Synthesis of tripeptides as potent Yersinia protein tyrosine phosphatase inhibitors
Lee, Kyeong, Boovanahalli, Shanthaveerappa K., Nam, Ky-Youb, Kang, Sang-Uk, Lee, Mijeoung, Phan, Jason, Wu, Li, Waugh, David S., Zhang, Zhong-Yin, No, Kyoung Tai, Lee, Jung Jun, Burke, Terrence R.
Published in Bioorganic & medicinal chemistry letters (15.09.2005)
Published in Bioorganic & medicinal chemistry letters (15.09.2005)
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α-Methylated simplified resiniferatoxin (sRTX) thiourea analogues as potent and stereospecific TRPV1 antagonists
Kim, Ho Shin, Jin, Mi-Kyoung, Kang, Sang-Uk, Lim, Ju-Ok, Tran, Phuong-Thao, Hoang, Van-Hai, Ann, Jihyae, Ha, Tae-Hwan, Pearce, Larry V., Pavlyukovets, Vladimir A., Blumberg, Peter M., Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
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N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the A-region
Kim, Yong Soo, Kil, Min-Jung, Kang, Sang-Uk, Ryu, HyungChul, Kim, Myeong Seop, Cho, Yongsung, Bhondwe, Rahul S., Thorat, Shivaji A., Sun, Wei, Liu, Keliang, Lee, Jin Hee, Choi, Sun, Pearce, Larry V., Pavlyukovets, Vladimir A., Morgan, Matthew A., Tran, Richard, Lazar, Jozsef, Blumberg, Peter M., Lee, Jeewoo
Published in Bioorganic & medicinal chemistry (01.01.2012)
Published in Bioorganic & medicinal chemistry (01.01.2012)
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α-Substituted N-(4- tert-butylbenzyl)- N′-[4-(methylsulfonylamino)benzyl]thiourea analogues as potent and stereospecific TRPV1 antagonists
Chung, Jae-Uk, Kim, Su Yeon, Lim, Ju-Ok, Choi, Hyun-Kyung, Kang, Sang-Uk, Yoon, Hae-Seok, Ryu, HyungChul, Kang, Dong Wook, Lee, Jeewoo, Kang, Bomi, Choi, Sun, Toth, Attila, Pearce, Larry V., Pavlyukovets, Vladimir A., Lundberg, Daniel J., Blumberg, Peter M.
Published in Bioorganic & medicinal chemistry (15.09.2007)
Published in Bioorganic & medicinal chemistry (15.09.2007)
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Methionyl adenylate analogues as inhibitors of methionyl-tRNA synthetase
Lee, Jeewoo, Kang, Sang Uk, Kang, Mee Kyoung, Chun, Moon Woo, Jo, Yeong Joon, Kkwak, Jin Hwan, Kim, Sunghoon
Published in Bioorganic & medicinal chemistry letters (17.05.1999)
Published in Bioorganic & medicinal chemistry letters (17.05.1999)
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Synthesis of α,α-disubstituted 4-phosphonophenylalanine analogues as conformationally-constrained phosphotyrosyl mimetics
Oishi, Shinya, Kang, Sang-Uk, Liu, Hongpeng, Zhang, Manchao, Yang, Dajun, Deschamps, Jeffrey R., Burke, Terrence R.
Published in Tetrahedron (22.03.2004)
Published in Tetrahedron (22.03.2004)
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N-[4-(methylsulfonylamino)benzyl]thiourea analogues as vanilloid receptor antagonists : Analysis of structure-activity relationships for the 'C-region'
JEEWOO LEE, KANG, Sang-Uk, BLUMBERG, Peter M, LIM, Ju-Ok, CHOI, Hyun-Kyung, JIN, Mi-Kyung, TOTH, Attila, PEARCE, Larry V, TRAN, Richard, YUN WANG, SZABO, Tamas
Published in Bioorganic & medicinal chemistry (15.01.2004)
Published in Bioorganic & medicinal chemistry (15.01.2004)
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N-4-Substituted-benzyl- N′- tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activity
Park, Hyeung-geun, Choi, Ji-yeon, Choi, Sea-hoon, Park, Mi-kyung, Lee, Jihye, Suh, Young-ger, Cho, Hawon, Oh, Uhtaek, Lee, Jiyoun, Kang, Sang-Uk, Lee, Jeewoo, Kim, Hee-Doo, Park, Young-Ho, Su Jeong, Yeon, Kyu Choi, Jin, Jew, Sang-sup
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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Analysis of structure–activity relationships for the ‘A-region’ of N-(4- t-butylbenzyl)- N′-[4-(methylsulfonylamino)benzyl]thiourea analogues as TRPV1 antagonists
Lee, Jeewoo, Kang, Sang-Uk, Kil, Min-Jung, Shin, Myoungyoup, Lim, Ju-Ok, Choi, Hyun-Kyung, Jin, Mi-Kyoung, Kim, Su Yeon, Kim, Sung-Eun, Lee, Yong-Sil, Min, Kyung-Hoon, Kim, Young-Ho, Ha, Hee-Jin, Tran, Richard, Welter, Jacqueline D., Wang, Yun, Szabo, Tamas, Pearce, Larry V., Lundberg, Daniel J., Toth, Attila, Pavlyukovets, Vladimir A., Morgan, Matthew A., Blumberg, Peter M.
