Advances in therapeutic peptides targeting G protein-coupled receptors
Davenport, Anthony P., Scully, Conor C. G., de Graaf, Chris, Brown, Alastair J. H., Maguire, Janet J.
Published in Nature reviews. Drug discovery (01.06.2020)
Published in Nature reviews. Drug discovery (01.06.2020)
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Journal Article
Synthesis of Aminoboronic Acid Derivatives from Amines and Amphoteric Boryl Carbonyl Compounds
Diaz, Diego B., Scully, Conor C. G., Liew, Sean K., Adachi, Shinya, Trinchera, Piera, St. Denis, Jeffrey D., Yudin, Andrei K.
Published in Angewandte Chemie (International ed.) (04.10.2016)
Published in Angewandte Chemie (International ed.) (04.10.2016)
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Journal Article
Exocyclic Control of Turn Induction in Macrocyclic Peptide Scaffolds
Zaretsky, Serge, Scully, Conor C. G., Lough, Alan J., Yudin, Andrei K.
Published in Chemistry : a European journal (23.12.2013)
Published in Chemistry : a European journal (23.12.2013)
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Journal Article
Passive Membrane Permeability of Macrocycles Can Be Controlled by Exocyclic Amide Bonds
Hickey, Jennifer L, Zaretsky, Serge, St. Denis, Megan A, Kumar Chakka, Sai, Morshed, M. Monzur, Scully, Conor C. G, Roughton, Andrew L, Yudin, Andrei K
Published in Journal of medicinal chemistry (09.06.2016)
Published in Journal of medicinal chemistry (09.06.2016)
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Journal Article
Site-Specific Integration of Amino Acid Fragments into Cyclic Peptides
White, Christopher J, Hickey, Jennifer L, Scully, Conor C. G, Yudin, Andrei K
Published in Journal of the American Chemical Society (12.03.2014)
Published in Journal of the American Chemical Society (12.03.2014)
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Journal Article
Conformational Modulation of in Vitro Activity of Cyclic RGD Peptides via Aziridine Aldehyde-Driven Macrocyclization Chemistry
Roxin, Áron, Chen, Juan, Scully, Conor C. G, Rotstein, Benjamin H, Yudin, Andrei K, Zheng, Gang
Published in Bioconjugate chemistry (18.07.2012)
Published in Bioconjugate chemistry (18.07.2012)
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Journal Article
Rational Design of Calpain Inhibitors Based on Calpastatin Peptidomimetics
Low, Kristin E, Ler, Spencer, Chen, Kevin J, Campbell, Robert L, Hickey, Jennifer L, Tan, Joanne, Scully, Conor C. G, Davies, Peter L, Yudin, Andrei K, Zaretsky, Serge
Published in Journal of medicinal chemistry (09.06.2016)
Published in Journal of medicinal chemistry (09.06.2016)
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Journal Article
Facile synthesis of borofragments and their evaluation in activity-based protein profiling
Adachi, Shinya, Cognetta, Armand B., Niphakis, Micah J., He, Zhi, Zajdlik, Adam, Denis, Jeffrey D. St, Scully, Conor C. G., Cravatt, Benjamin F., Yudin, Andrei K.
Published in Chemical communications (Cambridge, England) (28.02.2015)
Published in Chemical communications (Cambridge, England) (28.02.2015)
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Journal Article
Bending Rigid Molecular Rods: Formation of Oligoproline Macrocycles
Scully, Conor C. G., Rai, Vishal, Poda, Gennadiy, Zaretsky, Serge, Burns, Darcy C., Houliston, R. Scott, Lou, Tiantong, Yudin, Andrei K.
Published in Chemistry : a European journal (03.12.2012)
Published in Chemistry : a European journal (03.12.2012)
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Journal Article
Metal Clips That Induce Unstructured Pentapeptides To Be α-Helical In Water
Ma, Michelle T, Hoang, Huy N, Scully, Conor C. G, Appleton, Trevor G, Fairlie, David P
Published in Journal of the American Chemical Society (01.04.2009)
Published in Journal of the American Chemical Society (01.04.2009)
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Journal Article
Stereocontrolled Disruption of the Ugi Reaction toward the Production of Chiral Piperazinones: Substrate Scope and Process Development
Zaretsky, Serge, Adachi, Shinya, Rotstein, Benjamin H, Hickey, Jennifer L, Scully, Conor C. G, St. Denis, Jeffrey D, Courtemanche, Rebecca, Yu, Joy C. Y, Chung, Benjamin K. W, Yudin, Andrei K
Published in Journal of organic chemistry (07.11.2014)
Published in Journal of organic chemistry (07.11.2014)
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Journal Article
Potent complement C3a receptor agonists derived from oxazole amino acids: Structure–activity relationships
Singh, Ranee, Reed, Anthony N., Chu, Peifei, Scully, Conor C.G., Yau, Mei-Kwan, Suen, Jacky Y., Durek, Thomas, Reid, Robert C., Fairlie, David P.
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
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Journal Article