The Catalytic Mechanism of Human Parainfluenza Virus Type 3 Haemagglutinin-Neuraminidase Revealed
Dirr, Larissa, El-Deeb, Ibrahim M., Guillon, Patrice, Carroux, Cindy J., Chavas, Leonard M. G., von Itzstein, Mark
Published in Angewandte Chemie (International ed.) (02.03.2015)
Published in Angewandte Chemie (International ed.) (02.03.2015)
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Neurodegenerative Disease Treatment Drug PBT2 Breaks Intrinsic Polymyxin Resistance in Gram-Positive Bacteria
De Oliveira, David M P, Keller, Bernhard, Hayes, Andrew J, Ong, Cheryl-Lynn Y, Harbison-Price, Nichaela, El-Deeb, Ibrahim M, Li, Gen, Keller, Nadia, Bohlmann, Lisa, Brouwer, Stephan, Turner, Andrew G, Cork, Amanda J, Jones, Thomas R, Paterson, David L, McEwan, Alastair G, Davies, Mark R, McDevitt, Christopher A, Itzstein, Mark von, Walker, Mark J
Published in Antibiotics (Basel) (25.03.2022)
Published in Antibiotics (Basel) (25.03.2022)
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Cross-species malaria immunity induced by chemically attenuated parasites
Good, Michael F, Reiman, Jennifer M, Rodriguez, I Bibiana, Ito, Koichi, Yanow, Stephanie K, El-Deeb, Ibrahim M, Batzloff, Michael R, Stanisic, Danielle I, Engwerda, Christian, Spithill, Terry, Hoffman, Stephen L, Lee, Moses, McPhun, Virginia
Published in The Journal of clinical investigation (01.08.2013)
Published in The Journal of clinical investigation (01.08.2013)
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Journal Article
Chemical Synergy between Ionophore PBT2 and Zinc Reverses Antibiotic Resistance
Bohlmann, Lisa, De Oliveira, David M P, El-Deeb, Ibrahim M, Brazel, Erin B, Harbison-Price, Nichaela, Ong, Cheryl-Lynn Y, Rivera-Hernandez, Tania, Ferguson, Scott A, Cork, Amanda J, Phan, Minh-Duy, Soderholm, Amelia T, Davies, Mark R, Nimmo, Graeme R, Dougan, Gordon, Schembri, Mark A, Cook, Gregory M, McEwan, Alastair G, von Itzstein, Mark, McDevitt, Christopher A, Walker, Mark J
Published in mBio (11.12.2018)
Published in mBio (11.12.2018)
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Targeting Human Parainfluenza Virus Type-1 Haemagglutinin-Neuraminidase with Mechanism-Based Inhibitors
Eveno, Tanguy, Dirr, Larissa, El-Deeb, Ibrahim M, Guillon, Patrice, von Itzstein, Mark
Published in Viruses (05.05.2019)
Published in Viruses (05.05.2019)
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Discovery of Cofactor Competitive Inhibitors against the Human Methyltransferase Fibrillarin
Shi, Yun, El-Deeb, Ibrahim M, Masic, Veronika, Hartley-Tassell, Lauren, Maggioni, Andrea, Itzstein, Mark von, Ve, Thomas
Published in Pharmaceuticals (Basel, Switzerland) (24.12.2021)
Published in Pharmaceuticals (Basel, Switzerland) (24.12.2021)
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Curcumin⁻Copper Complex Nanoparticles for the Management of Triple-Negative Breast Cancer
Greish, Khaled, Pittalà, Valeria, Taurin, Sebastien, Taha, Safa, Bahman, Fatemah, Mathur, Aanchal, Jasim, Anfal, Mohammed, Fatima, El-Deeb, Ibrahim M, Fredericks, Salim, Rashid-Doubell, Fiza
Published in Nanomaterials (Basel, Switzerland) (01.11.2018)
Published in Nanomaterials (Basel, Switzerland) (01.11.2018)
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Journal Article
Multiple Bactericidal Mechanisms of the Zinc Ionophore PBT2
Harbison-Price, Nichaela, Ferguson, Scott A, Heikal, Adam, Taiaroa, George, Hards, Kiel, Nakatani, Yoshio, Rennison, David, Brimble, Margaret A, El-Deeb, Ibrahim M, Bohlmann, Lisa, McDevitt, Christopher A, von Itzstein, Mark, Walker, Mark J, Cook, Gregory M
Published in mSphere (18.03.2020)
Published in mSphere (18.03.2020)
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Design, synthesis and biological evaluation of new potent and highly selective ROS1-tyrosine kinase inhibitor
Park, Byung Sun, El-Deeb, Ibrahim M., Yoo, Kyung Ho, Oh, Chang-Hyun, Cho, Seung Joo, Han, Dong Keun, Lee, Hye-Seung, Lee, Jae Yeol, Lee, So Ha
