A fluorine scan of a tubulin polymerization inhibitor isocombretastatin A-4: Design, synthesis, molecular modelling, and biological evaluation
Naret, Timothée, Bignon, Jérôme, Bernadat, Guillaume, Benchekroun, Mohamed, Levaique, Helene, Lenoir, Christine, Dubois, Joelle, Pruvost, Alain, Saller, François, Borgel, Delphine, Manoury, Boris, Leblais, Veronique, Darrigrand, Romain, Apcher, Sébastien, Brion, Jean-Daniel, Schmitt, Etienne, Leroux, Frédéric R., Alami, Mouad, Hamze, Abdallah
Published in European journal of medicinal chemistry (01.01.2018)
Published in European journal of medicinal chemistry (01.01.2018)
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Synthesis and structural properties of hexaaza[5]helicene containing two [1,2,3]triazolo[1,5-a]pyridine moieties
Adam, Rosa, Ballesteros-Garrido, Rafael, Vallcorba, Oriol, Abarca, Belén, Ballesteros, Rafael, Leroux, Frédéric R., Colobert, Françoise, Amigó, José M., Rius, Jordi
Published in Tetrahedron letters (07.08.2013)
Published in Tetrahedron letters (07.08.2013)
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Ketenimines as Intermediates To Access Difluoromethoxylated Scaffolds
Loison, Anaïs, Hanquet, Gilles, Toulgoat, Fabien, Billard, Thierry, Panossian, Armen, Leroux, Frédéric R.
Published in Organic letters (18.11.2022)
Published in Organic letters (18.11.2022)
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Deprotonative Functionalization of the Difluoromethyl Group
Santos, Laura, Panossian, Armen, Donnard, Morgan, Vors, Jean-Pierre, Pazenok, Sergii, Bernier, David, Leroux, Frédéric R
Published in Organic letters (06.11.2020)
Published in Organic letters (06.11.2020)
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Palladium‐Catalyzed Silylcyanation of Ynamides: Regio‐ and Stereoselective Access to Tetrasubstituted 3‐Silyl‐2‐Aminoacrylonitriles
Hansjacob, Pierre, Leroux, Frédéric R., Gandon, Vincent, Donnard, Morgan
Published in Angewandte Chemie International Edition (28.03.2022)
Published in Angewandte Chemie International Edition (28.03.2022)
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A Major Advance in the Synthesis of Fluoroalkyl Pyrazoles: Tuneable Regioselectivity and Broad Substitution Patterns
Schmitt, Etienne, Panossian, Armen, Vors, Jean-Pierre, Funke, Christian, Lui, Norbert, Pazenok, Sergiy, Leroux, Frédéric R.
Published in Chemistry : a European journal (01.08.2016)
Published in Chemistry : a European journal (01.08.2016)
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Synthesis and Use of Trifluoromethylthiolated Ketenimines
Guérin, Thomas, Pikun, Nadiia V., Morioka, Ryutaro, Panossian, Armen, Hanquet, Gilles, Leroux, Frédéric R.
Published in Chemistry : a European journal (20.11.2020)
Published in Chemistry : a European journal (20.11.2020)
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Atropodiastereoselective CH Olefination of Biphenyl p-Tolyl Sulfoxides with Acrylates
Wesch, Thomas, Leroux, Frédéric R., Colobert, Françoise
Published in Advanced synthesis & catalysis (12.08.2013)
Published in Advanced synthesis & catalysis (12.08.2013)
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Unlocking the Power of Acyl Fluorides: A Comprehensive Guide to Synthesis and Properties
Bonnefoy, Clemence, Gallego, Adrien, Delobel, Clement, Raynal, Betty, Decourt, Maxime, Chefdeville, Emmanuel, Hanquet, Gilles, Panossian, Armen, Leroux, Frederic R., Toulgoat, Fabien, Billard, Thierry
Published in European journal of organic chemistry (13.05.2024)
Published in European journal of organic chemistry (13.05.2024)
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Traceless N‐Polyfluoroalkylation of Weakly Nucleophilic Nitrogen Containing Compounds
Santos, Laura, Audet, Florian, Donnard, Morgan, Panossian, Armen, Vors, Jean‐Pierre, Bernier, David, Pazenok, Sergii, Leroux, Frédéric R.
Published in Chemistry : a European journal (07.06.2023)
Published in Chemistry : a European journal (07.06.2023)
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The Winding Road towards an Atropo‐enantioselective ‘ARYNE Coupling’
Augros, David, Comoy, Corinne, Fort, Yves, Leroux, Frédéric R., Panossian, Armen
Published in European journal of organic chemistry (08.04.2021)
Published in European journal of organic chemistry (08.04.2021)
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