Design and Synthesis of Janus Kinase 2 (JAK2) and Histone Deacetlyase (HDAC) Bispecific Inhibitors Based on Pacritinib and Evidence of Dual Pathway Inhibition in Hematological Cell Lines
Yang, Eugene Guorong, Mustafa, Nurulhuda, Tan, Eng Chong, Poulsen, Anders, Ramanujulu, Pondy Murugappan, Chng, Wee Joo, Yen, Jeffrey J. Y, Dymock, Brian W
Published in Journal of medicinal chemistry (22.09.2016)
Published in Journal of medicinal chemistry (22.09.2016)
Get full text
Journal Article
Hydrogen sulfide promotes adipogenesis in 3T3L1 cells
Tsai, Chin-Yi, Peh, Meng Teng, Feng, Wei, Dymock, Brian William, Moore, Philip Keith
Published in PloS one (30.03.2015)
Published in PloS one (30.03.2015)
Get full text
Journal Article
Design and Synthesis of Ligand Efficient Dual Inhibitors of Janus Kinase (JAK) and Histone Deacetylase (HDAC) Based on Ruxolitinib and Vorinostat
Yao, Lianbin, Mustafa, Nurulhuda, Tan, Eng Chong, Poulsen, Anders, Singh, Prachi, Duong-Thi, Minh-Dao, Lee, Jeannie X. T, Ramanujulu, Pondy Murugappan, Chng, Wee Joo, Yen, Jeffrey J. Y, Ohlson, Sten, Dymock, Brian W
Published in Journal of medicinal chemistry (26.10.2017)
Published in Journal of medicinal chemistry (26.10.2017)
Get full text
Journal Article
Dual blockade of the lipid kinase PIP4Ks and mitotic pathways leads to cancer-selective lethality
Kitagawa, Mayumi, Liao, Pei-Ju, Lee, Kyung Hee, Wong, Jasmine, Shang, See Cheng, Minami, Noriaki, Sampetrean, Oltea, Saya, Hideyuki, Lingyun, Dai, Prabhu, Nayana, Diam, Go Ka, Sobota, Radoslaw, Larsson, Andreas, Nordlund, Pär, McCormick, Frank, Ghosh, Sujoy, Epstein, David M., Dymock, Brian W., Lee, Sang Hyun
Published in Nature communications (19.12.2017)
Published in Nature communications (19.12.2017)
Get full text
Journal Article
Discovery of New H2S Releasing Phosphordithioates and 2,3-Dihydro-2-phenyl-2-sulfanylenebenzo[d][1,3,2]oxazaphospholes with Improved Antiproliferative Activity
Feng, Wei, Teo, Xin-Yi, Novera, Wisna, Ramanujulu, Pondy Murugappan, Liang, Dong, Huang, Dejian, Moore, Philip K, Deng, Lih-Wen, Dymock, Brian W
Published in Journal of medicinal chemistry (27.08.2015)
Published in Journal of medicinal chemistry (27.08.2015)
Get full text
Journal Article
Predicting Tacrolimus Concentrations in the Skin of Adult Kidney Transplant Recipients: A Feasibility Study
Sartain, Felicity, Viecelli, Andrea K, Veitch, Margaret, Franklin, Michael E, Dymock, Brian W, Wells, James W, Campbell, Scott B
Published in Transplant international (2024)
Published in Transplant international (2024)
Get full text
Journal Article
Discovery of a potent histone deacetylase (HDAC) 3/6 selective dual inhibitor
Soumyanarayanan, Uttara, Ramanujulu, Pondy Murugappan, Mustafa, Nurulhuda, Haider, Shozeb, Fang Nee, Adina Huey, Tong, Jie Xin, Tan, Kevin S.W., Chng, Wee Joo, Dymock, Brian W.
