Chemogenetics revealed: DREADD occupancy and activation via converted clozapine
Gomez, Juan L., Bonaventura, Jordi, Lesniak, Wojciech, Mathews, William B., Sysa-Shah, Polina, Rodriguez, Lionel A., Ellis, Randall J., Richie, Christopher T., Harvey, Brandon K., Dannals, Robert F., Pomper, Martin G., Bonci, Antonello, Michaelides, Michael
Published in Science (American Association for the Advancement of Science) (04.08.2017)
Published in Science (American Association for the Advancement of Science) (04.08.2017)
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Journal Article
The Histone Methyltransferase Inhibitor A-366 Uncovers a Role for G9a/GLP in the Epigenetics of Leukemia
Pappano, William N, Guo, Jun, He, Yupeng, Ferguson, Debra, Jagadeeswaran, Sujatha, Osterling, Donald J, Gao, Wenqing, Spence, Julie K, Pliushchev, Marina, Sweis, Ramzi F, Buchanan, Fritz G, Michaelides, Michael R, Shoemaker, Alexander R, Tse, Chris, Chiang, Gary G
Published in PloS one (06.07.2015)
Published in PloS one (06.07.2015)
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Journal Article
Pharmacological and behavioral divergence of ketamine enantiomers: implications for abuse liability
Bonaventura, Jordi, Lam, Sherry, Carlton, Meghan, Boehm, Matthew A., Gomez, Juan L., Solís, Oscar, Sánchez-Soto, Marta, Morris, Patrick J., Fredriksson, Ida, Thomas, Craig J., Sibley, David R., Shaham, Yavin, Zarate, Carlos A., Michaelides, Michael
Published in Molecular psychiatry (01.11.2021)
Published in Molecular psychiatry (01.11.2021)
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Journal Article
Ultrapotent chemogenetics for research and potential clinical applications
Magnus, Christopher J, Lee, Peter H, Bonaventura, Jordi, Zemla, Roland, Gomez, Juan L, Ramirez, Melissa H, Hu, Xing, Galvan, Adriana, Basu, Jayeeta, Michaelides, Michael, Sternson, Scott M
Published in Science (American Association for the Advancement of Science) (12.04.2019)
Published in Science (American Association for the Advancement of Science) (12.04.2019)
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Journal Article
High-potency ligands for DREADD imaging and activation in rodents and monkeys
Bonaventura, Jordi, Eldridge, Mark A. G., Hu, Feng, Gomez, Juan L., Sanchez-Soto, Marta, Abramyan, Ara M., Lam, Sherry, Boehm, Matthew A., Ruiz, Christina, Farrell, Mitchell R., Moreno, Andrea, Galal Faress, Islam Mustafa, Andersen, Niels, Lin, John Y., Moaddel, Ruin, Morris, Patrick J., Shi, Lei, Sibley, David R., Mahler, Stephen V., Nabavi, Sadegh, Pomper, Martin G., Bonci, Antonello, Horti, Andrew G., Richmond, Barry J., Michaelides, Michael
Published in Nature communications (11.10.2019)
Published in Nature communications (11.10.2019)
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Journal Article
Progress towards a public chemogenomic set for protein kinases and a call for contributions
Drewry, David H, Wells, Carrow I, Andrews, David M, Angell, Richard, Al-Ali, Hassan, Axtman, Alison D, Capuzzi, Stephen J, Elkins, Jonathan M, Ettmayer, Peter, Frederiksen, Mathias, Gileadi, Opher, Gray, Nathanael, Hooper, Alice, Knapp, Stefan, Laufer, Stefan, Luecking, Ulrich, Michaelides, Michael, Müller, Susanne, Muratov, Eugene, Denny, R Aldrin, Saikatendu, Kumar S, Treiber, Daniel K, Zuercher, William J, Willson, Timothy M
Published in PloS one (02.08.2017)
Published in PloS one (02.08.2017)
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Journal Article
Elucidation of The Behavioral Program and Neuronal Network Encoded by Dorsal Raphe Serotonergic Neurons
Urban, Daniel J, Zhu, Hu, Marcinkiewcz, Catherine A, Michaelides, Michael, Oshibuchi, Hidehiro, Rhea, Darren, Aryal, Dipendra K, Farrell, Martilias S, Lowery-Gionta, Emily, Olsen, Reid H J, Wetsel, William C, Kash, Thomas L, Hurd, Yasmin L, Tecott, Laurence H, Roth, Bryan L
Published in Neuropsychopharmacology (New York, N.Y.) (01.04.2016)
Published in Neuropsychopharmacology (New York, N.Y.) (01.04.2016)
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Journal Article
Target deconvolution studies of (2R,6R)-hydroxynorketamine: an elusive search
Bonaventura, Jordi, Gomez, Juan L., Carlton, Meghan L., Lam, Sherry, Sanchez-Soto, Marta, Morris, Patrick J., Moaddel, Ruin, Kang, Hye Jin, Zanos, Panos, Gould, Todd D., Thomas, Craig J., Sibley, David R., Zarate, Carlos A., Michaelides, Michael
Published in Molecular psychiatry (01.10.2022)
Published in Molecular psychiatry (01.10.2022)
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Journal Article
The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification
