The Most Common Functional Groups in Bioactive Molecules and How Their Popularity Has Evolved over Time
Ertl, Peter, Altmann, Eva, McKenna, Jeffrey M
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Discovery of a Covalent FEM1B Recruiter for Targeted Protein Degradation Applications
Henning, Nathaniel J, Manford, Andrew G, Spradlin, Jessica N, Brittain, Scott M, Zhang, Erika, McKenna, Jeffrey M, Tallarico, John A, Schirle, Markus, Rape, Michael, Nomura, Daniel K
Published in Journal of the American Chemical Society (19.01.2022)
Published in Journal of the American Chemical Society (19.01.2022)
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Harnessing the anti-cancer natural product nimbolide for targeted protein degradation
Spradlin, Jessica N., Hu, Xirui, Ward, Carl C., Brittain, Scott M., Jones, Michael D., Ou, Lisha, To, Milton, Proudfoot, Andrew, Ornelas, Elizabeth, Woldegiorgis, Mikias, Olzmann, James A., Bussiere, Dirksen E., Thomas, Jason R., Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Nature chemical biology (01.07.2019)
Published in Nature chemical biology (01.07.2019)
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Covalent Ligand Screening Uncovers a RNF4 E3 Ligase Recruiter for Targeted Protein Degradation Applications
Ward, Carl C, Kleinman, Jordan I, Brittain, Scott M, Lee, Patrick S, Chung, Clive Yik Sham, Kim, Kenneth, Petri, Yana, Thomas, Jason R, Tallarico, John A, McKenna, Jeffrey M, Schirle, Markus, Nomura, Daniel K
Published in ACS chemical biology (15.11.2019)
Published in ACS chemical biology (15.11.2019)
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Bardoxolone conjugation enables targeted protein degradation of BRD4
Tong, Bingqi, Luo, Mai, Xie, Yi, Spradlin, Jessica N., Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Scientific reports (23.09.2020)
Published in Scientific reports (23.09.2020)
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Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC
Boike, Lydia, Cioffi, Alexander G., Majewski, Felix C., Co, Jennifer, Henning, Nathaniel J., Jones, Michael D., Liu, Gang, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in Cell chemical biology (21.01.2021)
Published in Cell chemical biology (21.01.2021)
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Chiral Diaryliodonium Phosphate Enables Light Driven Diastereoselective α‑C(sp3)–H Acetalization
Ye, Baihua, Zhao, Jie, Zhao, Ke, McKenna, Jeffrey M, Toste, F. Dean
Published in Journal of the American Chemical Society (05.07.2018)
Published in Journal of the American Chemical Society (05.07.2018)
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Chemoproteomics-enabled discovery of covalent RNF114-based degraders that mimic natural product function
Luo, Mai, Spradlin, Jessica N., Boike, Lydia, Tong, Bingqi, Brittain, Scott M., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Cell chemical biology (15.04.2021)
Published in Cell chemical biology (15.04.2021)
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Manumycin polyketides act as molecular glues between UBR7 and P53
Isobe, Yosuke, Okumura, Mikiko, McGregor, Lynn M., Brittain, Scott M., Jones, Michael D., Liang, Xiaoyou, White, Ross, Forrester, William, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in Nature chemical biology (01.11.2020)
Published in Nature chemical biology (01.11.2020)
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Deubiquitinase-targeting chimeras for targeted protein stabilization
Henning, Nathaniel J., Boike, Lydia, Spradlin, Jessica N., Ward, Carl C., Liu, Gang, Zhang, Erika, Belcher, Bridget P., Brittain, Scott M., Hesse, Matthew J., Dovala, Dustin, McGregor, Lynn M., Valdez Misiolek, Rachel, Plasschaert, Lindsey W., Rowlands, David J., Wang, Feng, Frank, Andreas O., Fuller, Daniel, Estes, Abigail R., Randal, Katelyn L., Panidapu, Anoohya, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in Nature chemical biology (01.04.2022)
Published in Nature chemical biology (01.04.2022)
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Targeted Protein Degradation through E2 Recruitment
Forte, Nafsika, Dovala, Dustin, Hesse, Matthew J., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
Published in ACS chemical biology (21.04.2023)
Published in ACS chemical biology (21.04.2023)
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Oxidative cyclization reagents reveal tryptophan cation–π interactions
Xie, Xiao, Moon, Patrick J., Crossley, Steven W. M., Bischoff, Amanda J., He, Dan, Li, Gen, Dao, Nam, Gonzalez-Valero, Angel, Reeves, Audrey G., McKenna, Jeffrey M., Elledge, Susanna K., Wells, James A., Toste, F. Dean, Chang, Christopher J.
Published in Nature (London) (21.03.2024)
Published in Nature (London) (21.03.2024)
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An Activity-Based Oxaziridine Platform for Identifying and Developing Covalent Ligands for Functional Allosteric Methionine Sites: Redox-Dependent Inhibition of Cyclin-Dependent Kinase 4
Gonzalez-Valero, Angel, Reeves, Audrey G., Page, Annika C. S., Moon, Patrick J., Miller, Edward, Coulonval, Katia, Crossley, Steven W. M., Xie, Xiao, He, Dan, Musacchio, Patricia Z., Christian, Alec H., McKenna, Jeffrey M., Lewis, Richard A., Fang, Eric, Dovala, Dustin, Lu, Yipin, McGregor, Lynn M., Schirle, Markus, Tallarico, John A., Roger, Pierre P., Toste, F. Dean, Chang, Christopher J.
Published in Journal of the American Chemical Society (21.12.2022)
Published in Journal of the American Chemical Society (21.12.2022)
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Ophiobolin A Covalently Targets Mitochondrial Complex IV Leading to Metabolic Collapse in Cancer Cells
Gowans, Flor A., Thach, Danny Q., Zhu, Zhouyang, Wang, Yangzhi, Altamirano Poblano, Belen E., Dovala, Dustin, Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Published in ACS chemical biology (21.06.2024)
Published in ACS chemical biology (21.06.2024)
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Discovery of Potent Pyrazoline‐Based Covalent SARS‐CoV‐2 Main Protease Inhibitors
Moon, Patrick, Zammit, Charlotte M., Shao, Qian, Dovala, Dustin, Boike, Lydia, Henning, Nathaniel J., Knapp, Mark, Spradlin, Jessica N., Ward, Carl C., Wolleb, Helene, Fuller, Daniel, Blake, Gabrielle, Murphy, Jason P., Wang, Feng, Lu, Yipin, Moquin, Stephanie A., Tandeske, Laura, Hesse, Matthew J., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Toste, F. Dean, Nomura, Daniel K.
Published in Chembiochem : a European journal of chemical biology (01.06.2023)
Published in Chembiochem : a European journal of chemical biology (01.06.2023)
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Lentigo Maligna/Lentigo Maligna Melanoma: Current State of Diagnosis and Treatment
McKENNA, JEFFREY K., FLORELL, SCOTT R., GOLDMAN, GLENN D., BOWEN, GLEN M.
Published in Dermatologic surgery (01.04.2006)
Published in Dermatologic surgery (01.04.2006)
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α- and α′-Lithiation–Electrophile Trapping of N‑Thiopivaloyl and N-tert-Butoxythiocarbonyl α‑Substituted Azetidines: Rationalization of the Regiodivergence Using NMR and Computation
Jackson, Kelvin E, Mortimer, Claire L, Odell, Barbara, McKenna, Jeffrey M, Claridge, Timothy D. W, Paton, Robert S, Hodgson, David M
Published in Journal of organic chemistry (16.10.2015)
Published in Journal of organic chemistry (16.10.2015)
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