Double Strain-Promoted Macrocyclization for the Rapid Selection of Cell-Active Stapled Peptides
Lau, Yu Heng, Wu, Yuteng, Rossmann, Maxim, Tan, Ban Xiong, de Andrade, Peterson, Tan, Yaw Sing, Verma, Chandra, McKenzie, Grahame J., Venkitaraman, Ashok R., Hyvönen, Marko, Spring, David R.
Published in Angewandte Chemie (International ed.) (14.12.2015)
Published in Angewandte Chemie (International ed.) (14.12.2015)
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Journal Article
Development of Cell‐Permeable, Non‐Helical Constrained Peptides to Target a Key Protein–Protein Interaction in Ovarian Cancer
Wiedmann, Mareike M., Tan, Yaw Sing, Wu, Yuteng, Aibara, Shintaro, Xu, Wenshu, Sore, Hannah F., Verma, Chandra S., Itzhaki, Laura, Stewart, Murray, Brenton, James D., Spring, David R.
Published in Angewandte Chemie International Edition (09.01.2017)
Published in Angewandte Chemie International Edition (09.01.2017)
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Journal Article
The Multifaceted Roles of Molecular Dynamics Simulations in Drug Discovery
Fox, Stephen John, Li, Jianguo, Tan, Yaw Sing, Nguyen, Minh N, Pal, Arumay, Ouaray, Zohra, Yadahalli, Shilpa, Kannan, Srinivasaraghavan
Published in Current pharmaceutical design (01.01.2016)
Published in Current pharmaceutical design (01.01.2016)
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Journal Article
HNF4A and HNF1A exhibit tissue specific target gene regulation in pancreatic beta cells and hepatocytes
Ng, Natasha Hui Jin, Ghosh, Soumita, Bok, Chek Mei, Ching, Carmen, Low, Blaise Su Jun, Chen, Juin Ting, Lim, Euodia, Miserendino, María Clara, Tan, Yaw Sing, Hoon, Shawn, Teo, Adrian Kee Keong
Published in Nature communications (22.06.2024)
Published in Nature communications (22.06.2024)
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Journal Article
A strategy for the diversity-oriented synthesis of macrocyclic scaffolds using multidimensional coupling
Beckmann, Henning S. G., Nie, Feilin, Hagerman, Caroline E., Johansson, Henrik, Tan, Yaw Sing, Wilcke, David, Spring, David R.
Published in Nature chemistry (01.10.2013)
Published in Nature chemistry (01.10.2013)
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Journal Article
Targeted covalent inhibitors of MDM2 using electrophile-bearing stapled peptides
Charoenpattarapreeda, Jiraborrirak, Tan, Yaw Sing, Iegre, Jessica, Walsh, Stephen J, Fowler, Elaine, Eapen, Rohan S, Wu, Yuteng, Sore, Hannah F, Verma, Chandra S, Itzhaki, Laura, Spring, David R
Published in Chemical communications (Cambridge, England) (14.07.2019)
Published in Chemical communications (Cambridge, England) (14.07.2019)
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Journal Article
The Application of Ligand-Mapping Molecular Dynamics Simulations to the Rational Design of Peptidic Modulators of Protein–Protein Interactions
Tan, Yaw Sing, Spring, David R, Abell, Chris, Verma, Chandra S
Published in Journal of chemical theory and computation (14.07.2015)
Published in Journal of chemical theory and computation (14.07.2015)
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Journal Article
The Use of Chlorobenzene as a Probe Molecule in Molecular Dynamics Simulations
Tan, Yaw Sing, Spring, David R, Abell, Chris, Verma, Chandra
Published in Journal of chemical information and modeling (28.07.2014)
Published in Journal of chemical information and modeling (28.07.2014)
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Journal Article
Incorporation of Putative Helix-Breaking Amino Acids in the Design of Novel Stapled Peptides: Exploring Biophysical and Cellular Permeability Properties
Partridge, Anthony W, Kaan, Hung Yi Kristal, Juang, Yu-Chi, Sadruddin, Ahmad, Lim, Shuhui, Brown, Christopher J, Ng, Simon, Thean, Dawn, Ferrer, Fernando, Johannes, Charles, Yuen, Tsz Ying, Kannan, Srinivasaraghavan, Aronica, Pietro, Tan, Yaw Sing, Pradhan, Mohan R, Verma, Chandra S, Hochman, Jerome, Chen, Shiying, Wan, Hui, Ha, Sookhee, Sherborne, Brad, Lane, David P, Sawyer, Tomi K
Published in Molecules (Basel, Switzerland) (20.06.2019)
Published in Molecules (Basel, Switzerland) (20.06.2019)
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Journal Article
A diversity-oriented synthesis strategy enabling the combinatorial-type variation of macrocyclic peptidomimetic scaffolds
Isidro-Llobet, Albert, Georgiou, Kathy Hadje, Galloway, Warren R. J. D., Giacomini, Elisa, Hansen, Mette R., Mendez-Abt, Gabriela, Tan, Yaw Sing, Carro, Laura, Sore, Hannah F., Spring, David R.