Published in European journal of medicinal chemistry (15.12.2019)
Published in European journal of medicinal chemistry (15.12.2019)
Get full text
Journal Article
Towards Selective Mycobacterial ClpP1P2 Inhibitors with Reduced Activity against the Human Proteasome
Moreira, Wilfried, Santhanakrishnan, Sridhar, Ngan, Grace J Y, Low, Choon Bing, Sangthongpitag, Kanda, Poulsen, Anders, Dymock, Brian W, Dick, Thomas
Published in Antimicrobial agents and chemotherapy (01.05.2017)
Published in Antimicrobial agents and chemotherapy (01.05.2017)
Get full text
Journal Article
Discovery of the Macrocycle 11-(2-Pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaene (SB1518), a Potent Janus Kinase 2/Fms-Like Tyrosine Kinase-3 (JAK2/FLT3) Inhibitor for the Treatment of Myelofibrosis and Lymphoma
William, Anthony D, Lee, Angeline C.-H, Blanchard, Stéphanie, Poulsen, Anders, Teo, Ee Ling, Nagaraj, Harish, Tan, Evelyn, Chen, Dizhong, Williams, Meredith, Sun, Eric T, Goh, Kee Chuan, Ong, Wai Chung, Goh, Siok Kun, Hart, Stefan, Jayaraman, Ramesh, Pasha, Mohammed Khalid, Ethirajulu, Kantharaj, Wood, Jeanette M, Dymock, Brian W
Published in Journal of medicinal chemistry (14.07.2011)
Published in Journal of medicinal chemistry (14.07.2011)
Get full text
Journal Article
Hydrogen sulfide is an endogenous regulator of aging in Caenorhabditis elegans
Qabazard, Bedoor, Li, Ling, Gruber, Jan, Peh, Meng Teng, Ng, Li Fang, Kumar, Srinivasan Dinesh, Rose, Peter, Tan, Choon-Hong, Dymock, Brian W, Wei, Feng, Swain, Suresh C, Halliwell, Barry, Stürzenbaum, Stephen R, Moore, Philip K
Published in Antioxidants & redox signaling (01.06.2014)
Published in Antioxidants & redox signaling (01.06.2014)
Get more information
Journal Article
NVP-AUY922: a novel heat shock protein 90 inhibitor active against xenograft tumor growth, angiogenesis, and metastasis
Eccles, Suzanne A, Massey, Andy, Raynaud, Florence I, Sharp, Swee Y, Box, Gary, Valenti, Melanie, Patterson, Lisa, de Haven Brandon, Alexis, Gowan, Sharon, Boxall, Frances, Aherne, Wynne, Rowlands, Martin, Hayes, Angela, Martins, Vanessa, Urban, Frederique, Boxall, Kathy, Prodromou, Chrisostomos, Pearl, Laurence, James, Karen, Matthews, Thomas P, Cheung, Kwai-Ming, Kalusa, Andrew, Jones, Keith, McDonald, Edward, Barril, Xavier, Brough, Paul A, Cansfield, Julie E, Dymock, Brian, Drysdale, Martin J, Finch, Harry, Howes, Rob, Hubbard, Roderick E, Surgenor, Alan, Webb, Paul, Wood, Mike, Wright, Lisa, Workman, Paul
Published in Cancer research (Chicago, Ill.) (15.04.2008)
Published in Cancer research (Chicago, Ill.) (15.04.2008)
Get full text
Journal Article
o-Vanillin binds covalently to MAL/TIRAP Lys-210 but independently inhibits TLR2
Rahaman, Md Habibur, Thygesen, Sara J, Maxwell, Michael J, Kim, Hyoyoung, Mudai, Prerna, Nanson, Jeffrey D, Jia, Xinying, Vajjhala, Parimala R, Hedger, Andrew, Vetter, Irina, Haselhorst, Thomas, Robertson, Avril A B, Dymock, Brian, Ve, Thomas, Mobli, Mehdi, Stacey, Katryn J, Kobe, Bostjan
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
Get full text
Journal Article