Wells, Carrow I, Al-Ali, Hassan, Andrews, David M, Asquith, Christopher R M, Axtman, Alison D, Dikic, Ivan, Ebner, Daniel, Ettmayer, Peter, Fischer, Christian, Frederiksen, Mathias, Futrell, Robert E, Gray, Nathanael S, Hatch, Stephanie B, Knapp, Stefan, Lücking, Ulrich, Michaelides, Michael, Mills, Caitlin E, Müller, Susanne, Owen, Dafydd, Picado, Alfredo, Saikatendu, Kumar S, Schröder, Martin, Stolz, Alexandra, Tellechea, Mariana, Turunen, Brandon J, Vilar, Santiago, Wang, Jinhua, Zuercher, William J, Willson, Timothy M, Drewry, David H
Published in International journal of molecular sciences (08.01.2021)
Published in International journal of molecular sciences (08.01.2021)
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Journal Article
Discovery and Development of Potent and Selective Inhibitors of Histone Methyltransferase G9a
Sweis, Ramzi F, Pliushchev, Marina, Brown, Peter J, Guo, Jun, Li, Fengling, Maag, David, Petros, Andrew M, Soni, Nirupama B, Tse, Chris, Vedadi, Masoud, Michaelides, Michael R, Chiang, Gary G, Pappano, William N
Published in ACS medicinal chemistry letters (13.02.2014)
Published in ACS medicinal chemistry letters (13.02.2014)
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Journal Article
A non-canonical striatopallidal Go pathway that supports motor control
Labouesse, Marie A., Torres-Herraez, Arturo, Chohan, Muhammad O., Villarin, Joseph M., Greenwald, Julia, Sun, Xiaoxiao, Zahran, Mysarah, Tang, Alice, Lam, Sherry, Veenstra-VanderWeele, Jeremy, Lacefield, Clay O., Bonaventura, Jordi, Michaelides, Michael, Chan, C. Savio, Yizhar, Ofer, Kellendonk, Christoph
Published in Nature communications (23.10.2023)
Published in Nature communications (23.10.2023)
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Journal Article
Motivational valence is determined by striatal melanocortin 4 receptors
Klawonn, Anna Mathia, Fritz, Michael, Nilsson, Anna, Bonaventura, Jordi, Shionoya, Kiseko, Mirrasekhian, Elahe, Karlsson, Urban, Jaarola, Maarit, Granseth, Björn, Blomqvist, Anders, Michaelides, Michael, Engblom, David
Published in The Journal of clinical investigation (01.07.2018)
Published in The Journal of clinical investigation (01.07.2018)
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Journal Article
Synthesis and preclinical evaluation of [11C]uPSEM792 for PSAM4-GlyR based chemogenetics
Nerella, Sridhar Goud, Telu, Sanjay, Liow, Jeih-San, Jenkins, Madeline D., Zoghbi, Sami S., Gomez, Juan L., Michaelides, Michael, Eldridge, Mark A. G., Richmond, Barry J., Innis, Robert B., Pike, Victor W.
Published in Scientific reports (22.01.2024)
Published in Scientific reports (22.01.2024)
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Journal Article
Whole-brain circuit dissection in free-moving animals reveals cell-specific mesocorticolimbic networks
Michaelides, Michael, Anderson, Sarah Ann R, Ananth, Mala, Smirnov, Denis, Thanos, Panayotis K, Neumaier, John F, Wang, Gene-Jack, Volkow, Nora D, Hurd, Yasmin L
Published in The Journal of clinical investigation (01.12.2013)
Published in The Journal of clinical investigation (01.12.2013)
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Journal Article
Discovery of Spiro Oxazolidinediones as Selective, Orally Bioavailable Inhibitors of p300/CBP Histone Acetyltransferases
Michaelides, Michael R, Kluge, Arthur, Patane, Michael, Van Drie, John H, Wang, Ce, Hansen, T. Matthew, Risi, Roberto M, Mantei, Robert, Hertel, Carmen, Karukurichi, Kannan, Nesterov, Alexandre, McElligott, David, de Vries, Peter, Langston, J. William, Cole, Philip A, Marmorstein, Ronen, Liu, Hong, Lasko, Loren, Bromberg, Kenneth D, Lai, Albert, Kesicki, Edward A
Published in ACS medicinal chemistry letters (11.01.2018)
Published in ACS medicinal chemistry letters (11.01.2018)
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Journal Article
Discovery of a Potent and Selective Covalent p300/CBP Inhibitor
Mastracchio, Anthony, Lai, Chunqiu, Digiammarino, Enrico, Ready, Damien B, Lasko, Loren M, Bromberg, Kenneth D, McClellan, William J, Montgomery, Debra, Manaves, Vlasios, Shaw, Bailin, Algire, Mikkel, Patterson, Melanie J, Sun, Chaohong C, Rosenberg, Saul, Lai, Albert, Michaelides, Michael R
Published in ACS medicinal chemistry letters (13.05.2021)
Published in ACS medicinal chemistry letters (13.05.2021)
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Journal Article
Interactions of calmodulin kinase II with the dopamine transporter facilitate cocaine-induced enhancement of evoked dopamine release
Keighron, Jacqueline D., Bonaventura, Jordi, Li, Yang, Yang, Jae-Won, DeMarco, Emily M., Hersey, Melinda, Cao, Jianjing, Sandtner, Walter, Michaelides, Michael, Sitte, Harald H., Newman, Amy Hauck, Tanda, Gianluigi
Published in Translational psychiatry (13.06.2023)
Published in Translational psychiatry (13.06.2023)
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