The discovery of rofecoxib, [MK 966, VIOXX ®, 4-(4′-methylsulfonylphenyl)-3-phenyl-2(5 H)-furanone], an orally active cyclooxygenase-2 inhibitor
Prasit, P, Wang, Z, Brideau, C, Chan, C.-C, Charleson, S, Cromlish, W, Ethier, D, Evans, J.F, Ford-Hutchinson, A.W, Gauthier, J.Y, Gordon, R, Guay, J, Gresser, M, Kargman, S, Kennedy, B, Leblanc, Y, Léger, S, Mancini, J, O'Neill, G.P, Ouellet, M, Percival, M.D, Perrier, H, Riendeau, D, Rodger, I, Tagari, P, Thérien, M, Vickers, P, Wong, E, Xu, L.-J, Young, R.N, Zamboni, R, Boyce, S, Rupniak, N, Forrest, M, Visco, D, Patrick, D
Published in Bioorganic & medicinal chemistry letters (05.07.1999)
Published in Bioorganic & medicinal chemistry letters (05.07.1999)
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From indomethacin to a selective COX-2 inhibitor: Development of indolalkanoic acids as potent and selective cyclooxygenase-2 inhibitors
Black, W.C., Bayly, C., Belley, M., Chan, C.-C., Charleson, S., Denis, D., Gauthier, J.Y., Gordon, R., Guay, D., Kargman, S., Lau, C.K., Leblanc, Y., Mancini, J., Ouellet, M., Percival, D., Roy, P., Skorey, K., Tagari, P., Vickers, P., Wong, E., Xu, L., Prasit, P.
Published in Bioorganic & medicinal chemistry letters (19.03.1996)
Published in Bioorganic & medicinal chemistry letters (19.03.1996)
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Synthesis and biological evaluation of both enantiomers of L-761,000 as inhibitors of cyclooxygenase 1 and 2
Leblanc, Y., Black, W.C., Chan, C.C., Charleson, S., Delorme, D., Denis, D., Gauthier, J.Y., Grimm, E.L., Gordon, R., Guay, D., Hamel, P., Kargman, S., Lau, C.K., Mancini, J., Ouellet, M., Percival, D., Roy, P., Skorey, K., Tagari, P., Vickers, P., Wong, E., Xu, L., Prasit, P.
Published in Bioorganic & medicinal chemistry letters (19.03.1996)
Published in Bioorganic & medicinal chemistry letters (19.03.1996)
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Neural plasticity of basal forebrain cholinergic neurons: effects of gangliosides
Stephens, P H, Tagari, P C, Garofalo, L, Maysinger, D, Piotte, M, Cuello, A C
Published in Neuroscience letters (11.09.1987)
Published in Neuroscience letters (11.09.1987)
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Substituted coumarins as potent 5-lipoxygenase inhibitors
Grimm, Erich L., Brideau, Christine, Chauret, Nathalie, Chan, Chi-Chung, Delorme, Daniel, Ducharme, Yves, Ethier, Diane, Falgueyret, Jean-Pierre, Friesen, Richard W., Guay, Jocelyne, Hamel, Pierre, Riendeau, Denis, Soucy-Breau, Chantal, Tagari, Philip, Girard, Yves
Published in Bioorganic & medicinal chemistry letters (01.05.2006)
Published in Bioorganic & medicinal chemistry letters (01.05.2006)
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Effects of COX-2 inhibitors on aortic prostacyclin production in cholesterol-fed rabbits
Wong, Elizabeth, Huang, JingQi, Tagari, Philip, Riendeau, Denis
Published in Atherosclerosis (01.08.2001)
Published in Atherosclerosis (01.08.2001)
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Quinolines as potent 5-lipoxygenase inhibitors: Synthesis and biological profile of L-746,530
Dubé, Daniel, Blouin, Marc, Brideau, Christine, Chan, Chi-Chung, Desmarais, Sylvie, Ethier, Diane, Falgueyret, Jean-Pierre, Friesen, Richard W., Girard, Mario, Girard, Yves, Guay, Jocelyne, Riendeau, Denis, Tagari, Philip, Young, Robert N.
Published in Bioorganic & medicinal chemistry letters (19.05.1998)
Published in Bioorganic & medicinal chemistry letters (19.05.1998)
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Mechanism of selective inhibition of human prostaglandin G/H synthase-1 and -2 in intact cells
Kargman, Stacia, Wong, Elizabeth, Greig, Gillian M., Falgueyret, Jean-Pierre, Cromlish, Wanda, Ethier, Diane, Yergey, Jim A., Riendeau, Denis, Evans, Jilly F., Kennedy, Brian, Tagari, Philip, Francis, Donna A., O'Neill, Gary P.
Published in Biochemical pharmacology (11.10.1996)
Published in Biochemical pharmacology (11.10.1996)
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Leukotriene D4 and the cerebral vasculature in vivo and in vitro
Tagari, P, Du Boulay, G H, Aitken, V, Boullin, D J
Published in Prostaglandins leukotrienes and medicine (01.07.1983)
Published in Prostaglandins leukotrienes and medicine (01.07.1983)
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Leukotriene D receptor blockade inhibits the immediate and late bronchoconstrictor responses to inhaled antigen in patients with asthma
RASMUSSEN, J, ERIKSSON, L, MARGOLSKEE, D, TAGARI, P, WILLIAMS, V, ANDERSSON, K
Published in Journal of allergy and clinical immunology (01.08.1992)
Published in Journal of allergy and clinical immunology (01.08.1992)
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BIO-fully automated sample treatment high-performance liquid chromatography and radioimmunoassay for leukotriene E4 in human urine from asthmatics
NICOLL-GRIFFITH, D, ZAMBONI, R, RASMUSSEN, J. B, ETHIER, D, CHARLESON, S, TAGARI, P
Published in Journal of chromatography (06.04.1990)
Published in Journal of chromatography (06.04.1990)
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(4-Piperidinylphenyl)aminoethyl amides as a novel class of non-covalent cathepsin K inhibitors
Kim, Tae-Seong, Hague, Andrew B., Lee, Tony I., Lian, Brian, Tegley, Christopher M., Wang, Xianghong, Burgess, Teresa L., Qian, Yi-Xin, Ross, Sandra, Tagari, Philip, Lin, Chi-Hwei, Mayeda, Carol, Dao, Jennifer, Jordan, Steven, Mohr, Christopher, Cheetham, Janet, Viswanadhan, Vellarkad, Tasker, Andrew S.
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
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Leukotriene D4 receptor blockade inhibits the immediate and late bronchoconstrictor responses to inhaled antigen in patients with asthma
RASMUSSEN, J. B, ERIKSSON, L.-O, MARGOLSKEE, D. J, TAGARI, P, WILLIAMS, V. C, ANDERSSON, K.-E
Published in Journal of allergy and clinical immunology (01.08.1992)
Published in Journal of allergy and clinical immunology (01.08.1992)
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Synthesis and biological evaluation of 2,3-diarylthiophenes as selective Cox-2 and Cox-1 inhibitors
Leblanc, Yves, Gauthier, JacquesYves, Ethier, Diane, Guay, Jocelyne, Mancini, Joseph, Riendeau, Denis, Tagari, Philip, Vickers, Philip, Wong, Elizabeth, Prasit, Petpiboon
Published in Bioorganic & medicinal chemistry letters (21.09.1995)
Published in Bioorganic & medicinal chemistry letters (21.09.1995)
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