Advances in high‐throughput mass spectrometry in drug discovery
Dueñas, Maria Emilia, Peltier‐Heap, Rachel E, Leveridge, Melanie, Annan, Roland S, Büttner, Frank H, Trost, Matthias
Published in EMBO molecular medicine (11.01.2023)
Published in EMBO molecular medicine (11.01.2023)
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A high-throughput MALDI-TOF MS biochemical screen for small molecule inhibitors of the antigen aminopeptidase ERAP1
Müller, Leonie, Burton, Amy K, Tayler, Chloe L, Rowedder, James E, Hutchinson, Jonathan P, Peace, Simon, Quayle, Julie M, Leveridge, Melanie V, Annan, Roland S, Trost, Matthias, Peltier-Heap, Rachel E, Dueñas, Maria Emilia
Published in SLAS discovery (01.01.2023)
Published in SLAS discovery (01.01.2023)
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A direct-to-biology high-throughput chemistry approach to reactive fragment screening
Thomas, Ross P, Heap, Rachel E, Zappacosta, Francesca, Grant, Emma K, Pogány, Peter, Besley, Stephen, Fallon, David J, Hann, Michael M, House, David, Tomkinson, Nicholas C. O, Bush, Jacob T
Published in Chemical science (Cambridge) (22.09.2021)
Published in Chemical science (Cambridge) (22.09.2021)
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Identifying Inhibitors of Inflammation: A Novel High-Throughput MALDI-TOF Screening Assay for Salt-Inducible Kinases (SIKs)
Heap, Rachel E., Hope, Anthony G., Pearson, Lesley-Anne, Reyskens, Kathleen M. S. E., McElroy, Stuart P., Hastie, C. James, Porter, David W., Arthur, J. Simon C., Gray, David W., Trost, Matthias
Published in SLAS discovery (01.12.2017)
Published in SLAS discovery (01.12.2017)
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A chemoproteomic platform for selective deubiquitinase inhibitor discovery
Cookson, Rosa, Vuorinen, Aini, Pettinger, Jonathan, Kennedy, Cassandra R., Kirkpatrick, Joanna M., Peltier-Heap, Rachel E., Powell, Andrew, Snijders, Ambrosius P., Skehel, Mark, House, David, Rittinger, Katrin, Bush, Jacob T.
Published in Cell reports physical science (18.10.2023)
Published in Cell reports physical science (18.10.2023)
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