Epsilon substituted lysinol derivatives as HIV-1 protease inhibitors
Jones, Kristen L.G., Holloway, M. Katharine, Su, Hua-Poo, Carroll, Steven S., Burlein, Christine, Touch, Sinoeun, DiStefano, Daniel J., Sanchez, Rosa I., Williams, Theresa M., Vacca, Joseph P., Coburn, Craig A.
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
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Discovery of aminoheterocycles as a novel β-secretase inhibitor class: pH dependence on binding activity part 1
Stachel, Shawn J., Coburn, Craig A., Rush, Diane, Jones, Kristen L.G., Zhu, Hong, Rajapakse, Hemaka, Graham, Samuel L., Simon, Adam, Katharine Holloway, M., Allison, Tim J., Munshi, Sanjeev K., Espeseth, Amy S., Zuck, Paul, Colussi, Dennis, Wolfe, Abigail, Pietrak, Beth L., Lai, Ming-Tain, Vacca, Joseph P.
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
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Discovery of selective, orally bioavailable, N-linked arylsulfonamide Na(v)1.7 inhibitors with pain efficacy in mice
Roecker, Anthony J., Egbertson, Melissa, Jones, Kristen L. G., Gomez, Robert, Kraus, Richard L., Li, Yuxing, Koser, Amy Jo, Urban, Mark O., Klein, Rebecca, Clements, Michelle, Panigel, Jacqueline, Daley, Christopher, Wang, Jixin, Finger, Eleftheria N., Majercak, John, Santarelli, Vincent, Gregan, Irene, Cato, Matthew, Filzen, Tracey, Jovanovska, Aneta, Wang, Ying-Hong, Wang, Deping, Joyce, Leo A., Sherer, Edward C., Peng, Xuanjia, Wang, Xiu, Sun, Haiyan, Coleman, Paul J., Houghton, Andrea K., Layton, Mark E.
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
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Discovery of selective, orally bioavailable, N-linked arylsulfonamide Nav1.7 inhibitors with pain efficacy in mice
Roecker, Anthony J., Egbertson, Melissa, Jones, Kristen L.G., Gomez, Robert, Kraus, Richard L., Li, Yuxing, Koser, Amy Jo, Urban, Mark O., Klein, Rebecca, Clements, Michelle, Panigel, Jacqueline, Daley, Christopher, Wang, Jixin, Finger, Eleftheria N., Majercak, John, Santarelli, Vincent, Gregan, Irene, Cato, Matthew, Filzen, Tracey, Jovanovska, Aneta, Wang, Ying-Hong, Wang, Deping, Joyce, Leo A., Sherer, Edward C., Peng, Xuanjia, Wang, Xiu, Sun, Haiyan, Coleman, Paul J., Houghton, Andrea K., Layton, Mark E.
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
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Journal Article
Discovery of selective, orally bioavailable, N-linked arylsulfonamide Na v 1.7 inhibitors with pain efficacy in mice
Roecker, Anthony J, Egbertson, Melissa, Jones, Kristen L G, Gomez, Robert, Kraus, Richard L, Li, Yuxing, Koser, Amy Jo, Urban, Mark O, Klein, Rebecca, Clements, Michelle, Panigel, Jacqueline, Daley, Christopher, Wang, Jixin, Finger, Eleftheria N, Majercak, John, Santarelli, Vincent, Gregan, Irene, Cato, Matthew, Filzen, Tracey, Jovanovska, Aneta, Wang, Ying-Hong, Wang, Deping, Joyce, Leo A, Sherer, Edward C, Peng, Xuanjia, Wang, Xiu, Sun, Haiyan, Coleman, Paul J, Houghton, Andrea K, Layton, Mark E
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
Published in Bioorganic & medicinal chemistry letters (15.05.2017)
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Compounds that bind APP and inhibit Abeta processing in vitro suggest a novel approach to Alzheimer disease therapeutics
Espeseth, Amy S, Xu, Min, Huang, Qian, Coburn, Craig A, Jones, Kristen L G, Ferrer, Marc, Zuck, Paul D, Strulovici, Berta, Price, Eric A, Wu, Guoxin, Wolfe, Abigail L, Lineberger, Janet E, Sardana, Mohinder, Tugusheva, Katherine, Pietrak, Beth L, Crouthamel, Ming-Chih, Lai, Ming-Tain, Dodson, Elizabeth Chen, Bazzo, Renzo, Shi, Xiao-Ping, Simon, Adam J, Li, Yueming, Hazuda, Daria J
Published in The Journal of biological chemistry (06.05.2005)
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Published in The Journal of biological chemistry (06.05.2005)
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Compounds That Bind APP and Inhibit Aβ Processing in Vitro Suggest a Novel Approach to Alzheimer Disease Therapeutics
Espeseth, Amy S., Xu, Min, Huang, Qian, Coburn, Craig A., Jones, Kristen L.G., Ferrer, Marc, Zuck, Paul D., Strulovici, Berta, Price, Eric A., Wu, Guoxin, Wolfe, Abigail L., Lineberger, Janet E., Sardana, Mohinder, Tugusheva, Katherine, Pietrak, Beth L., Crouthamel, Ming-Chih, Lai, Ming-Tain, Dodson, Elizabeth Chen, Bazzo, Renzo, Shi, Xiao-Ping, Simon, Adam J., Li, Yueming, Hazuda, Daria J.
Published in The Journal of biological chemistry (06.05.2005)
Published in The Journal of biological chemistry (06.05.2005)
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