Published in Organic & biomolecular chemistry (21.04.2015)
Published in Organic & biomolecular chemistry (21.04.2015)
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Journal Article
Anatomy of Mdm2 and Mdm4 in evolution
Tan, Ban Xiong, Liew, Hoe Peng, Chua, Joy S, Ghadessy, Farid J, Tan, Yaw Sing, Lane, David P, Coffill, Cynthia R
Published in Journal of molecular cell biology (01.02.2017)
Published in Journal of molecular cell biology (01.02.2017)
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Journal Article
Using Ligand-Mapping Simulations to Design a Ligand Selectively Targeting a Cryptic Surface Pocket of Polo-Like Kinase 1
Tan, Yaw Sing, Śledź, Paweł, Lang, Steffen, Stubbs, Christopher J., Spring, David R., Abell, Chris, Best, Robert B.
Published in Angewandte Chemie (International ed.) (01.10.2012)
Published in Angewandte Chemie (International ed.) (01.10.2012)
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Journal Article
Success probability of high-affinity DNA aptamer generation by genetic alphabet expansion
Kimoto, Michiko, Tan, Hui Pen, Tan, Yaw Sing, Mislan, Nur Afiqah Binte Mohd, Hirao, Ichiro
Published in Philosophical transactions of the Royal Society of London. Series B. Biological sciences (27.02.2023)
Published in Philosophical transactions of the Royal Society of London. Series B. Biological sciences (27.02.2023)
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Journal Article
Macrocyclized Extended Peptides: Inhibiting the Substrate-Recognition Domain of Tankyrase
Xu, Wenshu, Lau, Yu Heng, Fischer, Gerhard, Tan, Yaw Sing, Chattopadhyay, Anasuya, de la Roche, Marc, Hyvönen, Marko, Verma, Chandra, Spring, David R, Itzhaki, Laura S
Published in Journal of the American Chemical Society (15.02.2017)
Published in Journal of the American Chemical Society (15.02.2017)
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Journal Article
Progressive endoplasmic reticulum stress over time due to human insulin gene mutation contributes to pancreatic beta cell dysfunction
Amirruddin, Nur Shabrina, Tan, Wei Xuan, Tan, Yaw Sing, Gardner, Daphne Su-Lyn, Bee, Yong Mong, Verma, Chandra Shekhar, Hoon, Shawn, Lee, Kok Onn, Teo, Adrian Kee Keong
Published in Diabetologia (01.11.2021)
Published in Diabetologia (01.11.2021)
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Journal Article
Targeting cancer addiction for SALL4 by shifting its transcriptome with a pharmacologic peptide
Liu, Bee Hui, Jobichen, Chacko, Chia, C. S. Brian, Chan, Tim Hon Man, Tang, Jing Ping, Chung, Theodora X. Y., Li, Jia, Poulsen, Anders, Hung, Alvin W., Koh-Stenta, Xiaoying, Tan, Yaw Sing, Verma, Chandra S., Tan, Hong Kee, Wu, Chan-Shuo, Li, Feng, Hill, Jeffrey, Joy, Joma, Yang, Henry, Chai, Li, Sivaraman, J., Tenen, Daniel G.
Published in Proceedings of the National Academy of Sciences - PNAS (24.07.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (24.07.2018)
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Journal Article
Diversity-oriented synthesis as a tool for identifying new modulators of mitosis
Ibbeson, Brett M., Laraia, Luca, Alza, Esther, O' Connor, Cornelius J., Tan, Yaw Sing, Davies, Huw M.L., McKenzie, Grahame, Venkitaraman, Ashok R., Spring, David R.
Published in Nature communications (01.01.2014)
Published in Nature communications (01.01.2014)
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Journal Article
Kinetic and thermodynamic effects of phosphorylation on p53 binding to MDM2
Yadahalli, Shilpa, Neira, José L., Johnson, Christopher M., Tan, Yaw Sing, Rowling, Pamela J. E., Chattopadhyay, Anasuya, Verma, Chandra S., Itzhaki, Laura S.
Published in Scientific reports (24.01.2019)
Published in Scientific reports (24.01.2019)
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Journal Article