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Journal Article
Repurposing the Ionophore, PBT2, for Treatment of Multidrug-Resistant Neisseria gonorrhoeae Infections
Jen, Freda E-C, Edwards, Jennifer L, El-Deeb, Ibrahim M, Walker, Mark J, von Itzstein, Mark, Jennings, Michael P
Published in Antimicrobial agents and chemotherapy (20.09.2022)
Published in Antimicrobial agents and chemotherapy (20.09.2022)
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New antiviral approaches for human parainfluenza: Inhibiting the haemagglutinin-neuraminidase
Chibanga, Vimbaishe P., Dirr, Larissa, Guillon, Patrice, El-Deeb, Ibrahim M., Bailly, Benjamin, Thomson, Robin J., von Itzstein, Mark
Published in Antiviral research (01.07.2019)
Published in Antiviral research (01.07.2019)
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Journal Article
A drug candidate for Alzheimer’s and Huntington’s disease, PBT2, can be repurposed to render Neisseria gonorrhoeae susceptible to natural cationic antimicrobial peptides
Jen, Freda E -C, El-Deeb, Ibrahim M, Zalucki, Yaramah M, Edwards, Jennifer L, Walker, Mark J, von Itzstein, Mark, Jennings, Michael P
Published in Journal of antimicrobial chemotherapy (11.10.2021)
Published in Journal of antimicrobial chemotherapy (11.10.2021)
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Journal Article
Dysregulation of Streptococcus pneumoniae zinc homeostasis breaks ampicillin resistance in a pneumonia infection model
Brazel, Erin B., Tan, Aimee, Neville, Stephanie L., Iverson, Amy R., Udagedara, Saumya R., Cunningham, Bliss A., Sikanyika, Mwilye, De Oliveira, David M.P., Keller, Bernhard, Bohlmann, Lisa, El-Deeb, Ibrahim M., Ganio, Katherine, Eijkelkamp, Bart A., McEwan, Alastair G., von Itzstein, Mark, Maher, Megan J., Walker, Mark J., Rosch, Jason W., McDevitt, Christopher A.
Published in Cell reports (Cambridge) (11.01.2022)
Published in Cell reports (Cambridge) (11.01.2022)
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Journal Article
Repurposing a neurodegenerative disease drug to treat Gram-negative antibiotic-resistant bacterial sepsis
De Oliveira, David M P, Bohlmann, Lisa, Conroy, Trent, Jen, Freda E-C, Everest-Dass, Arun, Hansford, Karl A, Bolisetti, Raghu, El-Deeb, Ibrahim M, Forde, Brian M, Phan, Minh-Duy, Lacey, Jake A, Tan, Aimee, Rivera-Hernandez, Tania, Brouwer, Stephan, Keller, Nadia, Kidd, Timothy J, Cork, Amanda J, Bauer, Michelle J, Cook, Gregory M, Davies, Mark R, Beatson, Scott A, Paterson, David L, McEwan, Alastair G, Li, Jian, Schembri, Mark A, Blaskovich, Mark A T, Jennings, Michael P, McDevitt, Christopher A, von Itzstein, Mark, Walker, Mark J
Published in Science translational medicine (18.11.2020)
Published in Science translational medicine (18.11.2020)
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Journal Article
A dual drug regimen synergistically blocks human parainfluenza virus infection
Bailly, Benjamin, Dirr, Larissa, El-Deeb, Ibrahim M., Altmeyer, Ralf, Guillon, Patrice, von Itzstein, Mark
Published in Scientific reports (07.04.2016)
Published in Scientific reports (07.04.2016)
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Journal Article
Structure-guided discovery of potent and dual-acting human parainfluenza virus haemagglutinin–neuraminidase inhibitors
Guillon, Patrice, Dirr, Larissa, El-Deeb, Ibrahim M., Winger, Moritz, Bailly, Benjamin, Haselhorst, Thomas, Dyason, Jeffrey C., von Itzstein, Mark
Published in Nature communications (20.10.2014)
Published in Nature communications (20.10.2014)
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Journal Article
Exploring Human Parainfluenza Virus Type‑1 Hemagglutinin–Neuraminidase as a Target for Inhibitor Discovery
El-Deeb, Ibrahim M, Guillon, Patrice, Winger, Moritz, Eveno, Tanguy, Haselhorst, Thomas, Dyason, Jeffrey C, von Itzstein, Mark
Published in Journal of medicinal chemistry (25.09.2014)
Published in Journal of medicinal chemistry (25.09.2014)
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