Synthesis, biological evaluation, and computational investigation of ethyl 2,4,6-trisubstituted-1,4-dihydropyrimidine-5-carboxylates as potential larvicidal agents against Anopheles arabiensis
Duraisamy, Ramasamy, Al-Shar'i, Nizar A., Chandrashekharappa, Sandeep, Deb, Pran Kishore, Gleiser, Raquel M., Tratrat, Christophe, Chopra, Deepak, Muthukurpalya Bhojegowd, Madhusudana Reddy, Thirumalai, Dhakshanamurthy, Morsy, Mohamed A., Ibrahim, Yasmine F., Mohanlall, Viresh, Venugopala, Katharigatta N.
Published in Journal of biomolecular structure & dynamics (23.05.2024)
Published in Journal of biomolecular structure & dynamics (23.05.2024)
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1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector Anopheles arabiensis and In Silico Molecular Docking Study
Venugopala, Katharigatta N, Shinu, Pottathil, Tratrat, Christophe, Deb, Pran Kishore, Gleiser, Raquel M, Chandrashekharappa, Sandeep, Chopra, Deepak, Attimarad, Mahesh, Nair, Anroop B, Sreeharsha, Nagaraja, Mahomoodally, Fawzi M, Haroun, Michelyne, Kandeel, Mahmoud, Asdaq, Syed Mohammed Basheeruddin, Mohanlall, Viresh, Al-Shar'i, Nizar A, Morsy, Mohamed A
Published in Molecules (Basel, Switzerland) (21.04.2022)
Published in Molecules (Basel, Switzerland) (21.04.2022)
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Journal Article
Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis , In Silico ADMET Prediction and Molecular Target Investigation
Venugopala, Katharigatta N, Ramachandra, Pushpalatha, Tratrat, Christophe, Gleiser, Raquel M, Bhandary, Subhrajyoti, Chopra, Deepak, Morsy, Mohamed A, Aldhubiab, Bandar E, Attimarad, Mahesh, Nair, Anroop B, Sreeharsha, Nagaraja, Venugopala, Rashmi, Deb, Pran Kishore, Chandrashekharappa, Sandeep, Khalil, Hany Ezzat, Alwassil, Osama I, Abed, Sara Nidal, Bataineh, Yazan A, Palenge, Ramachandra, Haroun, Michelyne, Pottathil, Shinu, Girish, Meravanige B, Akrawi, Sabah H, Mohanlall, Viresh
Published in Molecules (Basel, Switzerland) (13.03.2020)
Published in Molecules (Basel, Switzerland) (13.03.2020)
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Culicidae community composition and temporal dynamics in Guapiaçu Ecological Reserve, Cachoeiras de Macacu, Rio de Janeiro, Brazil
Alencar, Jeronimo, de Mello, Cecilia Ferreira, Guimarães, Anthony Érico, Gil-Santana, Hélcio R, Silva, Júlia Dos Santos, Santos-Mallet, Jacenir R, Gleiser, Raquel M
Published in PloS one (27.03.2015)
Published in PloS one (27.03.2015)
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Journal Article
Biodiversity and Temporal Distribution of Immature Culicidae in the Atlantic Forest, Rio de Janeiro State, Brazil
Alencar, Jeronimo, de Mello, Cecília Ferreira, Serra-Freire, Nicolau Maués, Guimarães, Anthony Érico, Gil-Santana, Hélcio R, Gleiser, Raquel M
Published in PloS one (12.07.2016)
Published in PloS one (12.07.2016)
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Journal Article
Greener synthesis of indolizine analogues using water as a base and solvent: study for larvicidal activity against Anopheles arabiensis
Sandeep, Chandrashekharappa, Venugopala, Katharigatta N., Gleiser, Raquel M., Chetram, Abeen, Padmashali, Basavaraj, Kulkarni, Rashmi S., Venugopala, Rashmi, Odhav, Bharti
Published in Chemical biology & drug design (01.12.2016)
Published in Chemical biology & drug design (01.12.2016)
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Aedes aegypti oviposition dynamics in towns with low human population density in yungas and dry chaco, Salta, Argentina
Chanampa, Mariana M., Aparicio, Juan Pablo, Hodi, Soledad, Derlindati, Enrique, Rodriguez, Nicolas, Larsen, Roxana Alejandra García, Gleiser, Raquel M.
