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Published in Journal of organic chemistry (17.11.2023)
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Imidazo[2,1- b]thiazoles: Multitargeted inhibitors of both the insulin-like growth factor receptor and members of the epidermal growth factor family of receptor tyrosine kinases
Fidanze, Steve D., Erickson, Scott A., Wang, Gary T., Mantei, Robert, Clark, Richard F., Sorensen, Bryan K., Bamaung, Nwe Y., Kovar, Peter, Johnson, Eric F., Swinger, Kerren K., Stewart, Kent D., Zhang, Qian, Tucker, Lora A., Pappano, William N., Wilsbacher, Julie L., Wang, Jieyi, Sheppard, George S., Bell, Randy L., Davidsen, Steven K., Hubbard, Robert D.
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Published in Bioorganic & medicinal chemistry letters (15.04.2010)
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Potent and Selective Non-Benzodioxole-Containing Endothelin-A Receptor Antagonists
Tasker, Andrew S, Sorensen, Bryan K, Jae, Hwan-Soo, Winn, Martin, von Geldern, Thomas W, Dixon, Douglas B, Chiou, William J, Dayton, Brian D, Calzadila, Samuel, Hernandez, Lisa, Marsh, Kennan C, WuWong, J. Ruth, Opgenorth, Terry J
Published in Journal of medicinal chemistry (31.01.1997)
Published in Journal of medicinal chemistry (31.01.1997)
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Biaryl amide glucagon receptor antagonists
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Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Discovery of novel nonsteroidal glucocorticoid receptor modulators
LINK, J. T, SORENSEN, Bryan K, PATEL, Jyoti, EMERY, Maurice, GRYNFARB, Marlena, GOOS-NILSSON, Annika
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Synthesis, activity, metabolic stability, and pharmacokinetics of glucocorticoid receptor modulator–statin hybrids
Link, J.T, Sorensen, Bryan K, Lai, Chunqiu, Wang, Jiahong, Fung, Steven, Deng, Daisy, Emery, Maurice, Carroll, Sherry, Grynfarb, Marlena, Goos-Nilsson, Annika, von Geldern, Thomas
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Optimization and metabolic stabilization of a class of nonsteroidal glucocorticoid modulators
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Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Bile acid conjugates of a nonsteroidal glucocorticoid receptor modulator
Tu, Noah, Link, J.T, Sorensen, Bryan K, Emery, Maurice, Grynfarb, Marlena, Goos-Nilsson, Annika, Nguyen, Bach
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Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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2,4-Diarylpyrrolidine-3-carboxylic AcidsPotent ETA Selective Endothelin Receptor Antagonists. 1. Discovery of A-127722
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Published in Journal of medicinal chemistry (01.03.1996)
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An Evaluation of a C-Glucuronide as a liver targeting group: conjugate of a glucocorticoid antagonist
Sorensen, Bryan K., Link, J.T., von Geldern, Thomas, Emery, Maurice, Wang, Jiahong, Hickman, Bach, Grynfarb, Marlena, Goos-Nilsson, Annika, Carroll, Sherry
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
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Boyd, Steven A, Mantei, Robert A, Tasker, Andrew S, Liu, Gang, Sorensen, Bryan K, Henry Jr, Kenneth J, von Geldern, Thomas W, Winn, Martin, Wu-Wong, Jinshyun R, Chiou, William J, Dixon, Douglas B, Hutchins, Charles W, Marsh, Kennan C, Nguyen, Bach, Opgenorth, Terry J
Published in Bioorganic & medicinal chemistry (01.06.1999)
Published in Bioorganic & medicinal chemistry (01.06.1999)
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Wilsbacher, Julie L, Cheng, Min, Cheng, Dong, Trammell, Samuel A J, Shi, Yan, Guo, Jun, Koeniger, Stormy L, Kovar, Peter J, He, Yupeng, Selvaraju, Sujatha, Heyman, H Robin, Sorensen, Bryan K, Clark, Richard F, Hansen, T Matthew, Longenecker, Kenton L, Raich, Diana, Korepanova, Alla V, Cepa, Steven, Towne, Danli L, Abraham, Vivek C, Tang, Hua, Richardson, Paul L, McLoughlin, Shaun M, Badagnani, Ilaria, Curtin, Michael L, Michaelides, Michael R, Maag, David, Buchanan, F Gregory, Chiang, Gary G, Gao, Wenqing, Rosenberg, Saul H, Brenner, Charles, Tse, Chris
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Published in Molecular cancer therapeutics (01.07.2017)
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Potent and selective inhibitors of an aspartyl protease-like endothelin converting enzyme identified in rat lung
Shiosaki, Kazumi, Tasker, Andrew S, Sullivan, Gerard M, Sorensen, Bryan K, von Geldern, Thomas W, Wu-Wong, Jinshyun R, Marselle, Carol A, Opgenorth, Terry J
Published in Journal of medicinal chemistry (19.02.1993)
Published in Journal of medicinal chemistry (19.02.1993)
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Pyrrolidine-3-carboxylic acids as endothelin antagonists. 4. Side chain conformational restriction leads to ET(B) selectivity
von Geldern, T W, Tasker, A S, Sorensen, B K, Winn, M, Szczepankiewicz, B G, Dixon, D B, Chiou, W J, Wang, L, Wessale, J L, Adler, A, Marsh, K C, Nguyen, B, Opgenorth, T J
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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Rohde, Jeffrey J, Pliushchev, Marina A, Sorensen, Bryan K, Wodka, Dariusz, Shuai, Qi, Wang, Jiahong, Fung, Steven, Monzon, Katina M, Chiou, William J, Pan, Liping, Deng, Xiaoqing, Chovan, Linda E, Ramaiya, Atul, Mullally, Mark, Henry, Rodger F, Stolarik, DeAnne F, Imade, Hovis M, Marsh, Kennan C, Beno, David W A, Fey, Thomas A, Droz, Brian A, Brune, Michael E, Camp, Heidi S, Sham, Hing L, Frevert, Ernst Uli, Jacobson, Peer B, Link, J T
Published in Journal of medicinal chemistry (11.01.2007)
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Published in Journal of medicinal chemistry (11.01.2007)
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Second-Generation Peptidomimetic Inhibitors of Protein Farnesyltransferase Demonstrating Improved Cellular Potency and Significant in Vivo Efficacy
O'Connor, Stephen J, Barr, Kenneth J, Wang, Le, Sorensen, Bryan K, Tasker, Andrew S, Sham, Hing, Ng, Shi-Chung, Cohen, Jerome, Devine, Edward, Cherian, Sajeev, Saeed, Badr, Zhang, Haichao, Lee, Jang Yun, Warner, Robert, Tahir, Stephen, Kovar, Peter, Ewing, Patricia, Alder, Jeffrey, Mitten, Michael, Leal, Juan, Marsh, Kennan, Bauch, Joy, Hoffman, Daniel J, Sebti, Said M, Rosenberg, Saul H
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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Pyrrolidine-3-carboxylic acids as endothelin antagonists. 5. Highly selective, potent, and orally active ET(A) antagonists
Jae, H S, Winn, M, von Geldern, T W, Sorensen, B K, Chiou, W J, Nguyen, B, Marsh, K C, Opgenorth, T J
Published in Journal of medicinal chemistry (08.11.2001)
Published in Journal of medicinal chemistry (08.11.2001)
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