Selective androgen receptor modulators based on a series of 7H-[1,4]oxazino[3,2-g]quinolin-7-ones with improved in vivo activity
LONG, Yun Oliver, HIGUCHI, Robert I, KARANEWSKY, Donald S, LIN ZHI, CAFERRO, Thomas R, LAU, Thomas L. S, MIN WU, CUMMINGS, Marquis L, MARTINBOROUGH, Esther A, MARSCHKE, Keith B, CHANG, William Y, LOPEZ, Francisco J
Published in Bioorganic & medicinal chemistry (01.05.2008)
Published in Bioorganic & medicinal chemistry (01.05.2008)
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5 (Z) -Benzylidene -1,2 -dihydro -9 -hydroxy -10 -methoxy -2,2, 4 -trimethyl -5H-1 -aza -6 -oxa -chrysenes as non-steroidal glucocorticoid receptor modulators
ARDECKY, Robert J, HUDSON, Andrew R, LOPEZ, Francisco J, MARSCHKE, Keith B, MINER, Jeffrey N, KARANEWSKY, Donald S, NEGRO-VILAR, Andrés, LIN ZHI, PHILLIPS, Dean P, TYHONAS, John S, DECKHUT, Charlotte, LAU, Thomas L, YONGKAI LI, MARTINBOROUGH, Esther A, ROACH, Steven L, HIGUCHI, Robert I
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
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Inhibition of mast cell degranulation by novel small molecule MRGPRX2 antagonists
Wollam, Joshua, Solomon, Michelle, Villescaz, Christiane, Lanier, Marion, Evans, Samantha, Bacon, Corinne, Freeman, David, Vasquez, Alexis, Vest, Alan, Napora, Jim, Charlot, Brittney, Cavarlez, Christine, Kim, Andrew, Dvorak, Lisa, Selfridge, Brandon, Huang, Liming, Nevarez, Andres, Dedman, Harry, Brooks, Jennifer, Frischbutter, Stefan, Metz, Martin, Serhan, Nadine, Gaudenzio, Nicolas, Timony, Gregg, Martinborough, Esther, Boehm, Marcus F., Viswanath, Veena
Published in Journal of allergy and clinical immunology (01.10.2024)
Published in Journal of allergy and clinical immunology (01.10.2024)
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MRGPRX2 Antagonist EP262 Potently Inhibits Agonist-Induced Mast Cell Degranulation In Vitro and In Vivo
Wollam, Joshua, Solomon, Michelle, Villescaz, Christiane, Lanier, Marion, Brooks, Jennifer, Kim, Andrew, Anderson, Samantha, Freeman, David, Vasquez, Alexis, Pisacane, Corinne, Charlot, Brittney, Vest, Alan, Napora, Jim, Cavarlez, Christine, Dvorak, Lisa, Selfridge, Brandon, Huang, Liming, Sainz, Marcos, Nevarez, Andres, Dedman, Harry, Timony, Gregg, Martinborough, Esther, Viswanath, Veena, Boehm, Marcus
Published in Journal of allergy and clinical immunology (01.02.2023)
Published in Journal of allergy and clinical immunology (01.02.2023)
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Novel selective androgen receptor modulators: SAR studies on 6-bisalkylamino-2-quinolinones
van Oeveren, Arjan, Motamedi, Mehrnoush, Martinborough, Esther, Zhao, Shuo, Shen, Yixing, West, Sarah, Chang, William, Kallel, Adam, Marschke, Keith B., López, Francisco J., Negro-Vilar, Andrés, Zhi, Lin
Published in Bioorganic & medicinal chemistry letters (15.03.2007)
Published in Bioorganic & medicinal chemistry letters (15.03.2007)
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Journal Article
Selective androgen receptor modulators based on a series of 7 H-[1,4]oxazino[3,2- g]quinolin-7-ones with improved in vivo activity
Long, Yun Oliver, Higuchi, Robert I., Caferro, Thomas R., Lau, Thomas L.S., Wu, Min, Cummings, Marquis L., Martinborough, Esther A., Marschke, Keith B., Chang, William Y., López, Francisco J., Karanewsky, Donald S., Zhi, Lin
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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Journal Article
5( Z)-Benzylidene-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5 H-1-aza-6-oxa-chrysenes as non-steroidal glucocorticoid receptor modulators
Ardecky, Robert J., Hudson, Andrew R., Phillips, Dean P., Tyhonas, John S., Deckhut, Charlotte, Lau, Thomas L., Li, Yongkai, Martinborough, Esther A., Roach, Steven L., Higuchi, Robert I., Lopez, Francisco J., Marschke, Keith B., Miner, Jeffrey N., Karanewsky, Donald S., Negro-Vilar, Andrés, Zhi, Lin
Published in Bioorganic & medicinal chemistry letters (2007)
Published in Bioorganic & medicinal chemistry letters (2007)
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Journal Article