Published in Acta tropica (01.06.2024)
Published in Acta tropica (01.06.2024)
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Journal Article
Effects of the essential oils of Lippia turbinata and Lippia polystachya (Verbenaceae) on the temporal pattern of locomotion of the mosquito Culex quinquefasciatus (Diptera: Culicidae) larvae
Kembro, Jackelyn M, Marin, Raúl H, Zygadlo, Julio A, Gleiser, Raquel M
Published in Parasitology research (1987) (01.04.2009)
Published in Parasitology research (1987) (01.04.2009)
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Synthesis and antimosquito properties of 2,6-substituted benzo[d]thiazole and 2,4-substituted benzo[d]thiazole analogues against Anopheles arabiensis
Venugopala, Katharigatta Narayanaswamy, Krishnappa, Manjula, Nayak, Susanta K., Subrahmanya, Bhat K., Vaderapura, Jayashankaragowda P., Chalannavar, Raju K., Gleiser, Raquel M., Odhav, Bharti
Published in European journal of medicinal chemistry (01.07.2013)
Published in European journal of medicinal chemistry (01.07.2013)
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Journal Article
Larvicidal study of tetrahydropyrimidine scaffolds against Anopheles arabiensis and structural insight by single crystal X‐ray studies
Bairagi, Keshab M., Venugopala, Katharigatta N., Mondal, Pradip Kumar, Gleiser, Raquel M., Chopra, Deepak, García, Daniel, Odhav, Bharti, Nayak, Susanta K.
Published in Chemical biology & drug design (01.12.2018)
Published in Chemical biology & drug design (01.12.2018)
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Journal Article
Synthesis, Polymorphism, and Insecticidal Activity of Methyl 4-(4-chlorophenyl)-8-iodo-2-methyl-6-oxo-1,6-dihydro-4H-pyrimido[2,1-b]quinazoline-3-Carboxylate Against Anopheles arabiensis Mosquito
Venugopala, Katharigatta N., Nayak, Susanta K., Gleiser, Raquel M., Sanchez-Borzone, Mariela E., Garcia, Daniel A., Odhav, Bharti
Published in Chemical biology & drug design (01.07.2016)
Published in Chemical biology & drug design (01.07.2016)
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Journal Article
Synthesis and characterization of a novel series of 1,4‐dihydropyridine analogues for larvicidal activity against Anopheles arabiensis
Dharma Rao, Bhaskara D., Bhandary, Subhrajyoti, Chopra, Deepak, Venugopala, Katharigatta N., Gleiser, Raquel M., Kasumbwe, Kabange, Odhav, Bharti
Published in Chemical biology & drug design (01.09.2017)
Published in Chemical biology & drug design (01.09.2017)
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Journal Article
Membrane effects of dihydropyrimidine analogues with larvicidal activity
Sánchez-Borzone, Mariela E., Mariani, Maria E., Miguel, Virginia, Gleiser, Raquel M., Odhav, Bharti, Venugopala, Katharigatta N., García, Daniel A.
Published in Colloids and surfaces, B, Biointerfaces (01.02.2017)
Published in Colloids and surfaces, B, Biointerfaces (01.02.2017)
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Journal Article
Snail shells as larval habitat of Limatus durhamii (Diptera: Culicidae) in the Yungas of Argentina
Mangudo, Carolina, Campos, Raúl E., Rossi, Gustavo C., Gleiser, Raquel M.
Published in Acta tropica (01.03.2017)
Published in Acta tropica (01.03.2017)
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Journal Article
Vertical Oviposition Activity of Mosquitoes in the Atlantic Forest of Brazil with Emphasis on the Sylvan Vector, Haemagogus leucocelaenus (Diptera: Culicidae)
Alencar, Jeronimo, Mello, Cecilia Ferreira de, Gil-Santana, Hélcio R, Guimarães, Anthony Érico, Almeida, Sergio Antonio Silva de, Gleiser, Raquel M
Published in Journal of vector ecology (01.06.2016)
Published in Journal of vector ecology (01.06.2016)
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Journal Article
Tree Holes as Larval Habitats for Aedes aegypti in Public Areas in Aguaray, Salta Province, Argentina
Mangudo, Carolina, Aparicio, Juan P, Gleiser, Raquel M
Published in Journal of vector ecology (01.06.2011)
Published in Journal of vector ecology (01.06.2011)
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