published in Pharmazie (01.01.2019)
Published in Pharmazie (01.01.2019)
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Journal Article
Racemic synthesis and solid phase peptide synthesis application of the chimeric valine/leucine derivative 2-amino-3,3,4-trimethyl-pentanoic acid
Pelà, Zoppo, L. Del, Allegri, Marzola, Trapella, Ruzza, Calo, Perissutti, Frecentese, Salvadori, Guerrini
Published in Pharmazie (01.07.2014)
Published in Pharmazie (01.07.2014)
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Journal Article
Recent advances in synthesis of PAR ligands as therapeutic strategy for inflammatory diseases
Severino, B, Santagada, V, Perissutti, E, Fiorino, F, Frecentese, F, De Angelis, F, Esposito, A, Caliendo, G
Published in Mini reviews in medicinal chemistry (01.06.2009)
Published in Mini reviews in medicinal chemistry (01.06.2009)
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Journal Article
Synthesis and in vitro pharmacological evaluation of a new series of 5-HT1A 5-HT2A and 5-HT2C receptor ligands containing a norbornene nucleus
Fiorino, F., Severino, B., De Angelis, F., Perissutti, E., Magli, E., Frecentese, F., Esposito, A., Massarelli, P., Nencini, C., Viti, B., Santagada, V., Caliendo, G.
Published in Pharmazie (01.09.2009)
Published in Pharmazie (01.09.2009)
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Journal Article
In vitro mutagenicity of anti-inflammatory parsalmide analogues PA7, PA10, and PA31 triggered by biotransformation into hydroxy derivatives
Cardoso, H.S., Bicalho, B., Genari, P., Santagada, V., Caliendo, G., Perissutti, E., Donato, J.L., De Nucci, G.
Published in European journal of medicinal chemistry (01.03.2006)
Published in European journal of medicinal chemistry (01.03.2006)
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Journal Article
Comparative bioavailability of two losartan formulations in healthy human volunteers after a single dose administration
Oliveira, C H, Medeiros Silva, R, Santagada, V, Caliendo, G, Perissutti, E, Prado Galuppo, M, Marcondes Rezende, V, Barrientos-Astigarraga, R E, Mendes, G Duarte, De Nucci, G
Published in International journal of clinical pharmacology and therapeutics (01.03.2006)
Published in International journal of clinical pharmacology and therapeutics (01.03.2006)
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Journal Article
Human Tissue Kallikrein S1 Subsite Recognition of Non-Natural Basic Amino Acids
Melo, Robson L, Barbosa Pozzo, Roseli C, Pimenta, Daniel C, Perissutti, Elisa, Caliendo, Giuseppe, Santagada, Vincenzo, Juliano, Luiz, Juliano, Maria A
Published in Biochemistry (Easton) (01.05.2001)
Published in Biochemistry (Easton) (01.05.2001)
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Journal Article
Synthesis and in vitro activities of NK-1 antagonists derived from L-tryptophan
Caliendo, G, Fiorino, F, Grieco, P, Perissutti, E, Santagada, Calignano, A, Mancuso, F, Albrizio, S
Published in Farmaco (Società chimica italiana : 1989) (01.10.1997)
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Published in Farmaco (Società chimica italiana : 1989) (01.10.1997)
Journal Article
New 5-hydroxytryptamine(1A) receptor ligands containing a norbornene nucleus: Synthesis and in vitro pharmacological evaluation
Fiorino, F, Perissutti, E, Severino, B, Santagada, Cirillo, D, Terracciano, S, Massarelli, P, Bruni, G, Collavoli, E, Renner, C, Caliendo, G
Published in Journal of medicinal chemistry (25.08.2005)
Published in Journal of medicinal chemistry (25.08.2005)
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Journal Article
Synthesis and in vitro activities of highly potent and selective tripeptide antagonists of the neurokinin NK-1 receptor
Caliendo, G, Greco, G, Grieco, P, Perissutti, E, Santagada, Calignano, N, Mancuso, F, Novellino, E
Published in Farmaco (Società chimica italiana : 1989) (01.11.1995)
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Published in Farmaco (Società chimica italiana : 1989) (01.11.1995)
Journal Article
Modification of the potent peptide FK888 with unusual aminoacids: Effects on activity on neurokinin receptors
Caliendo, G, Greco, G, Grieco, P, Perissutti, E, Santagada, Calignano, A, Mancuso, F, Novellino, E
Published in Farmaco (Società chimica italiana : 1989) (01.03.1996)
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Published in Farmaco (Società chimica italiana : 1989) (01.03.1996)
Journal Article
Synthesis by microwave irradiation of a substituted benzoxazine parallel library with preferential relaxant activity for guinea pig trachealis
Caliendo, Giuseppe, Perissutti, Elisa, Santagada, Vincenzo, Fiorino, Ferdinando, Severino, Beatrice, Cirillo, Donatella, d’Emmanuele di Villa Bianca, Roberta, Lippolis, Laura, Pinto, Aldo, Sorrentino, Raffaella
Published in European journal of medicinal chemistry (01.10.2004)
Published in European journal of medicinal chemistry (01.10.2004)
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Journal Article
SYNTHESIS AND NEUROKININ ANTAGONIST ACTIVITY OF 2-BENZYLIDENE- AND 2-BENZYL-3-BENZYLAMINO QUINUCLIDINES
CALIENDO, G, GRECO, G, PERISSUTTI, E, SANTAGADA, SILIPO, C, VITTORIA, A, TURBANTI, L, RENZETTI, AR, BENEDETTI, E, PEDONE, C, SANTINI, A
Published in Farmaco (Società chimica italiana : 1989) (01.10.1993)
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Published in Farmaco (Società chimica italiana : 1989) (01.10.1993)
Journal Article
Synthesis of 6beta-D-glucosyl and 6-nitroxy (-)-galanthamine derivatives as acetylcholinesterase inhibitors
Perissutti, E, Fiorino, F, Severino, B, Frecentese, F, Massarelli, P, Nencini, C, Santagada, V, Caliendo, G
Published in Pharmazie (01.06.2007)
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Published in Pharmazie (01.06.2007)
Journal Article
Synthesis and muscarinic receptor binding profiles of antagonist benzotriazole derivatives
Cappello, B, Greco, G, Novellino, E, Perissutti, E, Santagada, V, Silipo, C, Vittoria, A, Di Carlo, R, Meli, R, Muccioli, G
Published in Farmaco (Società chimica italiana : 1989) (01.07.1993)
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Published in Farmaco (Società chimica italiana : 1989) (01.07.1993)
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