Development of Endocyclic Control Elements for Peptide Macrocycles
Appavoo, Solomon D, Kaji, Takuya, Frost, John R, Scully, Conor C. G, Yudin, Andrei K
Published in Journal of the American Chemical Society (18.07.2018)
Published in Journal of the American Chemical Society (18.07.2018)
Get full text
Journal Article
Synthesis of Aminoboronic Acid Derivatives from Amines and Amphoteric Boryl Carbonyl Compounds
Diaz, Diego B., Scully, Conor C. G., Liew, Sean K., Adachi, Shinya, Trinchera, Piera, St. Denis, Jeffrey D., Yudin, Andrei K.
Published in Angewandte Chemie (International ed.) (04.10.2016)
Published in Angewandte Chemie (International ed.) (04.10.2016)
Get full text
Journal Article
Exocyclic Control of Turn Induction in Macrocyclic Peptide Scaffolds
Zaretsky, Serge, Scully, Conor C. G., Lough, Alan J., Yudin, Andrei K.
Published in Chemistry : a European journal (23.12.2013)
Published in Chemistry : a European journal (23.12.2013)
Get full text
Journal Article
Passive Membrane Permeability of Macrocycles Can Be Controlled by Exocyclic Amide Bonds
Hickey, Jennifer L, Zaretsky, Serge, St. Denis, Megan A, Kumar Chakka, Sai, Morshed, M. Monzur, Scully, Conor C. G, Roughton, Andrew L, Yudin, Andrei K
Published in Journal of medicinal chemistry (09.06.2016)
Published in Journal of medicinal chemistry (09.06.2016)
Get full text
Journal Article
Site-Specific Integration of Amino Acid Fragments into Cyclic Peptides
White, Christopher J, Hickey, Jennifer L, Scully, Conor C. G, Yudin, Andrei K
Published in Journal of the American Chemical Society (12.03.2014)
Published in Journal of the American Chemical Society (12.03.2014)
Get full text
Journal Article
Solid-Phase Parallel Synthesis of Functionalised Medium-to-Large Cyclic Peptidomimetics through Three-Component Coupling Driven by Aziridine Aldehyde Dimers
Treder, Adam P., Hickey, Jennifer L., Tremblay, Marie-Claude J., Zaretsky, Serge, Scully, Conor C. G., Mancuso, John, Doucet, Annie, Yudin, Andrei K., Marsault, Eric
Published in Chemistry : a European journal (15.06.2015)
Published in Chemistry : a European journal (15.06.2015)
Get full text
Journal Article
The effect of backbone flexibility on site-selective modification of macrocycles
Scully, Conor C. G., White, Christopher J., Yudin, Andrei K.
Published in Organic & biomolecular chemistry (02.11.2016)
Published in Organic & biomolecular chemistry (02.11.2016)
Get full text
Journal Article
Conformational Modulation of in Vitro Activity of Cyclic RGD Peptides via Aziridine Aldehyde-Driven Macrocyclization Chemistry
Roxin, Áron, Chen, Juan, Scully, Conor C. G, Rotstein, Benjamin H, Yudin, Andrei K, Zheng, Gang
Published in Bioconjugate chemistry (18.07.2012)
Published in Bioconjugate chemistry (18.07.2012)
Get full text
Journal Article
Rational Design of Calpain Inhibitors Based on Calpastatin Peptidomimetics
Low, Kristin E, Ler, Spencer, Chen, Kevin J, Campbell, Robert L, Hickey, Jennifer L, Tan, Joanne, Scully, Conor C. G, Davies, Peter L, Yudin, Andrei K, Zaretsky, Serge
Published in Journal of medicinal chemistry (09.06.2016)
Published in Journal of medicinal chemistry (09.06.2016)
Get full text
Journal Article
Facile synthesis of borofragments and their evaluation in activity-based protein profiling
Adachi, Shinya, Cognetta, Armand B., Niphakis, Micah J., He, Zhi, Zajdlik, Adam, Denis, Jeffrey D. St, Scully, Conor C. G., Cravatt, Benjamin F., Yudin, Andrei K.
Published in Chemical communications (Cambridge, England) (28.02.2015)
Published in Chemical communications (Cambridge, England) (28.02.2015)
Get full text
Journal Article
Bending Rigid Molecular Rods: Formation of Oligoproline Macrocycles
Scully, Conor C. G., Rai, Vishal, Poda, Gennadiy, Zaretsky, Serge, Burns, Darcy C., Houliston, R. Scott, Lou, Tiantong, Yudin, Andrei K.
Published in Chemistry : a European journal (03.12.2012)
Published in Chemistry : a European journal (03.12.2012)
Get full text
Journal Article
Cyclic Penta- and Hexaleucine Peptides without N‑Methylation Are Orally Absorbed
Hill, Timothy A, Lohman, Rink-Jan, Hoang, Huy N, Nielsen, Daniel S, Scully, Conor C. G, Kok, W. Mei, Liu, Ligong, Lucke, Andrew J, Stoermer, Martin J, Schroeder, Christina I, Chaousis, Stephanie, Colless, Barbara, Bernhardt, Paul V, Edmonds, David J, Griffith, David A, Rotter, Charles J, Ruggeri, Roger B, Price, David A, Liras, Spiros, Craik, David J, Fairlie, David P
Published in ACS medicinal chemistry letters (09.10.2014)
Published in ACS medicinal chemistry letters (09.10.2014)
Get full text
Journal Article
Stereocontrolled Disruption of the Ugi Reaction toward the Production of Chiral Piperazinones: Substrate Scope and Process Development
Zaretsky, Serge, Adachi, Shinya, Rotstein, Benjamin H, Hickey, Jennifer L, Scully, Conor C. G, St. Denis, Jeffrey D, Courtemanche, Rebecca, Yu, Joy C. Y, Chung, Benjamin K. W, Yudin, Andrei K
Published in Journal of organic chemistry (07.11.2014)
Published in Journal of organic chemistry (07.11.2014)
Get full text
Journal Article
Predicting cyclic peptide chemical shifts using quantum mechanical calculations
Zaretsky, Serge, Hickey, Jennifer L., St. Denis, Megan A., Scully, Conor C.G., Roughton, Andrew L., Tantillo, Dean J., Lodewyk, Michael W., Yudin, Andrei K.
Published in Tetrahedron (21.10.2014)
Published in Tetrahedron (21.10.2014)
Get full text
Journal Article
Potent complement C3a receptor agonists derived from oxazole amino acids: Structure–activity relationships
Singh, Ranee, Reed, Anthony N., Chu, Peifei, Scully, Conor C.G., Yau, Mei-Kwan, Suen, Jacky Y., Durek, Thomas, Reid, Robert C., Fairlie, David P.
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
Get full text
Journal Article