Discovery of an inhibitor of the production of the Pseudomonas aeruginosa virulence factor pyocyanin in wild-type cells
Morkunas, Bernardas, Gal, Balint, Galloway, Warren R J D, Hodgkinson, James T, Ibbeson, Brett M, Tan, Yaw Sing, Welch, Martin, Spring, David R
Published in Beilstein journal of organic chemistry (11.07.2016)
Published in Beilstein journal of organic chemistry (11.07.2016)
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Journal Article
Decreased GLUT2 and glucose uptake contribute to insulin secretion defects in MODY3/HNF1A hiPSC-derived mutant β cells
Low, Blaise Su Jun, Lim, Chang Siang, Ding, Shirley Suet Lee, Tan, Yaw Sing, Ng, Natasha Hui Jin, Krishnan, Vidhya Gomathi, Ang, Su Fen, Neo, Claire Wen Ying, Verma, Chandra S., Hoon, Shawn, Lim, Su Chi, Tai, E. Shyong, Teo, Adrian Kee Keong
Published in Nature communications (25.05.2021)
Published in Nature communications (25.05.2021)
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Journal Article
HNF4A and HNF1A exhibit tissue specific target gene regulation in pancreatic beta cells and hepatocytes
Ng, Natasha Hui Jin, Ghosh, Soumita, Bok, Chek Mei, Ching, Carmen, Low, Blaise Su Jun, Chen, Juin Ting, Lim, Euodia, Miserendino, María Clara, Tan, Yaw Sing, Hoon, Shawn, Teo, Adrian Kee Keong
Published in Nature communications (22.06.2024)
Published in Nature communications (22.06.2024)
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Journal Article
Transcriptional repression by a secondary DNA binding surface of DNA topoisomerase I safeguards against hypertranscription
Lau, Mei Sheng, Hu, Zhenhua, Zhao, Xiaodan, Tan, Yaw Sing, Liu, Jinyue, Huang, Hua, Yeo, Clarisse Jingyi, Leong, Hwei Fen, Grinchuk, Oleg V., Chan, Justin Kaixuan, Yan, Jie, Tee, Wee-Wei
Published in Nature communications (13.10.2023)
Published in Nature communications (13.10.2023)
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Journal Article
The Eyes Absent family members EYA4 and EYA1 promote PLK1 activation and successful mitosis through tyrosine dephosphorylation
Nelson, Christopher B., Rogers, Samuel, Roychoudhury, Kaushik, Tan, Yaw Sing, Atkinson, Caroline J., Sobinoff, Alexander P., Tomlinson, Christopher G., Hsu, Anton, Lu, Robert, Dray, Eloise, Haber, Michelle, Fletcher, Jamie I., Cesare, Anthony J., Hegde, Rashmi S., Pickett, Hilda A.
Published in Nature communications (15.02.2024)
Published in Nature communications (15.02.2024)
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Journal Article
Incorporation of Putative Helix-Breaking Amino Acids in the Design of Novel Stapled Peptides: Exploring Biophysical and Cellular Permeability Properties
Partridge, Anthony W, Kaan, Hung Yi Kristal, Juang, Yu-Chi, Sadruddin, Ahmad, Lim, Shuhui, Brown, Christopher J, Ng, Simon, Thean, Dawn, Ferrer, Fernando, Johannes, Charles, Yuen, Tsz Ying, Kannan, Srinivasaraghavan, Aronica, Pietro, Tan, Yaw Sing, Pradhan, Mohan R, Verma, Chandra S, Hochman, Jerome, Chen, Shiying, Wan, Hui, Ha, Sookhee, Sherborne, Brad, Lane, David P, Sawyer, Tomi K
Published in Molecules (Basel, Switzerland) (20.06.2019)
Published in Molecules (Basel, Switzerland) (20.06.2019)
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Journal Article
Stereoisomerism of stapled peptide inhibitors of the p53-Mdm2 interaction: an assessment of synthetic strategies and activity profiles
Yuen, Tsz Ying, Brown, Christopher J, Xue, Yuezhen, Tan, Yaw Sing, Ferrer Gago, Fernando J, Lee, Xue Er, Neo, Jin Yong, Thean, Dawn, Kaan, Hung Yi Kristal, Partridge, Anthony W, Verma, Chandra S, Lane, David P, Johannes, Charles W
Published in Chemical science (Cambridge) (14.07.2019)
Published in Chemical science (Cambridge) (14.07.2019)
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Journal Article
An Efficient, Short Stimulus PANC-1 Cancer Cell Ablation and Electrothermal Therapy Driven by Hydrophobic Interactions
Meivita, Maria P, Lee, Denise, Naikar, J Shamita, Go, Shao-Xiang, Teoh, Wey Chyi, Tan, Yaw Sing, Bajalovic, Natasa, Loke, Desmond K
Published in Pharmaceutics (28.12.2022)
Published in Pharmaceutics (28.12.2022)
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Journal Article
Anatomy of Mdm2 and Mdm4 in evolution
Tan, Ban Xiong, Liew, Hoe Peng, Chua, Joy S, Ghadessy, Farid J, Tan, Yaw Sing, Lane, David P, Coffill, Cynthia R
Published in Journal of molecular cell biology (01.02.2017)
Published in Journal of molecular cell biology (01.02.2017)
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Journal Article
Inhibiting S100B(ββ) for Activating Wild-Type p53: Design of Stapled Peptides
Kannan, Srinivasaraghavan, Aronica, Pietro G. A, Tan, Yaw Sing, Verma, Chandra S
Published in ACS omega (31.03.2019)
Published in ACS omega (31.03.2019)
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Journal Article
Efficient development of stable and highly functionalised peptides targeting the CK2α/CK2β protein-protein interaction
Iegre, Jessica, Brear, Paul, Baker, David J, Tan, Yaw Sing, Atkinson, Eleanor L, Sore, Hannah F, O' Donovan, Daniel H, Verma, Chandra S, Hyvönen, Marko, Spring, David R
Published in Chemical science (Cambridge) (21.05.2019)
Published in Chemical science (Cambridge) (21.05.2019)
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Journal Article
Diversity-oriented synthesis as a tool for identifying new modulators of mitosis
Ibbeson, Brett M., Laraia, Luca, Alza, Esther, O' Connor, Cornelius J., Tan, Yaw Sing, Davies, Huw M.L., McKenzie, Grahame, Venkitaraman, Ashok R., Spring, David R.