Published in Bioorganic & medicinal chemistry letters (15.09.2005)
Published in Bioorganic & medicinal chemistry letters (15.09.2005)
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Analysis of structure–activity relationships for the ‘B-region’ of N-(4- t-butylbenzyl)- N′-[4-(methylsulfonylamino)benzyl]-thiourea analogues as TRPV1 antagonists
Lee, Jeewoo, Jin, Mi-Kyoung, Kang, Sang-Uk, Kim, Su Yeon, Lee, Jiyoun, Shin, Myoungyoup, Hwang, Jaemin, Cho, Sookhyun, Choi, Yeon-Sil, Choi, Hyun-Kyung, Kim, Sung-Eun, Suh, Young-Ger, Lee, Yong-Sil, Kim, Young-Ho, Ha, Hee-Jin, Toth, Attila, Pearce, Larry V., Tran, Richard, Szabo, Tamas, Welter, Jacqueline D., Lundberg, Daniel J., Wang, Yun, Lazar, Jozsef, Pavlyukovets, Vladimir A., Morgan, Matthew A., Blumberg, Peter M.
Published in Bioorganic & medicinal chemistry letters (15.09.2005)
Published in Bioorganic & medicinal chemistry letters (15.09.2005)
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Different vanilloid agonists cause different patterns of calcium response in CHO cells heterologously expressing rat TRPV1
Tóth, Attila, Wang, Yun, Kedei, Noémi, Tran, Richard, Pearce, Larry V., Kang, Sang-Uk, Jin, Mi-Kyung, Choi, Hyun-Kyung, Lee, Jeewoo, Blumberg, Peter M.
Published in Life sciences (1973) (06.05.2005)
Published in Life sciences (1973) (06.05.2005)
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Structure-activity relationships of simplified resiniferatoxin analogues with potent VR1 agonism elucidates an active conformation of RTX for VR1 binding
LEE, Jeewoo, SU YEON KIM, WELTER, Jacqueline D, SZABO, Tamas, TRAN, Richard, PEARCE, Larry V, TOTH, Attila, BLUMBERG, Peter M, PARK, Soyoung, LIM, Ju-Ok, KIM, Ji-Min, KANG, Myungshim, LEE, Jiyoun, KANG, Sang-Uk, CHOI, Hyun-Kyung, JIN, Mi-Kyung
Published in Bioorganic & medicinal chemistry (01.03.2004)
Published in Bioorganic & medicinal chemistry (01.03.2004)
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Analysis of structure-activity relationships for the 'b-region' of N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)-benzyl]thiourea analogues as vanilloid receptor antagonists: discovery of an N-hydroxythiourea analogue with potent analgesic activity
LEE, Jeewoo, KANG, Sang-Uk, HA, Hee-Jin, KIM, Young-Ho, PEARCE, Larry V, TRAN, Richard, LUNDBERG, Daniel J, YUN WANG, TOTH, Attila, BLUMBERG, Peter M, CHOI, Hyun-Kyung, LEE, Jiyoun, LIM, Ju-Ok, KIL, Min-Jung, JIN, Mi-Kyung, KIM, Kang-Pil, SUNG, Jong-Hyuk, CHUNG, Suk-Jae
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Journal Article
N-Alkoxysulfamide, N-hydroxysulfamide, and sulfamate analogues of methionyl and isoleucyl adenylates as inhibitors of methionyl-tRNA and isoleucyl-tRNA synthetases
Lee, Jeewoo, Kim, Sung Eun, Lee, Ji Young, Kim, Su Yeon, Kang, Sang Uk, Seo, Seung Hwan, Chun, Moon Woo, Kang, Taehee, Choi, Soo Young, Kim, Hea Ok
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
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Ester and hydroxamate analogues of methionyl and isoleucyl adenylates as inhibitors of methionyl-tRNA and isoleucyl-tRNA synthetases
Lee, Jeewoo, Kang, Sang Uk, Kim, Su Yeon, Kim, Sung Eun, Kang, Mee Kyoung, Jo, Yeong Joon, Kim, Sunghoon
Published in Bioorganic & medicinal chemistry letters (23.04.2001)
Published in Bioorganic & medicinal chemistry letters (23.04.2001)
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