Published in Nature communications (01.01.2014)
Published in Nature communications (01.01.2014)
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Journal Article
Macrocyclization of an all-d linear alpha-helical peptide imparts cellular permeability
Kannan, Srinivasaraghavan, Aronica, Pietro G. A., Ng, Simon, Lian, Dawn Thean Gek, Frosi, Yuri, Chee, Sharon, Jiang, Shimin, Yuen, Tsz Ying, Sadruddin, Ahmad, Kaan, Hung Yi Kristal, Chandramohan, Arun, Wong, Jin Huei, Tan, Yaw Sing, Chang, Zi Wei, Ferrer-Gago, Fernando J., Arumugam, Prakash, Han, Yi, Chen, Shiying, Renia, Laurent, Brown, Christopher J., Johannes, Charles W., Henry, Brian, Lane, David P., Sawyer, Tomi K., Verma, Chandra S., Partridge, Anthony W.
Published in Chemical science (Cambridge) (07.06.2020)
Published in Chemical science (Cambridge) (07.06.2020)
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Journal Article
Kinetic and thermodynamic effects of phosphorylation on p53 binding to MDM2
Yadahalli, Shilpa, Neira, José L., Johnson, Christopher M., Tan, Yaw Sing, Rowling, Pamela J. E., Chattopadhyay, Anasuya, Verma, Chandra S., Itzhaki, Laura S.
Published in Scientific reports (24.01.2019)
Published in Scientific reports (24.01.2019)
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Journal Article
Stapled peptides as a new technology to investigate protein-protein interactions in human platelets
Iegre, Jessica, Ahmed, Niaz S., Gaynord, Josephine S., Wu, Yuteng, Herlihy, Kara M., Tan, Yaw Sing, Lopes-Pires, Maria E., Jha, Rupam, Lau, Yu Heng, Sore, Hannah F., Verma, Chandra, O'Donovan, Daniel H., Pugh, Nicholas, Spring, David R.
Published in Chemical science (Cambridge) (28.05.2018)
Published in Chemical science (Cambridge) (28.05.2018)
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Journal Article
Efficient development of stable and highly functionalised peptides targeting the CK2α/CK2β protein–protein interaction† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc00798a
Iegre, Jessica, Brear, Paul, Baker, David J., Tan, Yaw Sing, Atkinson, Eleanor L., Sore, Hannah F., O' Donovan, Daniel H., Verma, Chandra S., Hyvönen, Marko, Spring, David R.
Published in Chemical science (Cambridge) (12.04.2019)
Published in Chemical science (Cambridge) (12.04.2019)
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Journal Article
Discovery of a small-molecule binder of the oncoprotein gankyrin that modulates gankyrin activity in the cell
Chattopadhyay, Anasuya, O’Connor, Cornelius J., Zhang, Fengzhi, Galvagnion, Celine, Galloway, Warren R. J. D., Tan, Yaw Sing, Stokes, Jamie E., Rahman, Taufiq, Verma, Chandra, Spring, David R., Itzhaki, Laura S.
Published in Scientific reports (05.04.2016)
Published in Scientific reports (05.04.2016)
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Journal Article
Functional characterization of p53 pathway components in the ancient metazoan Trichoplax adhaerens
Siau, Jia Wei, Coffill, Cynthia R., Zhang, Weiyun Villien, Tan, Yaw Sing, Hundt, Juliane, Lane, David, Verma, Chandra, Ghadessy, Farid
Published in Scientific reports (28.09.2016)
Published in Scientific reports (28.09.2016)
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Journal Article
Stereoisomerism of stapled peptide inhibitors of the p53-Mdm2 interaction: an assessment of synthetic strategies and activity profiles† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc01456j
Yuen, Tsz Ying, Brown, Christopher J., Xue, Yuezhen, Tan, Yaw Sing, Ferrer Gago, Fernando J., Lee, Xue Er, Neo, Jin Yong, Thean, Dawn, Kaan, Hung Yi Kristal, Partridge, Anthony W., Verma, Chandra S., Lane, David P., Johannes, Charles W.
Published in Chemical science (Cambridge) (30.05.2019)
Published in Chemical science (Cambridge) (30.05.2019)
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